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4-(5-{[1-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl)pyridine
3-[1-(2,1,3-benzothiadiazol-5-ylmethyl)piperidin-3-yl]-N-[(2-chlorophenyl)methyl]propanamide
2-(morpholin-3-yl)-N-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]acetamide
3-(2-chlorophenyl)-6-[3-(2-methyl-1H-imidazol-1-yl)propanoyl]-1-(pyridin-4-ylmethyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
5-(propan-2-yl)-N-[2-(pyridin-3-yl)ethyl]-1-[4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
3-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepane-1-carbonyl}-1-methyl-1,2-dihydropyridin-2-one
N-(1,3-benzoxazol-2-ylmethyl)-2-cyclopropyl-N-methyl-1,3-benzoxazole-6-carboxamide
N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}-4-propylbenzamide
[(3R,4S)-1-[(2-methoxy-4-methylphenyl)methyl]-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-3-yl]methanol
4-methoxy-N-{[1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)piperidin-3-yl]methyl}benzene-1-sulfonamide
N-[(3-methylphenyl)methyl]-10-oxo-3,9-diazaspiro[5.6]dodecane-3-carboxamide
1-[6-(2-chlorophenyl)-8-oxo-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carbonyl]piperidine-3-carbonitrile
1-{2-ethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}-4-(2-methoxybenzoyl)piperazine
1-[(1S,5R)-6-(5-methoxy-3-methyl-1H-indole-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
4-{4-[5-(hydroxymethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidine-5-carboxylic acid
8-[(1-methyl-1H-indol-3-yl)methyl]-1-(2-methylpropyl)-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(1-cyclopentyl-4-{[4-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)ethan-1-ol
3-{imidazo[1,2-a]pyridin-2-yl}-1-[3-(pyridin-2-yl)azetidin-1-yl]propan-1-one
4-[3-(2-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-2-(methylsulfanyl)-1,3-thiazole
3-butyl-1-methyl-4-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}piperazin-2-one
2-{5-cyclopropyl-1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-1H-pyrazole-4-carbonyl}-2-azabicyclo[2.2.1]heptane
1-[(4-chlorophenyl)methyl]-N-[2-methyl-2-(morpholin-4-yl)propyl]-6-oxopiperidine-3-carboxamide
5-(2-chloro-6-methoxyphenyl)-2-methyl-1,3-benzoxazole
{[1-butyl-2-(4-methylpentanesulfonyl)-1H-imidazol-5-yl]methyl}(methyl)[(1-methyl-1H-imidazol-2-yl)methyl]amine
4-[4-(pyrimidin-2-yl)-1,4-diazepane-1-carbonyl]-1,2-dihydroquinolin-2-one
(3S,4S)-1-(4-chloro-3-fluorobenzoyl)-4-{methyl[(4-methyl-1H-imidazol-2-yl)methyl]amino}pyrrolidin-3-ol
(2S,4S)-4-({[4-(benzyloxy)phenyl]methyl}amino)-1-[(4-chlorophenyl)methyl]-N-(2-methoxyethyl)pyrrolidine-2-carboxamide
3-fluoro-2-{3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridine
4-(3-hydroxy-3-methylbutyl)-N-[(1-methylpiperidin-2-yl)methyl]benzamide
3-({[(2-aminopyrimidin-5-yl)methyl](methyl)carbamoyl}amino)-N-(2-methoxyethyl)-2-methylbenzamide
[2-(2-ethoxyphenoxy)ethyl](furan-3-ylmethyl)methylamine
3-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}quinoline
2-amino-6-tert-butyl-4-[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]pyridine-3-carbonitrile
1-methyl-4-(2-{[(2-methylphenyl)methyl]sulfanyl}acetyl)-1,4,9-triazaspiro[5.6]dodecan-10-one
N-ethyl-N-[(1-methylpyrrolidin-3-yl)methyl]-5-(morpholin-4-ylmethyl)-1,2-oxazole-3-carboxamide
5,6-dimethyl-2-{2-[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-oxoethyl}-2,3-dihydropyridazin-3-one
N-(4-{[(prop-2-en-1-yl)(pyridin-2-ylmethyl)carbamoyl]methoxy}phenyl)propanamide
2-[(2R,3S,6R)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pyridine-4-carboxamide
1-[(5-fluoro-1-methyl-1H-indol-2-yl)methyl]-N-methylpiperidine-2-carboxamide
4-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidine-1-carbonyl}pyridin-2-amine
1-(2-aminopyrimidin-4-yl)-4-(quinolin-6-yloxy)piperidine-4-carboxylic acid
2-{2-[2-(furan-2-yl)azepan-1-yl]-2-oxoethyl}-1,2-dihydrophthalazin-1-one
2-ethoxy-6-{[4-(3-fluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}phenol
5-[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]-N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]pyridin-2-amine
[2-(6-methyl-2-propylpyrimidin-4-yl)phenyl]methanol
2-ethyl-N-[2-(1H-imidazol-1-yl)-1-phenylethyl]-4-methyl-1,3-oxazole-5-carboxamide
4-(2H-1,3-benzodioxol-5-ylmethyl)-7-chloro-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepine
3-(4-methyl-1,3-thiazol-5-yl)-N-{[5-methyl-2-(trifluoromethyl)furan-3-yl]methyl}propanamide
5-(1-cyclopentanecarbonylpiperidin-4-yl)-5-(pyridin-3-yl)-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
methyl({[4-(1H-pyrazol-1-yl)phenyl]methyl}){[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}amine