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2-(dimethylamino)-2-(4-fluorophenyl)-N-[3-(2-oxopyrrolidin-1-yl)propyl]acetamide
3,3-dimethyl-1-({5-[(1-propyl-1H-imidazol-2-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)urea
N-(1-methanesulfonylpiperidin-4-yl)-3-(1H-pyrazol-1-ylmethyl)benzamide
[3-(cyclopropylmethyl)-1-(2-methoxy-3-methylbenzoyl)piperidin-3-yl]methanol
6-methoxy-N-[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
3-[(dimethylamino)methyl]-1-[4-methyl-2-(propan-2-yl)pyrimidine-5-carbonyl]pyrrolidin-3-ol
N-[(3-ethoxyphenyl)methyl]-N-(2-hydroxyethyl)-2,5-dimethyl-1,3-thiazole-4-carboxamide
N-{2-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-oxoethyl}acetamide
N-[(3S,4R)-1-(4-fluoro-3-methoxybenzoyl)-4-(4-methoxyphenyl)pyrrolidin-3-yl]acetamide
(1R,3S)-7-(4-ethyl-5-methylpyrimidin-2-yl)-7-azaspiro[3.5]nonane-1,3-diol
4-{[5-(1-ethyl-1H-imidazol-5-yl)-4-phenyl-1H-imidazol-1-yl]methyl}-3,5-dimethyl-1,2-oxazole
N-[1-(3-chlorophenyl)cyclopropyl]-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
methyl({[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl})[3-(oxolan-2-yl)propyl]amine
1-(1H-1,3-benzodiazole-5-carbonyl)-3-[(2E)-3-phenylprop-2-en-1-yl]piperidine-3-carboxylic acid
N-[(3R,4S)-1-(dimethylsulfamoyl)-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
3-amino-3-(3,4-dimethoxyphenyl)-1-(7-methoxy-2,3,4,5-tetrahydro-1H-3-benzazepin-3-yl)propan-1-one
2-[3-(hydroxymethyl)-3-[(2-methylphenyl)methyl]piperidin-1-yl]pyridine-4-carbonitrile
N-[(3R,4S)-1-acetyl-4-cyclopropylpyrrolidin-3-yl]-5,7-dimethylpyrazolo[1,5-a]pyrimidine-3-carboxamide
3-chloro-2-{3,5-dimethyl-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyrazine-7-carbonyl}-6-methylpyrazolo[1,5-a]pyrimidine
N-(2-methoxyethyl)-N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-3-(methylsulfanyl)propanamide
1-[2-(4-methoxyphenyl)ethyl]-3-methyl-8-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
methyl 3-(2H-1,3-benzodioxol-5-ylmethyl)-9-[2-(2-fluorophenyl)ethoxy]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-({3-[(2-fluorophenyl)methoxy]-4-methoxyphenyl}methyl)-2,3-dimethyl-N-(pyridin-4-ylmethyl)-1H-indole-7-carboxamide
N-{[1-(2,2-dimethylpropyl)piperidin-3-yl]methyl}-4-methoxybenzene-1-sulfonamide
N-cyclopropyl-3-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]benzamide
N-[(3-ethoxyphenyl)methyl]-N-(prop-2-en-1-yl)-1,2-oxazole-3-carboxamide
N-(butan-2-yl)-2-(1-propylpiperidin-4-yl)-N-(pyridin-4-ylmethyl)acetamide
1-cyclopentyl-N-[2-(5-methoxy-1H-indol-3-yl)ethyl]piperidine-3-carboxamide
1-[1-(1-butyl-3-cyclopentyl-1H-1,2,4-triazol-5-yl)ethyl]pyrrolidin-2-one
2-(2-phenylethyl)-1-[4-(4H-1,2,4-triazol-4-yl)benzoyl]piperidine
6-ethyl-4-(2-ethyl-2,5-dihydro-1H-pyrrole-1-carbonyl)-1,2-dihydropyridin-2-one
1-[2-(2-hydroxyethyl)piperidin-1-yl]-2-(2,4,7-trimethyl-1H-indol-3-yl)ethan-1-one
N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]-1-(1,2-oxazol-3-ylmethyl)piperidine-4-carboxamide
N-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)-6-methylimidazo[2,1-b][1,3]thiazole-5-carboxamide
4-(2,5-dimethoxyphenyl)-6-(1H-pyrazol-1-yl)pyrimidine
2-[5-(2-ethylpyridin-4-yl)-3-methyl-1H-1,2,4-triazol-1-yl]acetic acid
5-(2-benzyl-1,3-thiazole-4-carbonyl)-N-(3-methoxypropyl)-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N,N-dimethyl-6-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrazin-2-amine
(3S,5S)-1-methyl-5-[3-(naphthalen-1-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]pyrrolidin-3-amine
methyl 6-({methyl[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]amino}methyl)-3-(2-phenoxyacetamido)thieno[2,3-b]pyridine-2-carboxylate
1-cycloheptanecarbonyl-4-[(4-propyl-1H-1,2,3-triazol-1-yl)methyl]piperidine
3-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}-1-[4-(1H-pyrazol-4-yl)phenyl]urea
1-(2,6-dimethylpyridin-4-yl)-4-{[4-(1H-imidazol-1-yl)phenyl]methyl}piperazine
{[1-(2,4-difluorophenyl)-3-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}[3-(dimethylamino)propyl]amine
3-[1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)piperidin-3-yl]-1-[4-(pyridin-2-yl)piperazin-1-yl]propan-1-one
3-(azepan-1-ylmethyl)-N-[(3R,4R)-3-hydroxypiperidin-4-yl]benzamide
1-[(4-chlorophenyl)methyl]-N-cyclobutyl-6-oxopiperidine-3-carboxamide
2-(3-methoxypropyl)-9-(2-methyl-1-benzofuran-5-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
1,4-dimethyl-N-[3-(oxolan-3-yl)propyl]piperidine-4-carboxamide
N-({1-[(5-ethylthiophen-2-yl)sulfonyl]piperidin-3-yl}methyl)pyridine-3-carboxamide