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N-ethyl-1,3-dimethyl-N-(oxan-4-yl)-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
N-{3-[({[1-(2-hydroxyethyl)piperidin-4-yl]methyl}(methyl)carbamoyl)amino]-4-methoxyphenyl}acetamide
N-[2-(1H-imidazol-1-yl)ethyl]-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-3-carboxamide
8-[6-(morpholine-4-carbonyl)pyrazin-2-yl]-1-oxa-8-azaspiro[4.5]decane
1-{3-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-2,3,4,9-tetrahydro-1H-carbazole
[2-methoxy-5-({[(2-methoxyphenyl)methyl](propyl)amino}methyl)phenyl]methanol
1-[1-(2-methylpyrimidin-4-yl)piperidin-4-yl]-N-(2-phenylethyl)piperidine-3-carboxamide
1-methyl-N-{1-[(2-methylphenyl)methyl]cyclopropyl}azepane-2-carboxamide
8-{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
(4aS,8aS)-2-{5-[(4-methylpiperazin-1-yl)methyl]pyridin-2-yl}-decahydro-2,7-naphthyridin-4a-ol
7-(4-chlorophenyl)-2-(4-methylpyridin-2-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
1-{1-[(2-methylphenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-4-phenylazepane
N,N,3-trimethyl-4-({[(1-phenylcyclopentyl)methyl]carbamoyl}amino)benzamide
(2S)-2-hydroxy-1-{2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}propan-1-one
N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}-2,3-dihydro-1H-inden-2-amine
5-cyclopropanecarbonyl-1'-(piperidin-3-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]-1-(thiophen-3-ylmethyl)piperidine
N-(3-chloro-4-methoxyphenyl)-3-{1-[3-(pyrazin-2-yl)propanoyl]piperidin-3-yl}propanamide
2-({[cyclopropyl(1-methyl-1H-imidazol-2-yl)methyl]amino}methyl)-6-methylquinolin-4-ol
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
8-[(4-hydroxyphenyl)methyl]-1-(2-methoxyethyl)-3-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-(1-{[4-chloro-2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}piperidin-3-yl)pyrimidine
N-(2H-1,3-benzodioxol-5-yl)-2-[4-(2-cyclohexylacetyl)morpholin-3-yl]acetamide
2-(3-hydroxypropyl)-9-{2-[methyl(phenyl)amino]acetyl}-2,9-diazaspiro[5.5]undecan-3-one
4-(1-hydroxy-2-phenylethyl)-N-(5-methyl-1,3,4-thiadiazol-2-yl)piperidine-1-carboxamide
2-(adamantan-1-yl)-4-hydroxy-N-[4-(methylamino)butyl]pyrimidine-5-carboxamide
(1S,5R)-3-benzoyl-6-[4-(prop-2-en-1-yl)benzoyl]-3,6-diazabicyclo[3.2.2]nonane
6-[4-(3-methylphenoxy)piperidine-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-(3-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-sulfonyl}benzoyl)piperazine
(4aR,7aS)-1-cyclopropanecarbonyl-4-(1-methyl-1H-pyrazole-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-{2-[3-(4-phenylbenzoyl)piperidin-1-yl]ethyl}morpholine
2-methyl-N-{2-[(pyridin-3-yl)amino]ethyl}-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
(1R,2R,6S,7S)-4-[5-(oxolan-2-yl)thiophene-2-carbonyl]-4-azatricyclo[5.2.1.02,6]decane
methyl({[1-(piperidin-1-yl)cyclohexyl]methyl}){4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}amine
N-{1-[4-(tert-butylcarbamoyl)phenyl]-1H-pyrazol-4-yl}oxane-4-carboxamide
1-{2-[4-(4-fluorophenyl)-1,4-diazepan-1-yl]-2-oxoethyl}-1,2-dihydroquinolin-2-one
N-benzyl-N-ethyl-5-(3-fluorophenoxymethyl)-1H-pyrazole-3-carboxamide
2-methyl-6-[1-(4-methyl-1,3-thiazol-2-yl)piperidin-3-yl]pyrimidin-4-ol
(1S,9S)-11-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one
N-[1-(morpholine-4-carbonyl)piperidin-4-yl]-4-(pyridin-3-yl)pyrimidin-2-amine
3-[(3S,5S,9S)-2,8-dioxo-1,7-diazatricyclo[7.3.0.03,7]dodecan-5-yl]-1-(5-fluoro-2-methylphenyl)urea
3-({4-[(dimethylcarbamoyl)methyl]piperazin-1-yl}methyl)-N-(1-methyl-1H-pyrazol-4-yl)benzamide
1-methanesulfonyl-4-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-1,4-diazepane
1-(2-methoxyphenyl)-2,2-dimethyl-4-{[1-(propan-2-yl)-1H-imidazol-5-yl]methyl}piperazine
1-[(1S,5R)-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
4-{3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}-1-[4-(propan-2-yl)phenyl]pyrrolidin-2-one
N-[(5-methylfuran-2-yl)methyl]-1,9-dioxaspiro[5.5]undecan-4-amine
N-cyclobutyl-2-{1-[(4-methoxy-3-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
{5-[3-(propan-2-yloxy)phenyl]-1H-1,3-benzodiazol-2-yl}methanol
(3S,4R)-1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-N,N-dimethyl-4-(propan-2-yl)pyrrolidin-3-amine