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1-[benzyl(methyl)amino]-3-[4-({[(4-fluorophenyl)methyl]amino}methyl)phenoxy]propan-2-ol
1-[(4-chlorophenyl)methyl]-N-cyclooctyl-6-oxopiperidine-3-carboxamide
2-{4-[(4-{[(3R)-3-hydroxypyrrolidin-1-yl]methyl}-1H-1,2,3-triazol-1-yl)methyl]piperidin-1-yl}pyridine-4-carbonitrile
methyl 3-methyl-4-({[4-(oxolan-2-yl)butyl]carbamoyl}amino)benzoate
3-{3-[2-(methylsulfanyl)benzoyl]piperidine-1-carbonyl}-4,5,6,7-tetrahydro-2H-indazole
1-(1,2-oxazole-3-carbonyl)-3-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidine
N-(6-cyanopyridin-3-yl)-4-{[3-(dimethylamino)pyrrolidin-1-yl]methyl}benzamide
1-cyclopentyl-4-{[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}piperazine
(3aR,6aS)-2-[(6-methoxynaphthalen-2-yl)methyl]-5-methyl-octahydropyrrolo[3,4-c]pyrrole
N-methyl-2-{1-[(4-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-(oxan-4-yl)acetamide
{2-[(2R,3R)-3-amino-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]-2-oxoethyl}urea
N-{4-[(4-{4-ethyl-1-[2-(4-methoxyphenyl)ethyl]-2,5-dioxoimidazolidin-4-yl}piperidin-1-yl)methyl]phenyl}acetamide
(2S,4S)-1-[(3,5-dimethylphenyl)methyl]-N-ethyl-4-[(3E)-hex-3-enamido]pyrrolidine-2-carboxamide
7-(3-chlorophenyl)-4-(1-methyl-1H-pyrazole-4-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
4-[(1H-imidazol-2-ylmethyl)amino]-1-[2-(4-methoxyphenyl)ethyl]pyrrolidin-2-one
4-{[(1-hydroxybutan-2-yl)(pyridin-3-ylmethyl)amino]methyl}-2,6-dimethylphenyl acetate
(5-{1-[1-(1H-indol-1-yl)propan-2-yl]-1H-imidazol-2-yl}furan-2-yl)methanol
N-methyl-N-(quinolin-8-ylmethyl)-2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetamide
N-{[4-(3-fluorophenyl)oxan-4-yl]methyl}-2-(methylamino)pyridine-4-carboxamide
[(4-methyl-1H-imidazol-5-yl)methyl][(5-methylthiophen-2-yl)methyl](prop-2-en-1-yl)amine
({2-[2-(dimethylamino)ethoxy]-3-methoxyphenyl}methyl)({2,3-dimethylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)amine
5-(morpholine-4-carbonyl)-2-(propan-2-yl)-1,3-benzoxazole
1-[(3-fluorophenyl)methyl]-4-[(2S)-2-hydroxy-3-phenylpropanoyl]piperazin-2-one
4-(5-fluoropyridin-2-yl)-N-(pyridin-4-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
3-(2-fluorophenyl)-N-(2-{2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}ethyl)-1H-pyrazole-5-carboxamide
4-[(2-fluorophenyl)methyl]-N-(3-methyl-1,2,4-thiadiazol-5-yl)piperidine-1-carboxamide
2-[(4-chlorophenyl)methyl]-N-(1-methoxypropan-2-yl)-1,3-benzoxazole-5-carboxamide
4-{thieno[3,2-d]pyrimidin-4-yl}-2-(trifluoromethyl)morpholine
2-{[1-(2-fluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}pyridine
(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)({[2-(ethylsulfanyl)pyrimidin-5-yl]methyl})methylamine
N-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
N-{1-[1-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}-2-(2-oxoazepan-1-yl)acetamide
1-[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl]cyclopropane-1-carbonitrile
(1R,2R)-2-[5-(2-phenoxyethyl)-3-(pyridin-4-yl)-1H-1,2,4-triazol-1-yl]cyclohexan-1-ol
1-{[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl}-3-(1H-pyrazol-5-yl)piperidine
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-4-hydroxy-2-(pyridin-2-yl)pyrimidine-5-carboxamide
N-cyclohexyl-3-[2-(2,5,7-trimethyl-1H-indol-3-yl)acetamido]propanamide
1-(1-ethyl-5-methyl-1H-pyrazole-4-carbonyl)-4-[(2-methylphenyl)sulfanyl]piperidine
(4aR,8aS)-6-benzoyl-1-(2,2-dimethyloxane-4-carbonyl)-decahydro-1,6-naphthyridine
2-[3-benzyl-1-(2-methoxyphenyl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-(cyclopropylmethyl)acetamide
3,5-difluoro-2-[4-(3-phenyl-1,2,4-oxadiazol-5-yl)piperidine-1-carbonyl]pyridine
{[(1R,5S,6S)-3-(1-benzothiophene-2-carbonyl)-3-azabicyclo[3.1.0]hexan-6-yl]methyl}dimethylamine
N-[(1-methanesulfonylpiperidin-3-yl)methyl]-3-methyl-1-propyl-1H-pyrazole-4-carboxamide
ethyl 1-[(4-hydroxyquinolin-2-yl)methyl]-4-(2-methoxyethyl)piperidine-4-carboxylate
2-{4-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-[(4-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
2-methyl-4-{3-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]phenyl}butan-2-ol
2-[3-({[1-(4-chlorophenyl)-3-hydroxypropan-2-yl]amino}methyl)-2-methyl-1H-indol-1-yl]acetamide
N-{1-[1-(1,4-dithiepan-6-yl)piperidin-4-yl]-1H-pyrazol-5-yl}pyridine-3-carboxamide
5-(2,3-difluoro-6-methoxyphenyl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
N-(2-methylphenyl)-2-oxo-2-[3-(pyridin-3-ylmethoxy)piperidin-1-yl]acetamide