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3-{[4-(4-methoxypyrimidin-2-yl)piperazin-1-yl]methyl}piperidin-3-ol
5-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]-1-(pyridin-2-ylmethyl)piperidin-2-one
N-(1-{7-[(2-ethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-3-methylbutyl)-5-(methoxymethyl)furan-2-carboxamide
3-cyclohexyl-N-[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-1H-pyrazole-4-carboxamide
[1-(6-methoxypyrimidin-4-yl)-3-[(2-methylphenyl)methyl]piperidin-3-yl]methanol
2-(furan-3-carbonyl)-6-methyl-5-[5-(1H-pyrrol-2-yl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydro-2,7-naphthyridine
N-(4-methoxy-2-methylphenyl)-3-[1-(2-methyl-1,3-thiazole-4-carbonyl)piperidin-3-yl]propanamide
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-4-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-methylbenzamide
(5S,9aS,9bS)-5-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-2-[(3-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-methyl-N-({2-[(2-oxopyrrolidin-1-yl)methyl]phenyl}methyl)-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
(3S,4S)-4-methyl-1-[6-(1-methyl-1H-imidazol-2-yl)pyridazin-3-yl]piperidine-3,4-diol
4-phenoxy-1-[2-(1,3-thiazol-4-yl)acetyl]piperidine-4-carboxylic acid
3-(5-{[2-(propan-2-yl)pyrimidin-5-yl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl)benzonitrile
N-cyclohexyl-4-methyl-N-(pyridin-4-ylmethyl)-3,4-dihydro-2H-1,4-benzoxazine-2-carboxamide
(4aS,7aR)-1-(2-methyl-4-phenylpyrimidine-5-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-(azepane-1-carbonyl)-1-ethyl-5-(thiomorpholin-4-yl)-4,5,6,7-tetrahydro-1H-indazole
2-(3-hydroxyphenyl)-1-{3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}ethan-1-one
({4-ethyl-5-[1-(2-methylpyridin-4-yl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
3-{4-[2-(piperidine-1-carbonyl)phenoxy]piperidin-1-yl}propane-1,2-diol
5-(3-{[2-(dimethylamino)ethyl](methyl)amino}piperidine-1-carbonyl)-6-methyl-2-oxo-1,2-dihydropyridine-3-carbonitrile
5-(2-{[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]amino}ethyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
(1R,7S)-3-[(3,4-dimethylphenyl)methyl]-N-methyl-4-oxo-N-propyl-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
N-(3-{4-[(5-hydroxyadamantan-2-yl)amino]piperidin-1-yl}phenyl)-4-phenylbutanamide
3-[3-(4-phenoxybenzoyl)piperidin-1-yl]propanoic acid
2,6-dimethyl-5-{2-oxo-2-[(1S,5R)-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethyl}-3,4-dihydropyrimidin-4-one
4-ethyl-3-(1-{[4-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
5-[1-(3-fluorophenyl)-1H-pyrazol-3-yl]-N-(furan-2-ylmethyl)-4-methyl-1,3-thiazol-2-amine
methyl 4-{[2-(4-methoxyphenyl)ethyl][(1-methylpiperidin-4-yl)methyl]carbamoyl}benzoate
1-(2,2-dimethylpropyl)-4-[(1H-imidazol-4-ylmethyl)amino]pyrrolidin-2-one
N-[(2,4-dimethoxyphenyl)methyl]-N'-(4-methylphenyl)propanediamide
1-(4-methoxyphenyl)-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}cyclopropane-1-carboxamide
4-methoxy-4-phenyl-1-[2-(pyrrolidin-3-yl)benzoyl]piperidine
N-[4-methoxy-2-(2-methylpropanamido)phenyl]-2,3-dihydro-1H-indene-2-carboxamide
5-(propan-2-yl)-N-{1-[2-(trifluoromethyl)phenyl]ethyl}pyrazolo[1,5-a]pyrimidin-7-amine
N-{[1-(6-methylpyridin-2-yl)-3-(oxolan-3-yl)-1H-1,2,4-triazol-5-yl]methyl}cyclopropanamine
4-(4-fluorophenyl)-1-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]piperidin-4-ol
N-[2-(furan-2-yl)ethyl]-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-4-carboxamide
2-[4-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-1,5-dimethyl-1H-indole
methyl({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)amine
2-amino-8-[1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-1,3,8-triazaspiro[4.5]dec-1-en-4-one
3-[(4aS,8aR)-decahydroisoquinoline-2-carbonyl]-1-cyclopentyl-5-(piperidine-1-carbonyl)-1,4-dihydropyridin-4-one
2-(1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}pyrrolidin-2-yl)-6-methyl-1H-1,3-benzodiazole
2-[2-(dimethylamino)ethyl]-9-(4-methylpyrimidine-5-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
6-[3-(4-propylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-2,3,4,5-tetrahydropyridazin-3-one
N-[(4-chlorophenyl)(phenyl)methyl]-2-oxo-6-(pyrrolidin-1-ylmethyl)-1,2-dihydropyridine-3-carboxamide
3-chloro-4-fluoro-N-({3-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-N-(pyridin-2-ylmethyl)benzene-1-sulfonamide
4-(2,1,3-benzoxadiazol-5-ylmethyl)-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
(3S,4S)-1-{[2-(3-methylphenyl)pyrimidin-5-yl]methyl}-4-[4-(pyridin-2-yl)piperazin-1-yl]pyrrolidin-3-ol
1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-2-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]piperidine
1-{[2-(butylsulfanyl)pyrimidin-5-yl]methyl}piperidine-3-carbonitrile