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ethyl 4-(3-{2-[(4-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}propanoyl)piperazine-1-carboxylate
1-(1-methyl-1H-pyrrole-2-carbonyl)-4-(pyridin-3-ylmethyl)-1,4-diazepane
4-{[1-(3,5-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]carbamoyl}pyridin-1-ium-1-olate
N-[3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propyl]-1H-1,2,3-triazole-5-carboxamide
4-[4-({[(5-chloro-1H-1,3-benzodiazol-2-yl)methyl](methyl)amino}methyl)phenyl]-2-methylbutan-2-ol
1-(2-methoxy-4-{[(2-methoxyethyl)amino]methyl}phenoxy)-3-(thiomorpholin-4-yl)propan-2-ol
5-methyl-1-(2-methylphenyl)-4-[3-(1H-pyrazol-1-yl)propanoyl]piperazin-2-one
(2-{2-[1-(3-fluoropyridin-4-yl)piperidin-3-yl]-1H-imidazol-1-yl}ethyl)dimethylamine
1-{5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}-4-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidine
4-methyl-5-[3-(1-methyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-2-phenylpyrimidine
6-[2-(2-methoxyphenyl)ethyl]-3-(propan-2-yl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl](methyl){[1-(propan-2-yl)-1H-imidazol-5-yl]methyl}amine
3-[1-(1-cyclopropylethyl)-1H-pyrazol-5-yl]-1-[2-(pyrrolidin-1-yl)ethyl]urea
N-methyl-2-[4-(1-methyl-1H-indol-2-yl)-1H-pyrazol-1-yl]acetamide
2-(2-methoxyethyl)-9-({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)-2,9-diazaspiro[5.5]undecan-3-one
N-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-3-(2-{[4-(methylsulfanyl)phenyl]methyl}-5-oxopyrrolidin-2-yl)propanamide
(3R,4R)-1-{[2-(difluoromethoxy)phenyl]methyl}-4-(4-hydroxypiperidin-1-yl)piperidin-3-ol
1-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}-4-(1H-1,2,3-triazol-4-ylmethyl)-1,4-diazepan-6-ol
6-(2-fluorophenyl)-N-[(3S,4S)-4-hydroxy-1-(propan-2-yl)pyrrolidin-3-yl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
ethyl 5-[(6-methylpyridin-2-yl)methyl]-1-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
N-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-1-methyl-3-propyl-1H-pyrazole-5-carboxamide
1-[(dimethyl-1,2-oxazol-4-yl)sulfonyl]-3-[2-(4-methoxyphenyl)ethyl]piperidine
1-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-3-(4-phenyl-1,2,3-thiadiazol-5-yl)urea
N-(2-hydroxyethyl)-3-{5-[2-(morpholin-4-yl)-2-oxoethyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
1-[(2S)-2-(hydroxymethyl)pyrrolidin-1-yl]-4-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}butan-1-one
2-(cyclopentylmethyl)-N-[2-(diethylamino)ethyl]-1,6-dimethyl-4-oxo-1,4-dihydropyridine-3-carboxamide
({1-[2-(4-fluorophenyl)ethyl]piperidin-4-yl}methyl)(methyl)[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]amine
(3-{2-[1-(2-methoxy-6-methylbenzoyl)piperidin-3-yl]-1H-imidazol-1-yl}propyl)dimethylamine
1-{4-[4-(3-hydroxyphenyl)piperazine-1-carbonyl]phenyl}imidazolidine-2,4-dione
3-[2-methyl-5-(2-oxopyrrolidin-1-yl)phenyl]-1-{2-[(3-methylpyridin-2-yl)amino]ethyl}urea
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)spiro[2.3]hexane-1-carboxamide
2-(dimethylamino)-1-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazin-1-yl}-2-(4-methylphenyl)ethan-1-one
2-(2,5-dimethoxyphenyl)-N-{[2-(3-hydroxypiperidin-1-yl)-8-methylquinolin-3-yl]methyl}-N-[(4-methoxyphenyl)methyl]acetamide
N-[3-(1H-imidazol-1-yl)propyl]-2-{3-oxo-1-[(2E)-3-phenylprop-2-en-1-yl]piperazin-2-yl}acetamide
2-methyl-4-{4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}quinoline
4-[(5-methyl-2-phenyl-1H-imidazol-4-yl)methyl]-1λ6-thiomorpholine-1,1-dione
methyl({[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl})[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]amine
N-methyl-N-(1H-pyrazol-5-ylmethyl)-2-{[1-(pyridine-3-carbonyl)piperidin-4-yl]oxy}benzamide
methyl (2S,4R)-4-(5-chloro-3-methyl-1H-indole-2-amido)-1-{[4-(methylsulfanyl)phenyl]methyl}pyrrolidine-2-carboxylate
3-{4-[3-(1H-imidazol-2-yl)piperidin-1-yl]-4-oxobutyl}-3,4-dihydroquinazolin-4-one
3-[4-(methylsulfanyl)benzoyl]-1-{[5-(propan-2-yl)-1H-pyrazol-3-yl]methyl}piperidine
{[4-(3-chlorophenyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}[(4-methoxy-2,3-dimethylphenyl)methyl]methylamine
5-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-2-yl}-2-(piperidin-1-yl)pyridine
3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)-N-[(2-methyl-1,3-thiazol-4-yl)methyl]propanamide
4-methoxy-3-{2-oxo-1-oxa-3,7-diazaspiro[4.5]decane-7-carbonyl}benzene-1-sulfonamide
2,2-bis(hydroxymethyl)-N-methyl-N-{2-[(4-methylphenyl)sulfanyl]ethyl}butanamide
methyl 2-[ethyl(2-methylprop-2-en-1-yl)sulfamoyl]-6-[(4-methoxy-3-methylphenyl)methyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
methyl 3-benzamido-5-{[(2E)-4-methylpent-2-en-1-yl]amino}-1-(oxolan-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-{2-[2-(4-fluorophenyl)azetidin-1-yl]-2-oxoethyl}-2-azaspiro[4.5]decan-3-one
2-({3-[4-(4-chlorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)-3-methoxyphenol