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N-[1-(4-methanesulfonylphenyl)ethyl]-4-(1H-pyrazol-4-yl)butanamide
1-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-4-(2-phenoxyethyl)piperazine
(2R)-2-{[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]amino}-3-phenylpropan-1-ol
2-{N-ethyl-1-[4-methyl-2-(pyridin-3-yl)pyrimidin-5-yl]formamido}propanamide
5-methyl-N-[1-(pyrrolidine-1-carbonyl)azepan-3-yl]-1,2-oxazole-3-carboxamide
1-[(3S,4R)-3-(dimethylamino)-4-(4-methylphenyl)pyrrolidin-1-yl]-2-[4-(hydroxymethyl)phenyl]ethan-1-one
N-ethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-6-{methyl[(5-methylfuran-2-yl)methyl]amino}pyridine-3-carboxamide
1-benzyl-3-(2-methoxyethyl)-8-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-({3-[3-(methoxymethyl)piperidine-1-carbonyl]-1H-pyrazol-5-yl}methyl)-5,6-dimethyl-1H-1,3-benzodiazole
N-({1-[(6-methylpyridin-2-yl)methyl]piperidin-3-yl}methyl)-3-(trifluoromethyl)benzamide
2,5-dimethyl-N-(2-propoxyethyl)-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
methyl (1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxylate
4,4-difluoro-1-({4-[2-(1H-imidazol-1-yl)ethoxy]phenyl}methyl)piperidine
1-{1-[(4-methylpiperazin-1-yl)sulfonyl]piperidin-3-yl}-3-phenylpropan-1-one
1-(oxolan-2-ylmethyl)-4-[4-(piperidin-1-ylmethyl)benzoyl]piperazine
2-(2-hydroxyethyl)-8-(1-methyl-1H-pyrrole-2-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
5-(2,5-dimethoxyphenyl)-1-[2-(1H-imidazol-1-yl)ethyl]-4-phenyl-1H-imidazole
2-{8-[3-(2-ethyl-1H-imidazol-1-yl)propanoyl]-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-3-yl}acetic acid
N-[1-(2-methoxyphenyl)propan-2-yl]-N-methyl-3-propanamidobenzamide
1-{4-[3-(propoxymethyl)pyrrolidine-1-carbonyl]phenyl}imidazolidine-2,4-dione
{1-[(3-ethoxy-4-methoxyphenyl)methyl]-3-[(2-methylphenyl)methyl]piperidin-3-yl}methanol
N-cyclohexyl-1-(1-cyclopropanecarbonylpiperidin-4-yl)piperidine-3-carboxamide
2-[5-(2-ethyl-4-methyl-1,3-oxazol-5-yl)-3-(oxolan-3-yl)-1H-1,2,4-triazol-1-yl]quinoxaline
ethyl (4aR,6R,8aS)-2-(2-methylpyridin-4-yl)-6-(morpholin-4-yl)-decahydroisoquinoline-8a-carboxylate
3-chloro-4-{[1-(cyclopent-1-ene-1-carbonyl)piperidin-4-yl]oxy}-N-cyclopentylbenzamide
N3-({8-methylimidazo[1,2-a]pyridin-2-yl}methyl)-N5-(2-methylpropyl)-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
2-oxo-3-(pentan-3-yl)-1-(pyridin-4-ylmethyl)-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylic acid
N-[(1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]-2-(1-methyl-1H-pyrrol-2-yl)-2-oxoacetamide
N-[3-(2-oxopyrrolidin-1-yl)propyl]-3-[5-(4-phenylbutyl)-1,3,4-oxadiazol-2-yl]propanamide
1-[(3S,4S)-4-methoxy-1-(propan-2-yl)pyrrolidin-3-yl]-3-[3-methyl-1-(propan-2-yl)-1H-pyrazol-5-yl]urea
N-cyclopentyl-2-[6-oxo-4-(pyrrolidin-1-yl)-1,6-dihydropyridazin-1-yl]-N-(thiophen-3-ylmethyl)acetamide
5-cyclobutyl-3-[(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)methyl]-1,2,4-oxadiazole
2-(1-{1-[3-(propan-2-yloxy)benzoyl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)propan-2-ol
8-(1-benzylpiperidin-4-yl)-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
2-(1-{1-oxa-8-azaspiro[4.5]decan-8-yl}-1-oxobutan-2-yl)-2,3-dihydro-1H-isoindol-1-one
6-methoxy-N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-N-methylpyrimidin-4-amine
5-(3,4-dimethoxyphenyl)-N-[1-(pyridin-3-yl)propan-2-yl]-1,2,4-triazin-3-amine
4-{[2-(4-fluoro-3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-chloro-3-(2-{4-[(dimethylamino)methyl]phenyl}piperidine-1-carbonyl)-1H-pyrazol-5-amine
2-(adamantan-1-yl)-4-hydroxy-N-(2-methanesulfonylethyl)pyrimidine-5-carboxamide
N-{2-[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]ethyl}pyrazolo[1,5-a]pyridine-7-carboxamide
1-(5-chloro-2-methylphenyl)-4-{[2-(3,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazine
2-methyl-4-[4-({4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}methyl)phenyl]butan-2-ol
1-methyl-4-{1-[4-(1-propyl-1H-imidazol-2-yl)-1H-1,2,3-triazol-1-yl]propan-2-yl}piperazine
5-acetyl-6-methyl-3-[(1R,5R)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-1,2-dihydropyridin-2-one
3-cyclohexyl-N-{[1-(morpholin-4-yl)cyclopentyl]methyl}-1H-pyrazole-4-carboxamide
N-[(1R,2R,4R)-bicyclo[2.2.1]hept-5-en-2-ylmethyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
4-(1-benzyl-1H-imidazol-2-yl)-1-(3-propyl-1H-pyrazole-4-carbonyl)piperidine
2-(4-oxo-3,4-dihydroquinazolin-3-yl)-N-[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]acetamide
N-[(7-fluoro-2-oxo-1,2-dihydroquinolin-3-yl)methyl]-2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]acetamide