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N-[(5-methylfuran-2-yl)methyl]-3-[1-(3-methylthiophene-2-carbonyl)piperidin-3-yl]propanamide
methyl 6-[3-(2-methoxybenzoyl)piperidin-1-yl]pyrazine-2-carboxylate
1-{2-oxo-2-[2-(pyrrolidine-1-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl]ethyl}azepan-2-one
1-(2-methylphenyl)-3-[1-(1-{[(4S)-4-(prop-1-en-2-yl)cyclohex-1-en-1-yl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]urea
(4aS,8aR)-1-(3-aminopropyl)-6-(2,1-benzoxazole-3-carbonyl)-decahydro-1,6-naphthyridin-2-one
N-({4-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-N-(oxolan-2-ylmethyl)pyridine-2-carboxamide
2-hydroxy-N,4-dimethyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}pentanamide
({3-methoxy-2-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)[2-methyl-1-(1-methyl-1H-imidazol-2-yl)propyl]amine
9-[(4-fluoro-3-methoxyphenyl)methyl]-2-(pyridin-3-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-{2-[(2-methyl-1,3-benzothiazol-6-yl)formamido]ethyl}pyridine-3-carboxamide
[1-(4-methyl-1H-imidazole-2-carbonyl)-4-propylpiperidin-4-yl]methanol
7-(5-methylthiophen-2-yl)-4-[2-(pyrrolidin-1-yl)ethyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-{1-[(2,3-difluoro-6-methoxyphenyl)methyl]piperidin-4-yl}methanesulfonamide
[2-(isoquinolin-1-yl)phenyl]methanol
N-(3-cyanophenyl)-2-[2-(2-oxopyrrolidin-1-yl)ethyl]piperidine-1-carboxamide
1-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-4-(pyridin-2-yl)piperidin-4-ol
(2S,4S)-4-amino-N,N-diethyl-1-(3-fluoropyridine-2-carbonyl)pyrrolidine-2-carboxamide
5-{4-[(4-fluorophenyl)methyl]-1,4-diazepane-1-carbonyl}-1,3-benzothiazole
N-{[1-(1,3-benzothiazole-6-carbonyl)piperidin-3-yl]methyl}thiophene-2-carboxamide
[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl](methyl)[1-(pyridin-2-yl)ethyl]amine
(1H-1,3-benzodiazol-2-ylmethyl)(methyl){[3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}amine
N-(2,1,3-benzoxadiazol-5-ylmethyl)-4-hydroxy-2-(1H-1,2,4-triazol-1-ylmethyl)pyrimidine-5-carboxamide
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
1-{[1-(2,4-difluorophenyl)-3-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}-3-(4-methyl-4H-1,2,4-triazol-3-yl)piperidine
[2-(2-ethoxypyridin-3-yl)phenyl]methanol
2-[(5-methylpyrazin-2-yl)methyl]-9-[2-oxo-2-(piperazin-1-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
3-[(4aR,7aS)-6,6-dioxo-4-(pyrrolidine-1-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]propanoic acid
5,7-dimethoxy-4-(2-phenylethyl)-1,2,3,4-tetrahydroquinolin-2-one
N-[1-(benzenesulfonyl)piperidin-4-yl]-1-methylazepane-2-carboxamide
2-{5-[4-(piperidine-1-carbonyl)pyridin-2-yl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl}ethan-1-ol
N-{[7-chloro-5-(2,5-dimethoxyphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(methylsulfanyl)acetamide
2-hydroxy-N-[(3R,4S)-4-(propan-2-yl)-1-[4-(trifluoromethyl)pyridin-2-yl]pyrrolidin-3-yl]acetamide
N,N-diethyl-2-(2,6,6-trimethyl-4-oxo-1-propyl-4,5,6,7-tetrahydro-1H-indol-3-yl)acetamide
1-[4-(4-fluorophenyl)-5-methylpyrimidin-2-yl]-N-methyl-N-(1-methylpiperidin-4-yl)-5-(thiophen-2-yl)-1H-pyrazole-4-carboxamide
(2R,3R,6R)-5-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
4-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]oxy}-N-(pyridin-2-ylmethyl)benzamide
2-{4-[(4-fluorophenyl)methyl]-1-(2-phenylethyl)piperazin-2-yl}ethan-1-ol
1-[(3-methylpyridin-2-yl)methyl]-4-(1-{[2-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carbonyl)piperazine
N-(1-{7-[(6-methylpyridin-2-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)cyclopropanecarboxamide
{[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)(quinolin-5-ylmethyl)amine
4'-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
2-(3-chloro-4-methoxyphenyl)-3-(piperidine-1-carbonyl)pyridine
N-cyclopropyl-4-methoxy-3-{[1-(3-phenylbutyl)piperidin-4-yl]oxy}benzamide
({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)[(5-methylthiophen-2-yl)methyl](prop-2-en-1-yl)amine
1-(2-chlorophenyl)-4-({8-methylimidazo[1,2-a]pyridin-2-yl}methyl)piperazin-2-one
(3aS,6aS)-N-[2-chloro-5-(trifluoromethyl)phenyl]-1-methyl-octahydropyrrolo[3,4-b]pyrrole-5-carboxamide
4-(oxane-4-carbonyl)-2-{[3-(trifluoromethyl)phenyl]methyl}morpholine
2-[7-(2-methoxyethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]-4,6-dimethylpyridine-3-carbonitrile
N-methyl-N-(1,2-oxazol-5-ylmethyl)-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
N,N-diethyl-5-{1-[3-(furan-2-yl)propanoyl]pyrrolidin-2-yl}thiophene-2-carboxamide