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ethyl 4-[1-methyl-2,4-dioxo-3-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decan-8-yl]piperidine-1-carboxylate
1-(2-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}-1,3-oxazole-4-carbonyl)azocane
N-[(5-ethylpyridin-2-yl)methyl]-3-(2-fluorophenyl)-N-methyl-1H-pyrazole-5-carboxamide
1-[1-(2-fluorobenzenesulfonyl)piperidin-3-yl]-4-(2-methoxyphenyl)piperazine
methyl 4-{[1-(3,4-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]carbamoyl}benzoate
N-[(2-chlorophenyl)methyl]-4-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}benzamide
[(3-benzyl-1,2,4-oxadiazol-5-yl)methyl]({[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl})methylamine
6-(4,4-diphenylpiperidine-1-carbonyl)piperazin-2-one
5-(2-methyloxolan-2-yl)-3-(thiophen-3-ylmethyl)-1,2,4-oxadiazole
2-benzyl-N-[(3R,4R)-4-(pyrrolidin-1-yl)oxolan-3-yl]-1,3-thiazole-4-carboxamide
1'-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]-3,4-dihydrospiro[1-benzopyran-2,3'-pyrrolidine]-4-one
1-[1-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-1H-1,2,3-triazole-4-carbonyl]-4-methylpiperidine
N-(4-{[3-(methanesulfonamidomethyl)pyrrolidin-1-yl]methyl}phenyl)acetamide
5-(propane-2-sulfonyl)-3-(thiophen-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
4-ethyl-1-methyl-3-[1-(1-phenylpiperidin-4-yl)piperidin-3-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
5-{[benzyl(methyl)amino]methyl}-N-[2-(4-methyl-1H-pyrazol-1-yl)ethyl]-1,2-oxazole-3-carboxamide
7-(2-methoxyethyl)-2-(2-methoxypyridine-4-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
2-(2,5-dimethylphenyl)-1-[4-(morpholin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
N-ethyl-4-methoxy-N-{[2-(prop-2-en-1-yloxy)phenyl]methyl}cyclohexane-1-carboxamide
4-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-6-(4-methylpiperazin-1-yl)pyrimidin-2-amine
(1S,5R)-3-benzyl-N-[(3-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
5-{2-cyclopentyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-yl}-4H,5H,6H,7H-[1,3]thiazolo[5,4-c]pyridin-2-amine
N-cyclohexyl-3-[1-ethyl-3-(2-methoxyethyl)-1H-1,2,4-triazol-5-yl]-N-methylpropanamide
2-[4-(4-fluorophenyl)-2-[(4-methylpiperazin-1-yl)methyl]phenoxy]-N-(3-methoxypropyl)acetamide
3-[(2-fluorophenyl)formamido]-N-[(2S)-1-hydroxy-3-phenylpropan-2-yl]propanamide
2-({4-[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]-1H-1,2,3-triazol-1-yl}methyl)pyridine
2-[1-(2-chlorophenyl)-3-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-[2-(pyridin-2-yl)ethyl]acetamide
{4-[(2-chlorophenyl)methyl]-1-(1,4-dithiepan-6-yl)piperidin-4-yl}methanol
(1R,5R)-6-[1-(2-ethoxyethyl)-3-methyl-1H-pyrazole-5-carbonyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
2-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N-methyl-N-[(3-methylpyridin-2-yl)methyl]benzamide
1-[1-(2,4-dimethylbenzoyl)piperidin-3-yl]-4-(2-methylphenyl)piperazine
N-cyclopropyl-5-(2,3-dihydro-1,4-benzodioxine-2-carbonyl)-1-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-[4-chloro-2-({[(dimethyl-1,2-oxazol-4-yl)methyl](methyl)amino}methyl)phenoxy]acetic acid
1-[(2-butyl-1H-imidazol-4-yl)methyl]-N-[3-(3-fluorophenyl)phenyl]piperidine-4-carboxamide
N-[(2-chlorophenyl)methyl]-1-ethyl-N-(propan-2-yl)-1H-pyrazole-3-carboxamide
N-{4-[2-methoxy-4-(pyrrolidin-1-ylmethyl)phenoxy]phenyl}acetamide
5-fluoro-2-(1-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}pyrrolidin-2-yl)-1H-1,3-benzodiazole
{3-[(3-chlorophenyl)methyl]-1-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]piperidin-3-yl}methanol
2-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}-1-(morpholin-4-yl)ethan-1-one
2-(3-fluorophenyl)-1-[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]azepane
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-N-methyl-6-(2-methylphenyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
4-[1-(2-{[2-(pyrrolidin-1-yl)ethyl]sulfanyl}acetyl)piperidin-3-yl]benzoic acid
5-{3-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]piperidine-1-carbonyl}-N,4-dimethyl-1,3-thiazol-2-amine
5-chloro-2-methoxy-N-[(3-methoxyphenyl)methyl]-N-(prop-2-en-1-yl)benzamide
N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-(1,3-thiazol-4-ylmethyl)cyclopropanamine
7-{1-[(4-methoxyphenyl)methyl]-1H-pyrazol-4-yl}-[1,2,4]triazolo[4,3-c]pyrimidin-5-amine
1-{4H,5H,6H,7H,8H-cyclohepta[b]thiophene-2-carbonyl}-4-(1H-imidazol-2-yl)piperidine
1-(morpholin-4-yl)-2-[4-({[1-(pyridin-4-yl)propan-2-yl]amino}methyl)phenoxy]ethan-1-one
N-[3-(1H-indazol-1-yl)propyl]pyrazin-2-amine
2-methoxy-N-(1-{1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-phenylacetamide