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2-(dimethylamino)-N-(2-hydroxyethyl)-2-(2-methylphenyl)-N-propylacetamide
2-{5-[(1R,2R)-2-phenylcyclopropanecarbonyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-1,3-benzodiazole
2-(4-{[3-(morpholin-4-yl)azetidin-1-yl]methyl}phenyl)-6-(pyridin-3-yl)-3,4-dihydropyrimidin-4-one
2-{1-[(2-fluorophenyl)methyl]-4-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl}ethan-1-ol
3,3-dimethyl-4-(morpholin-4-ylmethyl)-1-{[1,2,4]triazolo[1,5-a]pyrimidin-2-ylmethyl}piperidin-4-ol
{1-[5-methyl-1-(naphthalen-1-yl)-1H-pyrazol-4-yl]ethyl}[(5-methylthiophen-2-yl)methyl]amine
1-methyl-4-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}-2,3,4,5-tetrahydro-1H-1,4-benzodiazepine-2,5-dione
N4-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-6-methylpyrimidine-2,4-diamine
N-[1-(1-{[3-(2-hydroxyethoxy)phenyl]methyl}piperidin-4-yl)-2-phenylethyl]-N,1,3-trimethyl-1H-pyrazole-5-carboxamide
4-{4-[(5-methylthiophen-2-yl)methyl]piperazin-1-yl}-2-{[4-(trifluoromethyl)phenyl]methyl}-2,3-dihydro-1H-isoindole-1,3-dione
3-[3-(3-fluoro-4-methoxybenzoyl)piperidine-1-carbonyl]-2-methyl-4,5,6,7-tetrahydro-2H-indazole
4-(cyclopropylmethyl)-1-[2-(2-fluorophenyl)acetyl]-1,4-diazepan-5-one
N-{2-[(4-fluorophenyl)formamido]ethyl}-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
N-(butan-2-yl)-N-ethylquinoline-3-carboxamide
5-[3-(2-methoxyphenoxy)azetidine-1-carbonyl]-2-(methylsulfanyl)pyrimidine
4-(benzyloxy)-1-{imidazo[1,2-a]pyrimidine-2-carbonyl}piperidine
5-(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine-5-carbonyl)-2-methylpyrimidin-4-ol
2,6-difluoro-4-methoxy-N-(oxan-2-ylmethyl)benzamide
5-(2,5-dimethylphenoxymethyl)-N-[3-(2-methyl-1H-imidazol-1-yl)propyl]-1,2-oxazole-3-carboxamide
N-(oxan-4-yl)-2-{3-oxo-1-[(4-phenylphenyl)methyl]piperazin-2-yl}acetamide
4-[4,5-dimethyl-2-(1H-pyrrol-1-yl)thiophene-3-carbonyl]-2-(trifluoromethyl)morpholine
4-(1H-pyrazol-4-yl)-N-[2-(pyridin-3-ylformamido)ethyl]butanamide
3-[2-(2,2-dimethylpyrrolidin-1-yl)-2-oxoethyl]-N-(2-methoxyethyl)-4-methyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
5-[3-ethyl-4-(propan-2-yl)piperazine-1-carbonyl]-N-[2-(1H-imidazol-4-yl)ethyl]pyridin-2-amine
N-[2-methyl-5-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)phenyl]-4-(pyrazin-2-yl)piperazine-1-carboxamide
1-(4-methoxyphenyl)-5-[2-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-3-(propan-2-yl)-1H-1,2,4-triazole
3-ethyl-3-methyl-4-{[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperazin-2-one
1-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-3-{1-[(3-fluorophenyl)methyl]-1H-pyrazol-5-yl}urea
1-[(1-ethyl-1H-imidazol-2-yl)methyl]-2-(3-fluorophenyl)piperidine
N-[(5-methylpyrazin-2-yl)methyl]-1-(propan-2-yl)-1H-pyrazole-3-carboxamide
3-(3-methoxyphenyl)-5-(thian-4-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
1-{2-[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]ethyl}-5-(2-{[(4-methoxyphenyl)methyl]amino}ethyl)pyrrolidin-2-one
7-(2,3-dimethoxybenzoyl)-N,N,2-trimethyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
methyl (2R,4S)-4-hydroxy-1-{[2-(propylamino)pyrimidin-5-yl]methyl}piperidine-2-carboxylate
2-(cyclohex-1-en-1-yl)-1-{2-[(3-methoxyphenyl)methyl]morpholin-4-yl}ethan-1-one
N-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}-1-ethylpiperidine-4-carboxamide
N,4-dimethyl-N-[(3-methylthiophen-2-yl)methyl]-2-(propan-2-yl)pyrimidine-5-carboxamide
N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]-5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1,2-oxazole-3-carboxamide
1-[(2-methyl-1,3-thiazol-5-yl)methyl]-N-[3-(1H-1,2,3,4-tetrazol-1-yl)phenyl]piperidine-3-carboxamide
N-(1-{4-[(1S,4S)-2-azabicyclo[2.2.1]heptane-2-carbonyl]phenyl}-1H-pyrazol-4-yl)oxane-4-carboxamide
4-[4-hydroxy-4-(hydroxymethyl)piperidine-1-carbonyl]-N-propylbenzene-1-sulfonamide
N-phenyl-5-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
2-amino-7-[2,2-dimethyl-1-(thiophen-2-yl)cyclopropanecarbonyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-(2-methylphenyl)-4-(2-phenylbenzoyl)piperazin-2-one
3-[4-(2,3,4,5-tetrahydro-1-benzoxepine-4-carbonyl)piperazin-1-yl]-1,2-dihydropyrazin-2-one
[1-(1-methyl-1H-pyrazol-5-yl)propyl]({2-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)amine
N-methyl-2-(oxolan-2-ylmethoxy)-N-[(4-phenoxyphenyl)methyl]acetamide
N-(1-{1-[(4-acetamidophenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)acetamide
N-(6,6-dimethyl-1-phenyl-4,5,6,7-tetrahydro-1H-indazol-4-yl)-2-(3,4,5-trimethoxyphenyl)acetamide
3-{[5-(1-ethyl-1H-pyrazol-3-yl)-4-phenyl-1H-imidazol-1-yl]methyl}-2-(1H-1,2,4-triazol-1-yl)pyridine