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1-({5-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}amino)butan-2-ol
4-(piperidine-1-carbonyl)-2-(1H-pyrazol-4-yl)pyridine
2-amino-4-(1H-imidazol-4-yl)-6-(1H-indol-3-yl)pyridine-3-carbonitrile
(3R,4R)-4-(hydroxymethyl)-1-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}piperidin-3-ol
N-[4-(3-methoxyphenyl)phenyl]-1-[2-(methylsulfanyl)acetyl]piperidine-3-carboxamide
3-(4-methyl-1,3-thiazol-5-yl)-N-{[5-(thiophen-2-yl)-1,2,4-oxadiazol-3-yl]methyl}propanamide
1-[4-(3-{[(2,6-dimethylhept-5-en-1-yl)amino]methyl}pyridin-2-yl)piperazin-1-yl]ethan-1-one
N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-6-[4-(2-methylpropyl)benzoyl]-6-azaspiro[2.5]octane-1-carboxamide
8-[(4-phenyl-1,3-thiazol-2-yl)methyl]-1,3-dioxa-8-azaspiro[4.5]decan-2-one
3-[(dimethylamino)methyl]-1-{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}pyrrolidin-3-ol
4-[(4-fluorophenyl)methyl]-1-(2-methoxy-4-methyl-1,3-thiazole-5-carbonyl)piperidine
1-[(6-methoxy-1H-1,3-benzodiazol-2-yl)methyl]-5-oxopyrrolidine-3-carboxylic acid
N-(1-{5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-methyl-4H-1,2,4-triazol-3-yl}-2-phenylethyl)-2,4-dimethoxybenzamide
N-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-N,1-dimethylpyrrolidin-3-amine
1-[3-ethyl-3-(hydroxymethyl)piperidin-1-yl]-2-(4-phenylpiperidin-1-yl)ethan-1-one
4-(furan-3-ylmethyl)-7-(2-methylphenyl)-9-(oxolan-3-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-[1-(2,3-dihydro-1-benzofuran-5-carbonyl)piperidin-3-yl]-1H-1,3-benzodiazole
1,5-dimethyl-N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-N-(pyridin-3-ylmethyl)-1H-indole-2-carboxamide
1-{4-[(1R,5S)-3,8-diazabicyclo[3.2.1]octan-3-yl]-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
4-{3-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]piperidine-1-carbonyl}-N,N-dimethylaniline
2-{1-cyclohexyl-5-[(1,1-dioxo-1λ6-thian-4-yl)methyl]-1H-1,2,4-triazol-3-yl}acetamide
2-[3-(1H-pyrazol-3-yl)phenyl]-3-(pyrrolidine-1-carbonyl)pyridine
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-[(1-methyl-1H-imidazol-5-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
4-ethyl-1-[(2-phenyl-1,3-thiazol-4-yl)methyl]-3-(piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
(2S,4R)-4-({[4-(benzyloxy)phenyl]methyl}amino)-1-(2,3-dihydro-1H-inden-2-yl)-N-methylpyrrolidine-2-carboxamide
(3aS,6aR)-3-[2-(3-chlorophenyl)ethyl]-5-(2-cyclopropylacetyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
5-{[5-(oxolan-3-yl)-4-phenyl-1H-imidazol-1-yl]methyl}-2-(trifluoromethyl)pyridine
(2E)-3-(3-fluorophenyl)-N-{[4-methoxy-3-(pyridin-3-ylmethoxy)phenyl]methyl}-N-[(3S)-2-oxoazepan-3-yl]prop-2-enamide
2-[ethyl({[(3R,4R)-4-(hydroxymethyl)-1-[3-(pyridin-2-yl)-1H-pyrazole-5-carbonyl]pyrrolidin-3-yl]methyl})amino]ethan-1-ol
(3aS,6aR)-3-[3-(4-fluorophenyl)propyl]-5-(4-methyl-1H-imidazole-2-carbonyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
1-[5-(7-{[4-(propan-2-yl)phenyl]methyl}-2,7-diazaspiro[4.5]decane-2-carbonyl)-1H-pyrazol-3-yl]ethan-1-one
(3S,4S)-1-[6-methyl-2-(pyridin-3-yl)pyrimidin-4-yl]-4-(4-methylpiperazin-1-yl)pyrrolidin-3-ol
4-(2-chloropyridine-4-carbonyl)-7-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-{4-[4-(2-methylphenoxy)piperidin-1-yl]-4-oxobutyl}pyrrolidin-2-one
3-(2,5-dioxoimidazolidin-4-yl)-N-[(3-phenylphenyl)methyl]propanamide
N-(4-fluorophenyl)-3-[(3S,4R)-4-(morpholin-4-yl)-1-(naphthalen-1-ylmethyl)piperidin-3-yl]propanamide
1-(3-methoxypropyl)-8-(2-methylpropyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-[methyl({5-[4-(2-phenylethyl)piperidine-1-carbonyl]pyridin-2-yl})amino]propan-1-ol
3-(dimethyl-1,2-oxazol-4-yl)-1-[4-(2,6-dimethylpyridin-4-yl)piperazin-1-yl]propan-1-one
(1R,9aR)-1-{[4-(furan-2-carbonyl)-1,4-diazepan-1-yl]methyl}-octahydro-1H-quinolizin-1-ol
2-[(1S,5R)-6-[(5-cyclopentylthiophen-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N,N-dimethylacetamide
2-[1-(1-benzyl-4-phenylpiperidin-4-yl)-N-methylformamido]acetic acid
N-(cyclohex-1-en-1-ylmethyl)-1-methyl-2-oxo-1,2,5,6,7,8-hexahydroquinoline-3-carboxamide
1-(4-phenylazepan-1-yl)-2-{2-[(4-phenylpiperazin-1-yl)methyl]-4-(pyrimidin-2-yl)phenoxy}ethan-1-one
(furan-2-ylmethyl)({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})(pyridin-2-ylmethyl)amine
1-{[3-(3-fluorophenyl)oxolan-3-yl]methyl}-4-(3-methylpyridin-4-yl)piperazine
2-{[(3-ethoxyphenyl)methyl](quinolin-2-ylmethyl)amino}ethan-1-ol
4-[6-(4-fluorophenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]piperazin-2-one
1-[2-(2-phenylethyl)morpholin-4-yl]-3-(1H-1,2,4-triazol-1-yl)propan-1-one
N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}-2-(pyrrolidin-3-yl)benzamide