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1-(4-{[(2R,5S)-5-[(3-methoxyphenyl)methyl]oxolan-2-yl]methyl}piperazin-1-yl)ethan-1-one
1-[(1-cyclohexyl-1H-1,2,4-triazol-5-yl)methyl]-5-methyl-1H-1,2,3,4-tetrazole
(2R)-2-amino-N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-4-methylpentanamide
N-methyl-5-(phenoxymethyl)-N-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}-1H-pyrazole-3-carboxamide
4-fluoro-N-{[1-(oxane-4-carbonyl)piperidin-3-yl]methyl}benzamide
N-[3-(4-chloro-1H-pyrazol-1-yl)propyl]-3-(4-methoxyphenyl)-1H-pyrazole-5-carboxamide
2-{4-[(2-fluoro-5-methoxyphenyl)methyl]-1-(2-phenylethyl)piperazin-2-yl}ethan-1-ol
4-{[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}morpholine
3-[2-(4-fluorophenyl)ethyl]-1-[(2-methyl-1,3-oxazol-4-yl)methyl]piperidine
1-(5-methoxy-2-{[methyl(1,3-thiazol-2-ylmethyl)amino]methyl}phenoxy)-3-(4-methylpiperazin-1-yl)propan-2-ol
3-[(4-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)methyl]pyridin-2-amine
(8R,9aS)-2-[2-(tert-butylsulfanyl)ethyl]-8-hydroxy-octahydro-1H-pyrido[1,2-a]piperazine-1,4-dione
7-[(4-fluorophenyl)methyl]-3-phenyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
(2S)-2-acetamido-4-methyl-N-[2-(1H-pyrazol-4-yl)ethyl]pentanamide
4-{[3-(3-methoxyphenyl)-1,2-oxazol-5-yl]methyl}-1-(oxan-4-yl)piperidin-4-ol
(4aS,8aR)-6-(6-ethyl-2-methylpyrimidin-4-yl)-1-(4-hydroxybutyl)-decahydro-1,6-naphthyridin-2-one
4-{4-[1-(2,4-dimethylphenyl)-1H-pyrazol-4-yl]-1,2,3,6-tetrahydropyridin-1-yl}butanamide
2-(4-{[4-(2-methoxyphenoxy)piperidin-1-yl]methyl}phenyl)ethan-1-amine
5-{2-[7-(cyclopropylmethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-{[7-(cyclohex-1-ene-1-carbonyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}thiophene-3-sulfonamide
4-[2-(dimethylamino)-2-(2-fluorophenyl)acetamido]-N-ethylpiperidine-1-carboxamide
(furan-2-ylmethyl)(1H-imidazol-4-ylmethyl)(thiophen-3-ylmethyl)amine
(1S,5R)-6-{[4-(methylsulfanyl)phenyl]methyl}-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
1,3-dimethyl-N-[(4-phenyloxan-4-yl)methyl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
3-({4-[2-(pyridin-2-yl)ethyl]piperazin-1-yl}methyl)piperidin-3-ol
2-(4-fluoro-2-methylphenyl)-N-methyl-N-(1,3-thiazol-2-ylmethyl)acetamide
2-{[2-(dimethylamino)-4-methylpyrimidin-5-yl]formamido}-2-(3-fluorophenyl)acetic acid
1-[(2,4-dimethyl-5-{1-[(1-methylpyrrolidin-3-yl)methyl]-1H-imidazol-2-yl}phenyl)methyl]-1H-1,2,4-triazole
N-[(dimethyl-1,3-thiazol-5-yl)methyl]-1-[(4-methylphenyl)methyl]-5-oxopyrrolidine-3-carboxamide
(3S,4R)-4-(2,3-dimethoxyphenyl)-1-[3-(methylsulfanyl)propanoyl]pyrrolidine-3-carboxylic acid
2-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)-N-[1-methyl-4-(pyridin-3-yloxy)-1H-indazol-3-yl]acetamide
N-(1-benzothiophen-2-ylmethyl)-4-[(3-methoxypropyl)amino]-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
1-[3-(2-chlorophenyl)pyrrolidin-1-yl]-2-(pyridin-2-yl)ethan-1-one
2-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-5-(pyrrolidin-1-yl)-2,3-dihydropyridazin-3-one
N-[2-(5-cyclobutyl-1,2,4-oxadiazol-3-yl)ethyl]-2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)sulfanyl]propanamide
1-(4-{[cyclopropyl(ethyl)amino]methyl}phenoxy)-3-(4-methylpiperazin-1-yl)propan-2-ol
1-{5-[3-(3-phenylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}piperazine
3-[(3R,7S,8aS)-3-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-[(1R)-1-phenylethyl]urea
3-{1-[(3-cyclohexyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}-N-[(2-fluorophenyl)methyl]propanamide
N-[3-(1H-imidazol-1-yl)-1-phenylpropyl]-2,4-dimethylpyrimidine-5-carboxamide
ethyl 4-(1-{2-[(2-chlorophenyl)methyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}piperidine-3-carbonyl)piperazine-1-carboxylate
3-{5-[(2-methoxyphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1-(pyrrolidin-1-yl)propan-1-one
2-methyl-1-[4-({5-phenyl-5H,6H,7H-pyrrolo[3,2-d]pyrimidin-2-yl}amino)piperidin-1-yl]propan-1-one
1-methyl-4-(4-propylpyrimidine-5-carbonyl)-1,4,9-triazaspiro[5.6]dodecan-10-one
(1S,5R)-6-(5-methoxyfuran-2-carbonyl)-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
3-cyclopropyl-4-[3,5-dimethyl-2-(1H-pyrazol-1-yl)phenyl]-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
5-(dimethylamino)-2-[2-oxo-2-(4-phenylazepan-1-yl)ethyl]-2,3-dihydropyridazin-3-one
N-benzyl-N-butyl-1-[2-(1,1-dioxo-1λ6-thiolan-3-yl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]piperidine-3-carboxamide
3-(3,4-dimethoxybenzoyl)-1-[(2,5-dimethylthiophen-3-yl)sulfonyl]piperidine
3-(2-fluorophenyl)-N-[2-(N-methylmethanesulfonamido)ethyl]-3-phenylpropanamide