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(1-methyl-1H-imidazol-2-yl)[1-(pyridin-4-ylmethyl)piperidin-4-yl]methanol
dimethyl(2-{2-[1-(1-methyl-1H-indole-3-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}ethyl)amine
1-[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]propan-2-ol
1-{2-[5-(1H-imidazol-2-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}piperidine-3-carboxamide
N-[2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)ethyl]-N-methyl-1-(oxan-4-yl)piperidine-3-carboxamide
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-1H-pyrrole-2-carboxamide
2-(2-ethyl-4-methyl-1H-imidazol-5-yl)-5-(1H-1,2,3,4-tetrazol-1-yl)-1H-1,3-benzodiazole
4-(2-chlorophenoxy)-1-(1H-1,2,4-triazole-5-carbonyl)piperidine
4-(1-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}piperidin-3-yl)-5-(4-methylphenyl)pyrimidine
4-[(1E)-1-(furan-2-yl)prop-1-en-2-yl]-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N-{1-[2-(4-methoxyphenyl)ethyl]-5-oxopyrrolidin-3-yl}-2-(methylsulfanyl)pyridine-3-carboxamide
N-[3-(furan-2-yl)phenyl]-4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazine-1-carboxamide
7-(2-hydroxyethyl)-2-[3-(1H-indol-3-yl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one
4-ethyl-3-[(1-{6-methyl-2H-[1,3]dioxolo[4,5-g]quinolin-8-yl}piperidin-4-yl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
2-{3-[(1E)-pent-1-en-1-yl]-1H-1,2,4-triazol-5-yl}pyridine
5-[1-(cyclohexylmethyl)-4-hydroxypiperidin-4-yl]-N-(2,5-dimethoxyphenyl)-1-benzofuran-2-carboxamide
1-(3-chloro-4-fluorophenyl)-5-(2-methanesulfonylethyl)-1H-1,2,4-triazole
{[2-chloro-5-ethoxy-4-(propan-2-yloxy)phenyl]methyl}[(6-chloropyridin-3-yl)methyl]amine
(2S,4R)-4-[(4-fluorophenyl)sulfanyl]-1-[(4-methoxy-2,5-dimethylphenyl)methyl]-N,N-dimethylpyrrolidine-2-carboxamide
N-(3,5-dimethylphenyl)-N'-[(1S,2S)-2-hydroxycyclohexyl]propanediamide
1-(4-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-2-ethoxyethan-1-one
1,4-dimethyl-9-{[5-(oxolan-2-yl)thiophen-2-yl]methyl}-1,4,9-triazaspiro[5.5]undecane
5-methyl-1-(4-methylphenyl)-4-(1,2-oxazole-3-carbonyl)piperazin-2-one
N-(1-{1-[2-(3-methoxyphenyl)acetyl]piperidin-4-yl}-1H-pyrazol-5-yl)oxolane-3-carboxamide
N-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-3-(3-methoxyphenyl)-1H-pyrazole-4-carboxamide
N-{2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}piperidin-3-amine
4,4-difluoro-1-{5-methylpyrazolo[1,5-a]pyrimidin-7-yl}piperidine
{[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]amine
N-[3-(piperidin-1-ylmethyl)phenyl]-4-(pyrimidin-2-yl)piperazine-1-carboxamide
1-{4-[4-chloro-2-(thiomorpholine-4-carbonyl)phenoxy]piperidin-1-yl}ethan-1-one
(4aS,8aR)-6-(2,5-dimethylfuran-3-carbonyl)-1-[2-(1H-imidazol-4-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
2-(adamantan-1-yl)-N-[2-(1H-pyrazol-1-yl)ethyl]acetamide
1-{4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-3-(methylsulfanyl)propan-1-one
2-ethoxy-N-{1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl}pyridine-3-carboxamide
N-[1-(2-phenylethyl)piperidin-3-yl]-4-(1H-1,2,4-triazol-1-yl)butanamide
N-{[7-(1,5-dimethyl-1H-pyrazole-3-carbonyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-2-(thiophen-3-yl)acetamide
N-(furan-3-ylmethyl)-N-methyl-5-{1-[(5-methyl-1H-pyrazol-3-yl)methyl]pyrrolidin-2-yl}thiophene-2-carboxamide
ethyl 4-(5-acetylthiophene-3-carbonyl)piperazine-1-carboxylate
9-(5-chloro-6-oxo-1,6-dihydropyridine-3-carbonyl)-2-(3-methoxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
1-[(2-fluoro-4-methylphenyl)methyl]-3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
(1-{[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}piperidin-4-yl)(pyridin-2-yl)methanol
3-(3-hydroxy-1,2-oxazol-5-yl)-1-[2-methyl-4-(pyrrolidin-1-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]propan-1-one
3-[3-(dimethylamino)propyl]-8-[(1-ethyl-1H-pyrazol-4-yl)methyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-(3-ethoxy-2-hydroxypropyl)-1-[(4-methylphenyl)amino]cyclopentane-1-carboxamide
[(1-cyclopentylpiperidin-4-yl)methyl](oxolan-2-ylmethyl)(2-phenylethyl)amine
7-(2-methylphenyl)-4-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-[(1-methylpyrrolidin-3-yl)methyl]-2-[(quinolin-8-yloxy)methyl]-1,3-oxazole-4-carboxamide
N-ethyl-N-[2-(4-methoxyphenoxy)ethyl]-1-methylpiperidine-3-carboxamide
[1-(3-{1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-1H-1,2,3-triazol-4-yl}phenyl)ethyl]dimethylamine
4-{2-[5-(2H-1,3-benzodioxol-5-ylmethyl)-5-methyl-2-oxopiperidin-1-yl]ethyl}piperazin-2-one