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3-(oxolan-3-yl)-5-(5-propylthiophen-3-yl)-1,2,4-oxadiazole
5-[3-(4-benzyl-4-hydroxypiperidin-1-yl)-3-oxopropyl]imidazolidine-2,4-dione
7-(5-methylthiophen-2-yl)-4-[2-(1H-1,2,3,4-tetrazol-5-yl)ethyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-amino-7-methyl-4-[2-(propan-2-yl)pyrimidin-5-yl]-5H,7H-thieno[3,4-b]pyridine-3-carbonitrile
3-(4-{[3-(naphthalen-1-yl)-1H-pyrazol-4-yl]methyl}piperazin-1-yl)propanamide
(1S,5R)-3-(dimethyl-1,2-oxazole-4-carbonyl)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-oxo-N-({2-[4-(pyridin-2-yl)piperazin-1-yl]pyridin-3-yl}methyl)pentanamide
2-methyl-4-(4-{5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl}piperazin-1-yl)-6-(piperidin-4-yl)pyrimidine
5-{4-[(2,3-dimethyl-1H-indol-7-yl)methyl]piperazin-1-yl}-2-methyl-2,3-dihydropyridazin-3-one
3-{5-[2-(3-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}-N-[2-(6-methylpyridin-2-yl)ethyl]propanamide
4-hydroxy-N-[2-(1H-indol-1-yl)ethyl]-N-methyl-2-(pyridin-2-yl)pyrimidine-5-carboxamide
N-[3-(3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)-3-oxopropyl]methanesulfonamide
N-[2-(4,6-dihydroxypyrimidin-2-yl)ethyl]-3-(4-methoxyphenyl)-1H-pyrazole-5-carboxamide
N-(5-acetyl-2-methoxyphenyl)-3-(3-methylphenoxy)azetidine-1-carboxamide
5-chloro-6-(4-methoxy-2-methylphenyl)-2-methylpyrimidin-4-ol
N,4-dimethyl-2-(methylamino)-N-(pyrimidin-4-ylmethyl)-1,3-thiazole-5-carboxamide
N-{1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-2-(piperidin-1-yl)acetamide
5-{1-[(3-fluorophenyl)methyl]-1H-pyrazol-3-yl}-4-methyl-N-[(3-phenyl-1H-pyrazol-4-yl)methyl]-1,3-thiazol-2-amine
N-cycloheptyl-3-{5-[methoxy(phenyl)methyl]-1,3,4-oxadiazol-2-yl}propanamide
2-[(3,4-difluorophenyl)methyl]-8-(6-methoxypyrimidin-4-yl)-2,8-diazaspiro[4.5]decan-3-one
(1R,2S,9R)-11-(5-propyl-1,2,4-oxadiazol-3-yl)-7,11-diazatricyclo[7.3.1.02,7]tridecan-6-one
1-[(4-methoxyphenyl)methyl]-6-(pyridin-3-ylmethoxy)-4-(1,2,5-thiadiazole-3-carbonyl)-1,4-diazepan-2-one
4-[3-(cyclohexylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]morpholine
2-{4-[5-(1H-indol-1-ylmethyl)furan-2-carbonyl]morpholin-3-yl}acetic acid
2-[4-(benzyloxy)-3-fluorophenyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
1-[(1S,5R)-6-[(5-chlorothiophen-2-yl)sulfonyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
N-[4-({ethyl[(1-ethyl-1H-pyrazol-4-yl)methyl]carbamoyl}methyl)phenyl]butanamide
5,7-dimethyl-N-[1-methyl-4-(propan-2-yloxy)-1H-indazol-3-yl]-[1,2,4]triazolo[4,3-a]pyrimidine-3-carboxamide
4-(hydroxymethyl)-N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}benzamide
1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-5-methyl-N,N-bis(prop-2-en-1-yl)-1H-pyrazole-4-carboxamide
(2S,4S)-1-(2,3-dihydro-1H-inden-2-yl)-4-({[2-(prop-2-en-1-yloxy)phenyl]methyl}amino)-N-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
2-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)acetyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
3-[6-amino-5-cyano-4-(5-hydroxy-2-methoxyphenyl)pyridin-2-yl]benzoic acid
1-(2-methoxyphenyl)-4-[4-(propan-2-yl)benzoyl]piperazin-2-one
11-(cyclopentylamino)-4-[(2-methoxynaphthalen-1-yl)methyl]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
N-(furan-2-ylmethyl)-4-[1-(4-methoxyphenyl)-1H-pyrazol-4-yl]pyrimidin-2-amine
N-(1-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
5-(3-methoxyphenyl)-N-[2-(pyrrolidine-1-sulfonyl)ethyl]furan-2-carboxamide
N-[1-(1,3-dimethyl-1H-pyrazol-4-yl)ethyl]-9H-purin-6-amine
(2R,3R)-3-{1,4-dioxa-8-azaspiro[4.5]decan-8-yl}-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
6-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-2,5-dioxo-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
2-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]-7-methoxy-4-methylquinazoline
2-{4-[(5-propyl-1,3,4-oxadiazol-2-yl)amino]piperidin-1-yl}ethan-1-ol
N4-{[2-(dimethylamino)-1,3-thiazol-4-yl]methyl}-2-methylpyrimidine-4,6-diamine
(2R,3R,6R)-5-(1,3-dimethyl-1H-pyrazole-4-carbonyl)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
4-{5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-6-yl}-N-phenylpiperidine-1-carboxamide
1-methyl-N-[(4-methylpyridin-2-yl)methyl]-2-(morpholin-4-yl)-1H-1,3-benzodiazole-5-carboxamide
2,6-dimethyl-5-(2-oxo-2-{4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazin-1-yl}ethyl)-3,4-dihydropyrimidin-4-one
2-{4-[(1-ethyl-1H-pyrazol-4-yl)methyl]-1-(1-methylpiperidin-4-yl)piperazin-2-yl}ethan-1-ol
N-(1-{imidazo[1,2-a]pyrimidin-2-yl}propyl)-3-propyl-1H-pyrazole-5-carboxamide