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1-benzyl-5-[(4-methylphenyl)methyl]-N-(1,3-thiazol-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
5-[4-(4-fluorophenyl)-1,2,3,6-tetrahydropyridine-1-carbonyl]-4,6-dimethyl-1,2,3,4-tetrahydropyrimidin-2-one
2-amino-3-ethyl-N-[(4-hydroxyphenyl)methyl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
(1R,7S)-3-(4-fluorophenyl)-N-methyl-4-oxo-N-[3-(1H-pyrazol-1-yl)propyl]-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
1-{6-[3-(hydroxymethyl)-3-[(2-methylphenyl)methyl]piperidin-1-yl]pyridin-3-yl}ethan-1-one
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-[1-(2-methoxypyridine-3-carbonyl)piperidin-3-yl]piperazine
5-(2-fluorophenoxymethyl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-(propan-2-yl)-1H-pyrazole-3-carboxamide
2,7,8-trimethyl-4-[2-(5-methyl-1,2-oxazol-3-yl)piperidine-1-carbonyl]quinoline
1-(6-aminopyrimidin-4-yl)-3-[(2-fluorophenyl)methyl]piperidine-3-carboxylic acid
3-{2-[4-(2-fluorophenyl)piperazin-1-yl]-2-oxoethyl}-4-(3-methylbutyl)piperazin-2-one
1-(furan-3-carbonyl)-4-[3-(trifluoromethyl)phenoxy]piperidine
1-[(2S)-1-benzylpyrrolidine-2-carbonyl]-4-(1H-imidazol-2-yl)piperidine
1-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-4-ethyl-3-(piperidin-4-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
4-[(2,6-difluorophenyl)methyl]-1-phenylpiperazin-2-one
{[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}[1-(pyridin-4-yl)propyl]amine
2-(dimethylamino)-2-(3-methylphenyl)-N-[2-(pyridin-3-yl)ethyl]acetamide
[(1-cyclopentylpiperidin-4-yl)methyl]({[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl})(oxolan-2-ylmethyl)amine
2-(4-{[3-(1-benzofuran-2-yl)-1H-pyrazol-4-yl]methyl}piperazin-1-yl)-1,3-benzoxazole
2-amino-3-ethyl-N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
3-{3-methyl-5-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-1-yl}-1λ6-thiolane-1,1-dione
2-(morpholin-4-yl)-N-{[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]methyl}-2-(pyridin-3-yl)acetamide
N-butyl-N,1-dimethyl-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-[(2-ethyl-7-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)methyl]-4-methoxyphenol
1-({[3-(piperidine-1-carbonyl)-1-propyl-4,5,6,7-tetrahydro-1H-indazol-5-yl]amino}methyl)cyclohexan-1-ol
1-[2-(methylsulfanyl)acetyl]-4-(naphthalen-2-ylmethyl)-1,4-diazepan-5-one
5-cyclopropyl-1-[4-(2,5-dimethoxyphenyl)pyrimidin-2-yl]-N-[3-(morpholin-4-yl)propyl]-1H-pyrazole-4-carboxamide
2-(4-{[3-(2-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}piperazin-1-yl)pyrimidine
1-(4-amino-5-cyanopyrimidin-2-yl)-4-(4-fluorophenoxy)piperidine-4-carboxylic acid
(butan-2-yl)[(6-chloropyridin-3-yl)methyl](pyridin-3-ylmethyl)amine
3-{[3-(4-phenylphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}pyridine
4-(4-methylphenoxy)-1-(6-oxo-1,6-dihydropyridine-3-carbonyl)piperidine-4-carboxylic acid
2-(2-hydroxyethyl)-6-[2-(pyridin-3-yl)pyrimidine-5-carbonyl]-1H,2H,3H,4H,5H,6H,7H-pyrazolo[3,4-c]pyridin-3-one
N-ethyl-N-methyl-3-oxo-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecane-9-sulfonamide
2-({3-[4-(4-chlorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)-6-ethoxyphenol
1-[(2-chlorophenyl)methyl]-4-(1-ethyl-1H-1,2,4-triazol-5-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
2-[(4aR,7aS)-4-[(5-methylthiophen-2-yl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]acetic acid
(3R,5S)-N3-(2,3-dihydro-1H-inden-5-yl)-N5-[(2-methoxyphenyl)methyl]-1-(2-phenylethyl)piperidine-3,5-dicarboxamide
methyl 1-[(3R,5S)-1-[(3,4-difluorophenyl)methyl]-5-[(diphenylmethyl)carbamoyl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
3-[(3R,4R)-4-cyclopropyl-4-hydroxy-3-methylpiperidine-1-carbonyl]-1H,2H,5H,6H,7H-cyclopenta[b]pyridin-2-one
2-methoxy-N-[1-(6-methoxynaphthalen-2-yl)ethyl]-2-methylpropanamide
1-{[7-fluoro-2-(4-methylphenyl)quinolin-3-yl]methyl}-N-methylpyrrolidine-3-carboxamide
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-2-[3-oxo-1-(thiophen-2-ylmethyl)piperazin-2-yl]acetamide
N,N-diethyl-3-[({[3-(1H-pyrazol-1-yl)phenyl]methyl}amino)methyl]pyridin-2-amine
3-[(1-cyclopentyl-1H-imidazol-5-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[(3R,4S)-1-acetyl-4-cyclopropylpyrrolidin-3-yl]-4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzamide
1-{4-[3-({[(3-ethoxyphenyl)methyl]amino}methyl)pyridin-2-yl]piperazin-1-yl}ethan-1-one
1-(2-methoxyethyl)-8-[(1-methyl-1H-indol-3-yl)methyl]-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-[5-chloro-2-(piperidine-1-carbonyl)phenoxy]-1-[(4-methyl-1H-imidazol-2-yl)methyl]piperidine
8-[3-(2,4-difluorophenyl)propanoyl]-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-2-(phenylamino)pyrimidine-5-carboxamide