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3-{3-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]piperidin-1-yl}propanamide
3-[(4-ethylpiperazin-1-yl)methyl]-1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxypiperidin-2-one
3-[(dimethylamino)methyl]-1-(1-phenylcyclopropanecarbonyl)pyrrolidin-3-ol
5-(dimethylamino)-2-{2-[2-(3-fluorophenyl)piperidin-1-yl]-2-oxoethyl}-2,3-dihydropyridazin-3-one
3-(2H-1,3-benzodioxol-5-yl)-N,N-dimethyl-3-phenylpropanamide
N-[(1-benzyl-1H-pyrazol-4-yl)methyl]-2-(4-methyl-1,2,5-oxadiazol-3-yl)acetamide
2-acetamido-N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(pyridin-3-ylmethyl)acetamide
ethyl 3-(2-phenoxyethyl)-1-[3-(1H-pyrazol-1-yl)propanoyl]piperidine-3-carboxylate
2-methyl-5-(4-{[3-(5-methylfuran-2-yl)phenyl]methyl}piperazin-1-yl)-2,3-dihydropyridazin-3-one
1-{4-[(3-fluorophenyl)methyl]piperazin-1-yl}-2-(morpholin-3-yl)ethan-1-one
N-cyclopentyl-6-hydroxy-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)pyridine-3-carboxamide
2-(dimethylamino)-7-(1-ethyl-5-methyl-1H-pyrazole-4-carbonyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-propyl-3-(1H-pyrazol-4-yl)propanamide
4-[2-(1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}piperidin-2-yl)ethyl]phenol
1-butyl-3-{2-[3-(methoxymethyl)piperidin-1-yl]-2-oxoethyl}-2-methyl-4,5,6,7-tetrahydro-1H-indol-4-one
(4aS,7aR)-1-(3-aminopropanoyl)-4-(pyridin-4-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[3-(2-oxo-1,3-oxazolidin-3-yl)phenyl]-3-[2-(2-oxoimidazolidin-1-yl)ethyl]urea
methyl (2S,4S)-1-methyl-4-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)benzamido]pyrrolidine-2-carboxylate
3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)-N-[(1R)-1-(3-methoxyphenyl)ethyl]propanamide
1-[2-methyl-7-(1-methyl-1H-pyrazole-4-carbonyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]piperidine
3-[(2R,3R,6R)-5-(3,5-dimethylbenzoyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
1-(2-aminoethyl)-N-{[5-(4-methoxyphenyl)-1,2-oxazol-3-yl]methyl}-1H-1,2,3-triazole-4-carboxamide
N-methyl-4-[3-(phenoxymethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]pyridin-2-amine
1-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-2-[2-(thiophen-2-yl)ethyl]piperidine
N-[2-(4-ethylphenyl)ethyl]-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
1-[3-(2-propyl-1H-imidazol-1-yl)phenyl]ethan-1-ol
1-[4-(5,6-dimethylpyrimidin-4-yl)piperazin-1-yl]-2-(1-propylpiperidin-4-yl)ethan-1-one
8-[2-(methylsulfanyl)propanoyl]-2-(3-phenylpropyl)-2,8-diazaspiro[4.5]decan-3-one
1-[2-methyl-2-(morpholin-4-yl)propyl]-4-(pyridin-4-yl)-1,4-diazepan-6-ol
4-{4-[(propan-2-yl)carbamoyl]pyridin-2-yl}piperazine-2-carboxylic acid
(4S)-4-(methoxymethyl)-3,3-dimethyl-1-{[2-(methylsulfanyl)phenyl]methyl}piperidin-4-ol
5-{3,7-dimethyl-3,7,11-triazaspiro[5.6]dodecane-11-carbonyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-(2-{[4-(2-fluorophenyl)piperazin-1-yl]methyl}-1,3-oxazole-4-carbonyl)pyrrolidin-3-amine
2-[(4-benzylpiperazin-1-yl)methyl]-N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-1,3-oxazole-4-carboxamide
1-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)-3-(pyrrolidine-1-carbonyl)piperazine
3-methoxy-1-[4-(2-methoxyphenoxy)piperidin-1-yl]propan-1-one
2-oxo-N-[4-(oxolan-2-ylmethoxy)phenyl]-1-oxa-3,8-diazaspiro[4.5]decane-8-carboxamide
N-(1-{6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}pyrrolidin-3-yl)acetamide
1-methyl-3,8-bis(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-(1-methyl-1H-pyrazol-4-yl)-N-[1-(5,6,7,8-tetrahydronaphthalen-2-yl)ethyl]propanamide
N-cyclohexyl-N-(pyridin-3-ylmethyl)-3-(trimethyl-1H-pyrazol-4-yl)propanamide
N-[(3S,5S)-1-cycloheptyl-5-(ethylcarbamoyl)pyrrolidin-3-yl]-2-methylpyrimidine-5-carboxamide
3-[(1-{imidazo[1,2-a]pyrimidin-2-yl}propyl)sulfamoyl]-N-propylbenzamide
1,3-dimethyl-5-{[3-(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}imidazolidine-2,4-dione
(3aR,6aR)-2-cyclopentyl-N-(oxan-4-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
methyl 4-{methyl[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]carbamoyl}butanoate
1-{2-[2-(dimethylamino)ethyl]morpholin-4-yl}-2-(phenylsulfanyl)ethan-1-one
3,5-dichloro-N-[1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]-4-methylbenzamide
5-[(2R,3R,6R)-3-(2-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]-2,3-dihydro-1H-pyrazol-3-one
7-(cyclopropylmethyl)-2-[3-(2-oxo-1,2-dihydropyridin-1-yl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one