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(4aR,7aS)-1-cyclobutanecarbonyl-4-[5-(hydroxymethyl)furan-2-carbonyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-[3-(2-fluorophenyl)pyrrolidin-1-yl]-5-propyl-1,3,4-oxadiazole
2-{3-[({[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl}(methyl)amino)methyl]phenyl}-6-methyl-3,4-dihydropyrimidin-4-one
5-(2,6-difluoro-3-methylphenyl)-1-methyl-4-phenyl-1H-imidazole
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(5-methylpyrazine-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
{3-[4-(3-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]-3-oxopropyl}urea
4-(1H-imidazol-1-ylmethyl)-1-{[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methyl}piperidin-4-ol
1-cyclopentyl-4-(1,2-oxazole-3-carbonyl)-1,4-diazepane-6-carboxylic acid
2-(2-methoxy-4-{[3-(4H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}phenoxy)acetamide
1-{1-[2-(methylamino)acetyl]piperidin-4-yl}-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
(3S,9aR)-3-propyl-8-[4-(trifluoromethoxy)benzoyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-(furan-3-ylmethyl)-N-[4-(1H-pyrazol-1-yl)phenyl]piperidine-2-carboxamide
4-[(1-cyclohexyl-1H-imidazol-5-yl)methyl]-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
1-[3-(1H-pyrazol-1-yl)benzoyl]-4-(pyrimidin-2-yl)-1,4-diazepane
2-[2-(diethylamino)ethyl]-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
5-(propan-2-yl)-N-[1-(pyrimidin-2-yl)piperidin-3-yl]-1,2-oxazole-3-carboxamide
2-(3-chloro-4-fluorophenyl)pyridine-3-carboxamide
1-(1,3-benzothiazol-2-yl)-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-3-amine
6-{1-[(2E)-3,7-dimethylocta-2,6-dien-1-yl]piperidin-3-yl}-2-methylpyrimidin-4-ol
N-[(5-methylfuran-2-yl)methyl]-3-{1-[(5-methylthiophen-2-yl)sulfonyl]piperidin-3-yl}propanamide
2-(4-methanesulfonylbenzenesulfonyl)-2,7-diazaspiro[4.5]decane
N-[3-(4-{[4-(pyridin-2-yl)piperazin-1-yl]methyl}phenoxy)propyl]thiophene-2-sulfonamide
N-{2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]ethyl}-5-(2-fluorophenyl)-1,2,4-triazin-3-amine
2,3-difluoro-5-[2-(3-hydroxypropyl)-1H-1,3-benzodiazol-1-yl]phenol
(3S,4S)-4-cyclopropyl-1-[(3-fluoro-2-methylphenyl)methyl]pyrrolidine-3-carboxylic acid
2-[3-(2H-1,3-benzodioxol-5-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-N-(oxolan-2-ylmethyl)acetamide
3-(dimethyl-1,2-oxazol-4-yl)-1-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}urea
2-[(3aR,6aS)-octahydropyrrolo[3,4-c]pyrrole-2-carbonyl]-5-chloro-3-phenyl-1H-indole
1-[3-({[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]amino}methyl)pyridin-2-yl]piperidin-3-ol
1-[(2-fluorophenyl)methyl]-N-[2-(5-methylfuran-2-yl)ethyl]-6-oxopiperidine-3-carboxamide
N-(4-fluoro-2-methylphenyl)-3-[1-(pyridazine-4-carbonyl)piperidin-3-yl]propanamide
1-(2H-1,3-benzodioxol-4-ylmethyl)-3-(5-fluoro-2-methoxybenzoyl)piperidine
N-{7-methoxy-2-oxo-4-[(1s,4s)-4-aminocyclohexyl]-1,2,3,4-tetrahydroquinolin-6-yl}-3-methylbutanamide
N-{2-[7-(2,3,6-trifluorobenzoyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}cyclohexanecarboxamide
N-(1-cycloheptylpiperidin-3-yl)-2-methyl-1,3-thiazole-4-carboxamide
N-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-N-methyl-5-(oxolan-2-yl)thiophene-2-carboxamide
1-({3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-4-(2-methylphenyl)piperazine
N-{1,9-dioxaspiro[5.5]undecan-4-yl}-1-(pyridin-3-ylmethyl)piperidin-4-amine
1-{6-chloroimidazo[1,2-a]pyridine-2-carbonyl}-3-(hydroxymethyl)piperidin-3-ol
2-methyl-5-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]-1,3-benzothiazole
3-[2-(2-methyl-1H-imidazol-1-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-(3-hydroxy-1,2-oxazol-5-yl)-N-[(3R,4S)-1-methanesulfonyl-4-propylpyrrolidin-3-yl]propanamide
2,2-diphenyl-1-(4-{pyrazolo[1,5-a]pyrimidine-3-carbonyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)ethan-1-ol
N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)-2-(pyridin-4-yl)acetamide
methyl[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]{[5-methyl-2-(5-methylfuran-2-yl)-1,3-oxazol-4-yl]methyl}amine
1-(2-{[7-(pyrazin-2-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]amino}ethyl)imidazolidin-2-one
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-methyl-N-(thiophen-3-ylmethyl)piperidine-3-carboxamide
(1R,7S)-N-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-3-[2-(4-methylphenyl)ethyl]-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
4-(1H-imidazol-1-yl)-1-[6-(morpholin-4-yl)pyrimidin-4-yl]piperidine-4-carboxylic acid
1-(4-{[3-(2,5-difluorobenzoyl)piperidin-1-yl]methyl}phenyl)imidazolidin-2-one