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N-(2,5-dimethylphenyl)-3-[4-(pyridin-3-ylmethoxy)piperidin-1-yl]propanamide
(4aS,8aR)-1-butyl-6-(2-propylpyridine-4-carbonyl)-decahydro-1,6-naphthyridin-2-one
1-{[4-chloro-2-(dimethylamino)-1,3-thiazol-5-yl]methyl}-N-phenylpiperidin-3-amine
4-{1-[1-(4-chlorobenzoyl)piperidin-4-yl]piperidine-4-carbonyl}morpholine
3-[5-(2H-1,3-benzodioxol-5-yl)-1,3,4-oxadiazol-2-yl]-1-(3-propoxypiperidin-1-yl)propan-1-one
5-ethyl-N-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]pyrazolo[1,5-a]pyrimidin-7-amine
N-methyl-N-[(4-methyl-1,3-thiazol-2-yl)methyl]-2-(2-phenylethyl)-1,3-benzoxazole-5-carboxamide
1-[(2-fluoro-5-methoxyphenyl)methyl]-4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidine
2-({4-[5-(furan-2-yl)-4-phenyl-1H-imidazol-1-yl]piperidin-1-yl}methyl)pyridine
5-(oxolan-2-yl)-N-[(2,3,6-trifluorophenyl)methyl]thiophene-2-carboxamide
methyl 2-oxo-1-(prop-2-en-1-yloxy)-8-(quinolin-4-ylmethyl)-1,8-diazaspiro[4.5]decane-4-carboxylate
methyl[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}amine
N,N-dimethyl-3-(2-phenylethyl)piperidine-1-sulfonamide
3-tert-butyl-4-[3-(4-fluorophenyl)-1H-pyrazol-4-yl]-1-methyl-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
2-{1-[(4-methoxy-3-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
1-{6-chloroimidazo[1,2-a]pyrimidine-2-carbonyl}-3-(pyrrolidin-1-yl)piperidine
{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl){[6-(pyrrolidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}amine
3-(1-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-4-phenyl-1H-imidazol-5-yl)pyridine
N-[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]-2-(phenylsulfanyl)acetamide
4-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}quinoline
1-(2-methylphenyl)-4-{[4-(pyridin-2-ylmethoxy)phenyl]methyl}piperazin-2-one
3-(4-cyano-2-ethylphenyl)-1-(3-hydroxypropyl)-1-(pyridin-3-ylmethyl)urea
1-{[5-methyl-2-(thiophen-3-yl)-1,3-oxazol-4-yl]methyl}-3-phenylpiperidine
N-(3-hydroxypropyl)-1-{1-[(4-methoxy-2,5-dimethylphenyl)methyl]piperidin-4-yl}-1H-1,2,3-triazole-4-carboxamide
N-[2-(1-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}piperidin-3-yl)ethyl]methanesulfonamide
(2S,4S)-4-amino-N-methyl-1-{4-[(pyridin-2-ylsulfanyl)methyl]benzoyl}pyrrolidine-2-carboxamide
4-({4-benzyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}methyl)-1-(propan-2-yl)piperidine
3-methyl-2-({4-[4-(pyrrolidine-1-carbonyl)phenoxy]piperidin-1-yl}methyl)-1H-indole
4-[4-(cyclohex-3-en-1-ylmethyl)piperazin-1-yl]-2-[2-(1H-pyrazol-1-yl)ethyl]-2,3-dihydro-1H-isoindole-1,3-dione
3-[(3S,4R)-1-benzyl-4-(morpholin-4-yl)piperidin-3-yl]-N-(4-methylphenyl)propanamide
N-[2-(2-oxopyrrolidin-1-yl)ethyl]-2-(N-phenylmethanesulfonamido)propanamide
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-4-yl}methyl)-2-(2-fluorophenyl)-N-methylacetamide
N-[(3R,4R)-1-(1H-1,3-benzodiazol-2-ylmethyl)-3-hydroxypiperidin-4-yl]pyridine-4-carboxamide
N-[(2R,4R,6S)-2-cyclohexyl-6-(1,3-thiazol-2-yl)oxan-4-yl]acetamide
(1R,5R)-6-[2-(3-fluoro-4-hydroxyphenyl)acetyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
1-{2,7-dimethylpyrazolo[1,5-a]pyrimidine-5-carbonyl}-3-(4-ethyl-1H-pyrazol-5-yl)piperidine
methyl 3-(oxane-4-carbonyl)-7-oxo-9-(3-phenylpropoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-(2-methoxyethyl)-6-[3-(piperidin-1-ylmethyl)piperidin-1-yl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
3-[1-({5-methylpyrazolo[1,5-a]pyrimidin-7-yl}amino)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
{6-[4-(1-benzyl-1H-imidazol-2-yl)piperidine-1-carbonyl]pyridin-2-yl}methanol
1-methyl-N-[2-(morpholin-4-yl)ethyl]-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-[(1-methyl-1H-imidazol-2-yl)methyl]-3-(thiomorpholine-4-carbonyl)benzene-1-sulfonamide
ethyl 1-[(2S)-2-acetamido-4-(methylsulfanyl)butanoyl]-4-[(4-methoxyphenyl)methyl]piperidine-4-carboxylate
3-{[4-(hydroxymethyl)oxan-4-yl]methyl}-3-methyl-1-{3-[(2-methylprop-2-en-1-yl)oxy]phenyl}urea
1-[(3-cyclopropyl-1-phenyl-1H-1,2,4-triazol-5-yl)methyl]-4-phenylpyrrolidin-2-one
3-[({[4-(dimethylamino)oxan-4-yl]methyl}amino)methyl]-1-(2,2-dimethylpropyl)-3-hydroxypiperidin-2-one
(1R,2S,9R)-11-[6-(pyrrolidine-1-carbonyl)pyrazin-2-yl]-7,11-diazatricyclo[7.3.1.02,7]tridecan-6-one
(2S)-1-[2-(4-butanamidophenyl)acetyl]pyrrolidine-2-carboxamide
ethyl 4-[(8-chloro-4-hydroxyquinolin-2-yl)methyl]piperazine-1-carboxylate
1-methyl-4-{[5-(4-phenyl-1H-imidazol-5-yl)-1,2,4-oxadiazol-3-yl]methyl}piperidine