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N-benzyl-2-(4-{4-[4-(thiophen-2-ylmethyl)piperazin-1-yl]piperidin-1-yl}phenyl)acetamide
N,N-dimethyl-4-(3,4,5-trimethoxyphenyl)-5,6,7,8-tetrahydroquinazolin-2-amine
2-(dimethylamino)-N-(3-hydroxypropyl)-2-(3-methylphenyl)acetamide
(3R,4S)-3,4-dimethyl-1-[1-methyl-3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]piperidin-4-ol
(2R,3R,6R)-5-(4-ethenylbenzoyl)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-(2-methoxyphenyl)-N-[5-oxo-1-(2-phenylethyl)pyrrolidin-3-yl]acetamide
5-{1-[3-(1H-imidazol-1-yl)propyl]-1H-imidazol-2-yl}-2-(pyrrolidin-1-yl)-1,3-thiazole
1-[3-(2-chlorophenyl)propanoyl]-3-(2-methoxyethyl)piperidine-3-carboxylic acid
1-(3-methoxyphenyl)-4-[2-(oxolan-2-ylmethoxy)acetyl]piperazin-2-one
1-benzyl-N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]piperidin-4-amine
4-chloro-1,5-dimethyl-3-[2-(thiophen-2-yl)azetidine-1-carbonyl]-1H-pyrazole
4-{5-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-3-yl}-1H-indole
N-[2-(dimethylamino)-2-(furan-2-yl)ethyl]-1-{thieno[3,2-d]pyrimidin-4-yl}piperidin-4-amine
(2R,6R)-10-methoxy-4-[2-(2-oxopiperidin-1-yl)acetyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
N-{[1-(1,2,4-oxadiazol-3-ylmethyl)piperidin-3-yl]methyl}-4-phenylbenzamide
(3aR,6aR)-2-[(dimethyl-1,3-thiazol-5-yl)methyl]-5-(2-methoxyethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-(morpholin-4-yl)-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)pyrimidine-5-carboxamide
1-(2-amino-9H-purin-6-yl)-4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]-1,4-diazepan-6-ol
N-[(1R,3R)-3-aminocyclopentyl]-2-(methylamino)-1,3-thiazole-4-carboxamide
4-[3-(hydroxymethyl)-3-(2-methoxyethyl)piperidine-1-carbonyl]benzene-1-sulfonamide
2-[3-(pyridin-3-ylmethoxy)piperidine-1-carbonyl]-1H-indole
4-(1H-imidazol-1-yl)-1-{6-methylpyrazolo[1,5-a]pyrimidine-3-carbonyl}piperidine-4-carboxylic acid
N-(2-phenylethyl)-4-{[1-(pyrimidin-2-yl)piperidin-4-yl]oxy}benzamide
2-cyclopropyl-N-[3-(morpholin-4-yl)propyl]pyrimidine-5-carboxamide
8-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propanoyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
N,1-dimethyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-(cyclohexylmethyl)-4-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]morpholine
2-(4-{[5-(methoxymethyl)furan-2-yl]methyl}-1-(propan-2-yl)piperazin-2-yl)ethan-1-ol
2-methyl-1-[2-(4H-1,2,4-triazol-4-yl)ethyl]-1,4-dihydroquinolin-4-one
{1-[1-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]amine
N-[2-(5-amino-1H-1,2,4-triazol-3-yl)ethyl]-1-(6-methyl-2-propylpyrimidin-4-yl)piperidin-4-amine
(benzylsulfamoyl)({[1-(ethoxymethyl)cyclobutyl]methyl})amine
1-(3-chloro-4-methoxyphenyl)-5-oxo-N-(pyrimidin-4-ylmethyl)pyrrolidine-3-carboxamide
N-cyclopentyl-2-methyl-4-(morpholin-4-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-7-carboxamide
1-ethyl-4-{5-[3-(trifluoromethyl)phenoxymethyl]-1H-pyrazole-3-carbonyl}piperazine
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-[(3-hydroxy-4-methoxyphenyl)methyl]piperidine-2-carboxamide
3-{[3-(naphthalen-1-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]sulfonyl}pyridine
8-{5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}-1-oxa-8-azaspiro[4.5]decane
1-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]-2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethan-1-one
2-{[2-(dimethylamino)ethyl][(3-methylthiophen-2-yl)methyl]amino}acetic acid
N-[(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)methyl]-1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
(3aR,5R,6S,7aS)-2-[1-(2,3-dimethylphenyl)piperidin-4-yl]-octahydro-1H-isoindole-5,6-diol
2-butyl-N-[(4-methyl-1,3-thiazol-2-yl)methyl]-1,3-benzoxazole-5-carboxamide
3-{2-[4-(6-methoxy-2,3-dihydro-1H-inden-5-yl)-1H-1,2,3-triazol-1-yl]ethyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
1-{[1-(cyclohexylmethyl)-2-cyclopropylmethanesulfonyl-1H-imidazol-5-yl]methyl}-4-methoxypiperidine
({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)(methyl){[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}amine
1-(cyclohexylmethyl)-5-(ethylamino)-N-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-cyclohexyl-3-ethyl-N-(2-hydroxy-2-phenylethyl)-5-methyl-1,2-oxazole-4-carboxamide
2-{[2-(2,3-dimethoxyphenyl)-1H-imidazol-1-yl]methyl}-4-methanesulfonylmorpholine
7-chloro-N-ethyl-N-[2-hydroxy-2-(3-hydroxyphenyl)ethyl]-1-methyl-1H-indole-2-carboxamide