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1-(2-aminoethyl)-N-[1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-yl]-1H-1,2,3-triazole-4-carboxamide
1-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-4-{[1,2,4]triazolo[4,3-a]pyrimidin-5-yl}piperazine
4-methyl-2-{1-[2-(7-methyl-2,3-dihydro-1,4-benzodioxin-6-yl)-1H-imidazol-1-yl]ethyl}-1,3-thiazole
2-{[(3-cyclohexyl-1,2,4-oxadiazol-5-yl)methyl]amino}propan-1-ol
4-{3-[(diethylamino)methyl]-4-methoxyphenyl}-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridine-3-carboxylic acid
3-{1-[(4-methoxyphenyl)methyl]-1H-1,2,4-triazol-5-yl}propanamide
N-[4-(quinolin-2-yl)-1H-pyrrolo[2,3-b]pyridin-6-yl]piperidin-4-amine
7-cyclopropanecarbonyl-N-[3-(oxolan-3-yl)propyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
1-(2H-1,3-benzodioxol-4-ylmethyl)-4-[2-(piperidine-1-carbonyl)phenoxy]piperidine
(1S,3R)-3-[2-(3,6-dioxo-1,2,3,6-tetrahydropyridazin-4-yl)acetamido]-N,N-dipropylcyclopentane-1-carboxamide
N-[(3-fluorophenyl)methyl]-2-(morpholin-4-ylmethyl)piperidine-1-carboxamide
2-(2-fluorophenyl)-1-{4-[4-(2-hydroxypropan-2-yl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}ethan-1-one
4-(2,6-dimethylpyridin-3-yl)-N-[(1-ethylpiperidin-3-yl)methyl]-N-methylpyrimidin-2-amine
N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]-5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
4-[1-(2-phenylethyl)-5-(1H-1,2,3,4-tetrazol-1-ylmethyl)-1H-1,2,4-triazol-3-yl]benzamide
3-(3-hydroxy-3-methylbutyl)-N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}benzamide
5-{3-[1-(prop-2-en-1-yl)-1H-pyrazol-3-yl]phenyl}pyrimidine
4-{[1-(2-ethoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1,3-dimethyl-1H-pyrazole
5-methyl-1-[(2-methylpyridin-4-yl)methyl]-5-phenylpiperidin-2-one
N-[(7R,8aS)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]acetamide
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-4-(4-methylpiperazine-1-carbonyl)pyridin-2-amine
3-(2H-1,3-benzodioxol-5-yl)-5-(3-methylthiophene-2-carbonyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
2-({methyl[2-(4-methyl-1,3-thiazol-5-yl)ethyl]amino}methyl)benzoic acid
N-(3-hydroxy-3-phenylpropyl)-N,4-dimethyl-2-(pyridin-3-yl)pyrimidine-5-carboxamide
(4S,4aS,8aS)-1-{[2-(methylamino)-1,3-thiazol-4-yl]methyl}-4-phenyl-decahydroquinolin-4-ol
1-[(4aS,8aR)-1-(3-hydroxypropyl)-2-oxo-decahydro-1,6-naphthyridine-6-carbonyl]cyclopropane-1-carboxamide
4-{3-[2-(2,5-dimethoxyphenyl)-1H-imidazol-1-yl]-4-methylphenyl}-4H-1,2,4-triazole
2-methyl-6-{3-[3-(4-methylpiperazin-1-yl)-3-oxopropyl]piperidine-1-carbonyl}-4H-pyran-4-one
N-(3-phenylpropyl)-5-[(quinolin-8-yloxy)methyl]-1,2-oxazole-3-carboxamide
{[2-(3,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(1H-imidazol-2-ylmethyl)methylamine
N-[2-(4-methoxyphenyl)ethyl]-N-(pyridin-2-ylmethyl)morpholine-2-carboxamide
(2R,6S)-2,6-dimethyl-4-[(3-{[3-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)methyl]morpholine
ethyl 4-[(4-chlorophenyl)methyl]-1-{[4-ethoxy-3-(hydroxymethyl)phenyl]methyl}piperidine-4-carboxylate
1-(1H-indol-2-ylmethyl)-4-(oxan-4-yl)-1,4-diazepan-6-ol
3-[(4-butyl-1H-1,2,3-triazol-1-yl)methyl]-1-(3,5-dimethyl-1H-pyrrole-2-carbonyl)piperidine
8-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-methyl-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
methyl (2S,4R)-4-(3-methoxybenzamido)-1-(naphthalen-1-ylmethyl)pyrrolidine-2-carboxylate
N-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-3-(2-oxoimidazolidin-1-yl)benzamide
3-(3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidine-1-carbonyl)benzonitrile
1-(difluoromethyl)-5-methyl-4-[4-(1H-pyrazol-1-yl)phenyl]-1H-pyrazole
4-ethyl-3-({1-[(4-ethylphenyl)methyl]piperidin-4-yl}methyl)-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
4-hydroxy-N-[4-(4-methyl-4H-1,2,4-triazol-3-yl)phenyl]-4-(pyridin-3-yl)piperidine-1-carboxamide
2-{2-[3-(4-fluorophenyl)pyrrolidin-1-yl]-2-oxoethyl}-2-azaspiro[4.5]decan-3-one
1-cyclopentyl-3-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidine
2-methyl-N-{[1-(morpholin-4-yl)cycloheptyl]methyl}-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
1-[9-(furan-2-ylmethyl)-7-(hydroxymethyl)-3,9-diazaspiro[5.5]undecan-3-yl]ethan-1-one
4-{5-[4-(dimethylamino)-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-1H-pyrazol-3-yl}phenol
[5-({[3-(1H-imidazol-1-yl)propyl](pyridin-3-ylmethyl)amino}methyl)furan-2-yl]methanol
7-chloro-2-[2-(dimethylamino)pyrimidin-5-yl]-N,N-dimethylquinoline-4-carboxamide
2-methoxy-4-[2-methoxy-4-(pyrrolidin-1-ylmethyl)phenoxy]pyridine-3-carbonitrile