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2-[(3-fluorophenyl)methyl]-4-[2-(1H-imidazol-2-yl)benzoyl]morpholine
{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}(methyl)(thiophen-3-ylmethyl)amine
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-N,2,4-trimethyl-1,3-thiazole-5-carboxamide
6,7-dimethoxy-2-[1-(3-methylbutyl)piperidin-3-yl]-1,2,3,4-tetrahydroisoquinoline
ethyl 1-[(4-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-2-oxo-6-(propan-2-yl)-1,2-dihydropyridine-3-carboxamide
4-[3-(cyclopropylcarbamoyl)piperidin-1-yl]-N-phenylpiperidine-1-carboxamide
ethyl 1-[3-(dimethyl-1,2-oxazol-4-yl)propanoyl]-3-[(2E)-3-phenylprop-2-en-1-yl]piperidine-3-carboxylate
2-chloro-N-{1-oxa-8-azaspiro[4.5]decan-3-yl}-5-(trifluoromethyl)benzamide
3-methyl-N-propyl-4-[({[1-(1H-pyrazol-1-ylmethyl)cyclopropyl]methyl}carbamoyl)amino]benzamide
2-[(1E)-2,6-dimethylhepta-1,5-dien-1-yl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
1-(2-methylpropyl)-3-(pyridin-2-ylmethyl)-8-(1,3-thiazol-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-{1-[(5-methylfuran-2-yl)methyl]-4-{[2-(2-methylphenyl)pyrimidin-5-yl]methyl}piperazin-2-yl}ethan-1-ol
3-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-1-[3-(5-ethyl-4H-1,2,4-triazol-3-yl)phenyl]urea
(R)-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl](phenyl)methanol
3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)-1-[4-(pyrimidin-2-yl)-1,4-diazepan-1-yl]propan-1-one
2-(2-aminopyrimidin-5-yl)-N-cyclohexyl-N-ethyl-8-methylquinoline-4-carboxamide
1-[(3R,5S)-3-[(dimethylamino)methyl]-5-(hydroxymethyl)piperidin-1-yl]-3-[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]propan-1-one
4-[(3aS,6aS)-octahydropyrrolo[2,3-c]pyrrole-1-carbonyl]-3-cyclohexyl-1H-pyrazole
N-{2-[5-(hydroxymethyl)-1,2,4-oxadiazol-3-yl]ethyl}-2-(1H-indol-3-yl)acetamide
N,N-dimethyl-4-(1,2,3,4-tetrahydroisoquinolin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-2-amine
1-{[5-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}-4-(pyridin-3-ylmethyl)piperazine
4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(3-phenylpropyl)piperidine
3-ethyl-8-(1H-indol-2-ylmethyl)-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)-N-[2-(1-oxo-1,2-dihydrophthalazin-2-yl)ethyl]acetamide
1-methyl-3-[1-(2-methylpropyl)-1H-pyrazol-5-yl]-1-(1,3-thiazol-2-ylmethyl)urea
N-[2-(dimethylamino)ethyl]-2-(3-methyl-1H-pyrazol-1-yl)-N-{[2-(3-methylphenyl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}acetamide
2-(4-{[4-(thiophen-3-yl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)pyrimidine
2-methyl-2-{5-[(2E)-pent-2-en-3-yl]-4-phenyl-1H-imidazol-1-yl}propane-1,3-diol
N-[2-(6-hydroxy-2-methylpyrimidin-4-yl)ethyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
4-[1-(3,4-dihydro-2H-1-benzopyran-3-carbonyl)piperidin-4-yl]thiomorpholine
N-[2-(4-chloro-1H-pyrazol-1-yl)ethyl]-1,3-dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
3-[5-(1H-indol-5-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propanoic acid
4-[(1-ethyl-1H-pyrazol-4-yl)sulfonyl]-1,9-dimethyl-1,4,9-triazaspiro[5.6]dodecan-10-one
5-{[3-(3-chlorobenzoyl)piperidin-1-yl]methyl}-N,N-dimethyl-1,3-thiazol-2-amine
1-methyl-2-(2,3,4-trimethoxy-6-methylphenyl)-1H-1,3-benzodiazole
3-(3-fluorophenyl)-N-methyl-N-[3-(1-methyl-1H-imidazol-2-yl)propyl]-1H-pyrazole-4-carboxamide
1-[3-(benzyloxy)azetidin-1-yl]-2-[4-(pyrimidin-2-yl)piperazin-1-yl]ethan-1-one
5-methyl-1-(4-methylphenyl)-4-(4-oxo-4-phenylbutyl)piperazin-2-one
1-{4-[2-(2H-1,3-benzodioxol-5-yl)-5-fluoro-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}-3-(3,5-dimethyl-1H-pyrazol-1-yl)propan-1-one
1-ethyl-5-{[2-(1H-indol-1-yl)ethyl](methyl)amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
N-ethyl-5-{[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]methyl}pyrimidin-2-amine
N-ethyl-1-(1H-imidazol-1-ylmethyl)-N-{[2-(prop-2-en-1-yloxy)phenyl]methyl}cyclopropane-1-carboxamide
N-[(3R,4S)-1-(5-chloropyridin-2-yl)-4-cyclopropylpyrrolidin-3-yl]oxane-4-carboxamide
2-ethyl-4-methyl-N-{2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}-1,3-thiazole-5-carboxamide
N-[(4-methoxypyridin-2-yl)methyl]-1-(2-methyl-6-propylpyrimidin-4-yl)piperidin-4-amine
2-methyl-6-[3-(2-methylphenoxy)azetidine-1-carbonyl]phenol
N'-(2,3-dimethylphenyl)-N-[(2S)-oxolan-2-ylmethyl]propanediamide
N,1,3-trimethyl-N-{1-[1-(6-oxo-1,4,5,6-tetrahydropyridazine-3-carbonyl)piperidin-4-yl]-2-phenylethyl}-1H-pyrazole-5-carboxamide
3-{4-[5-(pyrrolidin-1-ylmethyl)pyridin-2-yl]phenyl}propanoic acid