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N-[2-(dimethylsulfamoyl)ethyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
1-hydroxy-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}naphthalene-2-carboxamide
1-[2-(4-methoxyphenyl)ethyl]-8-[(4-methoxyphenyl)methyl]-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-{2-[(2,3-dimethoxyphenyl)formamido]ethyl}-N-(2-methylpropyl)-1H-1,2,3-triazole-4-carboxamide
1-[2-(1H-imidazol-2-yl)benzoyl]-4-(3-methylpyridin-4-yl)-1,4-diazepane
1-[(3R,4S)-4-hydroxy-3,4-dimethylpiperidin-1-yl]-3-(morpholin-4-yl)propan-1-one
7-{[5-chloro-1-methyl-3-(5-methyl-1,2-oxazol-3-yl)-1H-pyrazol-4-yl]methyl}-2-oxa-7-azaspiro[4.5]decane
[(5,6-dimethyl-1H-1,3-benzodiazol-2-yl)methyl](methyl){[5-methyl-2-(thiophen-3-yl)-1,3-oxazol-4-yl]methyl}amine
N-(1-methyl-1H-1,2,3-triazol-4-yl)-1-(3-phenylphenyl)piperidin-4-amine
N2,N2,N4-trimethyl-N4-{[3-(thiophen-2-yl)-1H-pyrazol-5-yl]methyl}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-2,4-diamine
(2S,4R)-4-amino-N-cyclopentyl-N-(prop-2-en-1-yl)pyrrolidine-2-carboxamide
4-(3-methylphenoxy)-1-[3-(1H-pyrrol-1-yl)propanoyl]piperidine-4-carboxylic acid
1-methyl-3-(3-methyl-1,2,4-thiadiazol-5-yl)-1-(oxan-4-yl)urea
N,2-dimethyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-1,3-thiazole-5-carboxamide
N-[(2-ethoxypyridin-3-yl)methyl]-2,2-dimethyloxane-4-carboxamide
3-[4-(2,6-difluorophenyl)-1H-pyrazol-5-yl]-1-[(2,3-difluorophenyl)methyl]piperidine
1-[(5-{[2-(dimethylamino)pyrimidin-5-yl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)methyl]-3,3-dimethylurea
5-(1-benzofuran-2-yl)pyridine-2-carbonitrile
6-[(diethylamino)methyl]-N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
1-{[2-(difluoromethoxy)phenyl]methyl}-4-(hydroxymethyl)azepan-4-ol
1-{2-[(4,4-difluoropiperidin-1-yl)methyl]phenoxy}-3-(piperidin-1-yl)propan-2-ol
1-(3-{3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl}-3-oxopropyl)pyrrolidin-2-one
2-(6-methoxynaphthalen-2-yl)-4-(pyridin-3-ylmethyl)morpholine
3-{5-[2-(1H-indol-3-yl)ethyl]-1,3,4-oxadiazol-2-yl}-N-(2-methoxyethyl)-N-(propan-2-yl)propanamide
N-benzyl-2-{[3-(pyridin-3-yl)-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]sulfanyl}acetamide
2-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
3-[4-(3-hydroxyphenyl)piperidine-1-carbonyl]piperidine-1-carboxamide
N-[2-(2-chlorophenyl)-2-hydroxyethyl]-1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
(2S,4R)-4-amino-1-(1,4-dithiepan-6-yl)-N-methylpyrrolidine-2-carboxamide
2-[(furan-2-ylmethyl)({[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl})amino]butan-1-ol
2-[4-(2-aminopyrimidin-4-yl)-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl]ethan-1-ol
4-[({imidazo[1,2-a]pyridin-3-ylmethyl}(methyl)amino)methyl]-N-(6-methylpyridazin-3-yl)benzamide
9-methoxy-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-3-{2-[4-(methylsulfanyl)phenyl]acetyl}-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
4-(dimethylamino)-N,N-dimethyl-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-sulfonamide
({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)(isoquinolin-5-ylmethyl)methylamine
13-(4-methoxy-2,5-dimethylphenyl)-5-thia-2,7,10-triazatricyclo[6.5.0.02,6]trideca-1(8),3,6-trien-11-one
3-(2-fluorophenyl)-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-1H-pyrazole-5-carboxamide
N-{[1-(furan-2-ylmethyl)piperidin-3-yl]methyl}-1,5-dimethyl-1H-pyrazole-4-carboxamide
5-[3-(2,3-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]-N-methyl-N-(1,2-oxazol-3-ylmethyl)pyridin-2-amine
2-(1-methyl-1H-imidazol-2-yl)-1-(2-{[(4-methyl-1H-imidazol-5-yl)methyl]sulfanyl}ethyl)-1H-imidazole
1-{2-[(6-methylpyridin-2-yl)methyl]-2,7-diazaspiro[4.5]decan-7-yl}-2-phenoxyethan-1-one
N-[(1-methylpiperidin-4-yl)methyl]-2,7-dioxo-N-(2-phenylethyl)-1,3-diazepane-4-carboxamide
3-[4-(2,6-difluorophenyl)-1H-pyrazol-5-yl]-1-[(2,4-dimethoxyphenyl)methyl]piperidine
1-[6-(3-fluorophenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]azocane
methyl 1-({4-[3-(1,3-benzothiazol-2-yl)propanoyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)piperidine-4-carboxylate
2-ethoxy-1-{4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}ethan-1-one
(3aS,7aR)-5-methyl-2-(5-oxo-1-phenyl-2,5-dihydro-1H-pyrazole-3-carbonyl)-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
3-[4-(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-8-fluoro-1,4-dihydroquinolin-4-one
5-[(2-chloro-3-hydroxy-4-methoxyphenyl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylic acid
3-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}-3H,4H-thieno[3,2-d]pyrimidin-4-one