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1-(1-ethyl-1H-pyrazole-5-carbonyl)-4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-5-one
{1-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]piperidin-4-yl}(1-methyl-1H-imidazol-2-yl)methanol
8-[2-(1H-imidazol-1-yl)acetyl]-2-(3-methoxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
1-(1-methyl-5-{[3-(4-methylphenoxy)azetidin-1-yl]methyl}-1H-pyrrol-3-yl)ethan-1-one
5-chloro-N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-N-(2-methylpropyl)thiophene-2-carboxamide
1-(4-{[3-(2-hydroxyethyl)-4-[(4-methoxy-2,3-dimethylphenyl)methyl]piperazin-1-yl]methyl}thiophen-2-yl)ethan-1-one
N-{[1-(propan-2-yl)-1H-1,3-benzodiazol-2-yl]methyl}-2-(pyridin-4-yl)pyrimidine-5-carboxamide
3-[1-(2-methoxyphenyl)-3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]-N,N-dimethylpropanamide
2-methyl-4-(piperidin-3-yl)-6-{1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}pyrimidine
3-methoxy-1-[(2R,3S,6R)-3-(2-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]propan-1-one
3-[3-(2,5-dimethoxyphenyl)pyrrolidine-1-carbonyl]-1-methyl-1H-indole
4-(4-methyl-1H-pyrazol-1-yl)-1-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]piperidine-4-carboxylic acid
2-methoxy-N-({5-[(2,4,5-trifluorophenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)acetamide
N,8-dimethyl-3-({methyl[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amino}methyl)-N-(2-phenylethyl)imidazo[1,2-a]pyridine-2-carboxamide
N-methyl-5-({4-[1-(3-methylpyridin-2-yl)-1H-pyrazol-4-yl]-1,2,3,6-tetrahydropyridin-1-yl}methyl)furan-2-carboxamide
11-[2-(butan-2-yloxy)-3-methoxyphenyl]-4,6,10,12-tetraazatricyclo[7.3.0.03,7]dodeca-1,3(7),8,10-tetraen-5-one
(1R,5R)-6-[(5-chlorothiophen-2-yl)methyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
3-{3-ethyl-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-8-yl}propanoic acid
N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-9H-purin-6-amine
1-{3-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepan-1-yl]-3-oxopropyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-{[2-(1H-imidazol-1-yl)phenyl]methyl}-2-methyl-3-(1H-1,2,4-triazol-1-yl)propanamide
1-[2-(methylamino)pyridine-4-carbonyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
3-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}-3H,4H-pyrido[4,3-d]pyrimidin-4-one
6-(1H-imidazol-2-ylmethyl)-3-(8-methoxy-2-methylquinolin-5-yl)-1-methyl-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
ethyl 1-[(1R,2R,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]-4-[(2-chlorophenyl)methyl]piperidine-4-carboxylate
1-[3-(phenoxymethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-3-(1H-pyrrol-1-yl)propan-1-one
2-(3,5-dimethyl-1H-pyrazol-4-yl)-2-(isoquinolin-1-ylformamido)acetic acid
(2R,3R,6R)-5-(1,2-oxazole-3-carbonyl)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
5-(2-methyloxolan-2-yl)-3-(thiophen-2-ylmethyl)-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazole
N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-2H-1,3-benzodioxole-5-carboxamide
2-[8-(3-methylbutyl)-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl]pyridine-4-carbonitrile
N-[1-(4-methoxyphenyl)propyl]-N,2-dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
6-methyl-2-[2-(trifluoromethyl)phenyl]pyridine-3-carboxamide
1-[(5-chlorofuran-2-yl)methyl]-2-[2-(1H-imidazol-1-yl)ethyl]piperidine
4-benzyl-3-ethyl-1-{pyrazolo[1,5-a]pyrimidine-3-carbonyl}-1,4-diazepan-5-one
(2S,4S)-N-ethyl-1-(furan-3-ylmethyl)-4-[2-(1-methyl-1H-pyrrol-2-yl)-2-oxoacetamido]pyrrolidine-2-carboxamide
(3S,4S)-1-{[4-(methylsulfanyl)phenyl]methyl}-4-[4-(pyridin-2-yl)piperazin-1-yl]pyrrolidin-3-ol
(4aS,8aR)-1-[2-(1H-imidazol-4-yl)ethyl]-6-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-decahydro-1,6-naphthyridin-2-one
2-methyl-8-[2-(4-methylphenoxy)ethanesulfonyl]-2,8-diazaspiro[4.5]decan-3-one
4-{[methyl({[4-(1H-pyrazol-1-yl)phenyl]methyl})amino]methyl}benzonitrile
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-1-[(2-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
2-[1-(3-methylbutyl)-4-[(3-methylquinoxalin-2-yl)methyl]piperazin-2-yl]ethan-1-ol
N-[(2-chloro-6-fluorophenyl)methyl]-1-(2-methyl-6-propylpyrimidin-4-yl)piperidin-4-amine
N-[2-(dimethylsulfamoyl)ethyl]-2-(ethylamino)pyrimidine-5-carboxamide
N-[1-(cyclohex-1-en-1-yl)ethyl]-N'-(4-methylphenyl)propanediamide
3-[(3R,4R)-3-cyclopropyl-3-hydroxy-4-methylpyrrolidine-1-carbonyl]-4-methylbenzene-1-sulfonamide
N-[2-(4-chlorophenyl)ethyl]-5-(morpholin-4-ylmethyl)furan-3-carboxamide
methyl 3-[2-(3-fluorophenyl)acetyl]-9-[(1-methyl-5-oxopyrrolidin-3-yl)methoxy]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
(4aR,7aS)-1-[2-(morpholin-4-yl)pyrimidin-4-yl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-ethyl-5-(1-{2-[3-(1H-pyrazol-1-ylmethyl)phenyl]-1H-imidazol-1-yl}ethyl)-1,2,4-oxadiazole