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N-[3-(dimethyl-1,3-thiazol-2-yl)propyl]-5-methanesulfonyl-2-methylpyrimidin-4-amine
{[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}(methyl)(1,2-oxazol-3-ylmethyl)amine
5-(azepane-1-carbonyl)-1-(butan-2-yl)-N-[2-(4-methoxyphenyl)ethyl]-4-oxo-1,4-dihydropyridine-3-carboxamide
14-[3,5-dimethyl-2-(1H-pyrazol-1-yl)phenyl]-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
2-{4-[2-(hydroxymethyl)-1H-1,3-benzodiazol-1-yl]phenoxy}propanamide
(1R,9S)-5-amino-3-[6-(dimethylamino)pyridin-3-yl]-12-methyl-6,12-diazatricyclo[7.2.1.02,7]dodeca-2,4,6-triene-4-carbonitrile
N3-[2-(2-chlorophenyl)ethyl]-1-cyclohexyl-N5-cyclopropyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
N-butyl-5-[4-(4-methylphenyl)piperazine-1-carbonyl]-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3-carboxamide
3-[(1-cyclopentylpiperidin-4-yl)oxy]-N-(2,3-dihydro-1H-inden-1-yl)benzamide
4-[4-(3,5-dimethyl-1H-pyrazol-1-yl)benzamido]oxane-4-carboxylic acid
2,5,6-trimethyl-N-(oxan-2-ylmethyl)pyrimidin-4-amine
2-(3-{[methyl(thiophen-2-ylmethyl)amino]methyl}phenyl)-6-(pyridin-3-yl)-3,4-dihydropyrimidin-4-one
2-[5-(3-hydroxy-3-methylbut-1-yn-1-yl)thiophen-2-yl]-1H-1,3-benzodiazole-6-carboxylic acid
1-(2-ethylpiperidin-1-yl)-3-[5-(5-methyl-1,2-oxazol-3-yl)-1,3,4-oxadiazol-2-yl]propan-1-one
4-[(2-methylprop-2-en-1-yl)oxy]-N-[(3R,4R)-4-(piperidin-1-yl)oxolan-3-yl]benzamide
N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}-3-(2-oxooxolan-3-yl)propanamide
(1R,3R)-N1-[5-(propan-2-yl)pyrimidin-4-yl]cyclopentane-1,3-diamine
2-amino-4-(4-methoxyphenyl)-6-(pyridin-3-ylmethyl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
1-(5-cyclopropyl-1,3-oxazole-4-carbonyl)-4-(3-methylpyridin-2-yl)piperazine
1-[6-benzyl-2-(dimethylamino)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-4-yl]piperidin-4-ol
2-[1-(1,4-dioxan-2-ylmethyl)-4-phenyl-1H-imidazol-5-yl]benzoic acid
3-[1-(cyclopent-1-ene-1-carbonyl)piperidin-3-yl]-1-(pyrrolidin-1-yl)propan-1-one
{[3-cyclopropyl-1-(4-methoxyphenyl)-1H-1,2,4-triazol-5-yl]methyl}urea
2-(2-fluoro-5-methylphenyl)-1H-1,3-benzodiazole-6-carboxylic acid
2-{[6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]methyl}-3,5-dimethyl-1,4-dihydropyridin-4-one
4-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepine-8-carbonyl}-2,6,8-trimethylquinoline
2-[2-(1-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}piperidin-3-yl)-1H-imidazol-1-yl]acetamide
N-methyl-N-(oxan-4-ylmethyl)-6-oxo-1-[2-(pyridin-2-yl)ethyl]piperidine-3-carboxamide
N-(1-cyclohexyl-1H-pyrazol-5-yl)-2-[3,5-dimethyl-4-(5-methylfuran-2-yl)-1H-pyrazol-1-yl]acetamide
5-butyl-4-(1-methyl-1H-pyrrole-2-carbonyl)-1-(3-phenylphenyl)piperazin-2-one
2-(1-{[3-(4-phenylphenyl)-1H-pyrazol-4-yl]methyl}pyrrolidin-2-yl)pyridine
2-acetamido-2-methyl-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}propanamide
3-(2H-1,3-benzodioxol-5-yl)-1-{3-[(3,4-difluorophenyl)amino]piperidin-1-yl}propan-1-one
8-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decan-3-one
6-cyclopentyl-1-methyl-N-[1-(pyridin-3-yl)propyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-(1,1-dioxo-1λ6-thian-4-yl)-N-[(3R,4S)-1-methyl-4-phenylpyrrolidin-3-yl]acetamide
1-[(3R,4S)-3-amino-4-(4-methoxyphenyl)pyrrolidin-1-yl]-3-(2-ethyl-1H-imidazol-1-yl)propan-1-one
1-(diethylamino)-3-[2-methoxy-4-({[(3-methyloxetan-3-yl)methyl]amino}methyl)phenoxy]propan-2-ol
5-(2-chloro-4-methoxyphenoxymethyl)-N-methyl-N-(oxolan-3-yl)-1,2-oxazole-3-carboxamide
N-({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N,2-dimethyl-6-oxo-1,6-dihydropyrimidine-5-carboxamide
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-{2-[(3-{[(5-ethylfuran-2-yl)methyl]amino}-5-[(2-methylphenyl)sulfamoyl]phenyl)formamido]ethyl}acetamide
{6-[(1S,4S)-2-azabicyclo[2.2.1]heptan-2-yl]-2-methylpyrimidin-4-yl}methanamine
5-{[2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-N,N-dimethylpyridin-2-amine
1-methyl-2-(morpholin-4-yl)-N-(1,4-oxazepan-6-ylmethyl)-1H-1,3-benzodiazole-5-carboxamide
(3S,4R)-4-phenyl-1-[3-(piperidin-1-yl)propanoyl]pyrrolidine-3-carboxylic acid
N-[2-(7-methyl-1H-indol-3-yl)ethyl]-1-(pyridin-2-ylmethyl)piperidin-4-amine
3-(1H-pyrazol-1-yl)-N-{2-[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]ethyl}benzamide
1-(6-methoxy-3-methyl-1-benzofuran-2-amido)cyclopentane-1-carboxylic acid
N-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-1-methyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine