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N4-[1-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-6-ethyl-5-methylpyrimidine-2,4-diamine
7-methyl-3-{[methyl({[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl})amino]methyl}quinolin-2-ol
2-[4-phenyl-5-(pyridin-2-yl)-1H-imidazol-1-yl]acetic acid
N-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-N-methyl-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
3-(3-methyl-1,2,4-thiadiazol-5-yl)-1-[1-(morpholin-4-ylmethyl)cyclopentyl]urea
methyl 3-(2-chlorobenzenesulfonamido)-5-[(2-phenoxyacetamido)methyl]benzoate
1-{[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}-3-methylpiperidin-3-ol
5-ethyl-N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]pyrazolo[1,5-a]pyrimidin-7-amine
2-fluoro-N-{[1-(4-methylphenyl)pyrrolidin-3-yl]methyl}-5-sulfamoylbenzamide
1-{4-[1-(2H-1,3-benzodioxol-5-yl)-3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]piperidin-1-yl}ethan-1-one
3-{[4-(2-hydroxyethyl)-1H-1,2,3-triazol-1-yl]methyl}-N-(2-methoxyphenyl)piperidine-1-carboxamide
1-[(1R,2S,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]-4-[(2-fluorophenyl)methyl]-1,4-diazepan-5-one
3-(3-hydroxy-3-methylbutyl)-N-(1H-imidazol-2-ylmethyl)benzamide
2-cyclopropyl-N-methyl-6-oxo-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]-1,6-dihydropyrimidine-5-carboxamide
1-(3,4-dimethoxyphenyl)-3-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}urea
1-[2-(3,4-dichlorophenyl)morpholin-4-yl]-4-(1H-imidazol-1-yl)butan-1-one
4-[4-(2-chlorophenyl)piperidin-4-yl]-N-[3-(dimethylamino)propyl]pyrimidin-2-amine
1-[(1S,3R)-3-hydroxy-1-methoxy-1-methyl-7-azaspiro[3.5]nonan-7-yl]-2-[(2-methylphenyl)sulfanyl]ethan-1-one
2-{4-[(5-acetylthiophen-3-yl)methyl]piperazin-1-yl}acetamide
N-methyl-2-[methyl(piperidin-4-yl)amino]-N-{[3-(methylsulfanyl)phenyl]methyl}acetamide
(1S,4S)-2-({6-chloro-2-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]imidazo[1,2-a]pyridin-3-yl}methyl)-2-azabicyclo[2.2.1]heptane
2-(4-fluorophenoxy)-N-methyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]acetamide
7-fluoro-3-{[2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-1H-imidazol-1-yl]methyl}-1,2-dihydroquinolin-2-one
5-(1-methyl-3-phenyl-1H-pyrazol-5-yl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
3-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)-N-[1-(4-methylpyridin-2-yl)propyl]propanamide
4-methyl-2-(pyridin-3-yl)-6-[3-(pyridin-3-ylmethyl)piperidin-1-yl]pyrimidine
2-methyl-1-{5-propanoyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-3-(1H-1,2,4-triazol-1-yl)propan-1-one
3-(4-fluorophenyl)-N-{3-[4-(4-methylpiperazine-1-carbonyl)-1H-1,2,3-triazol-1-yl]propyl}benzamide
4-[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]-2-(trifluoromethyl)morpholine
6-chloro-8-methyl-3-(1-methyl-2-oxopyrrolidin-3-yl)-3,4-dihydroquinazolin-4-one
2-(2-phenyl-1H-imidazol-1-yl)-N-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}acetamide
4-benzyl-1-(2,6-dimethylbenzoyl)-3-ethyl-1,4-diazepan-5-one
methyl({[1-(3-methylbutyl)-2-(propane-2-sulfonyl)-1H-imidazol-5-yl]methyl})[(1-methylpyrrolidin-2-yl)methyl]amine
2-amino-3-ethyl-N-{[5-methyl-2-(trifluoromethyl)furan-3-yl]methyl}-3H-imidazo[4,5-b]pyridine-6-carboxamide
1-{[1-(cyclohexylmethyl)-2-cyclopropylmethanesulfonyl-1H-imidazol-5-yl]methyl}piperidine-3-carboxamide
{[3-(2-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}({[1-(pyrimidin-2-yl)piperidin-3-yl]methyl})amine
2-(4-chlorophenyl)-N-{[1-(3-fluoropropyl)-1,2,3,6-tetrahydropyridin-4-yl]methyl}acetamide
(3aR,6aS)-2-(cyclopropylmethyl)-5-[(furan-2-ylmethyl)carbamoyl]-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-(3-{3-[2-(4-methoxyphenyl)ethyl]piperidin-1-yl}-3-oxopropyl)methanesulfonamide
(1R,5R)-3-methanesulfonyl-6-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-3,6-diazabicyclo[3.2.2]nonane
1-{2-[5-(4-chlorophenyl)-1,2,4-oxadiazol-3-yl]ethyl}pyrrolidin-2-one
(1R,5S,8S)-8-methoxy-N-(1-methyl-1H-1,3-benzodiazol-5-yl)-3-azabicyclo[3.2.1]octane-3-carboxamide
1-{4-[(3-methylphenyl)methyl]piperazin-1-yl}-3-(4H-1,2,4-triazol-4-yl)propan-1-one
5-cyclopropyl-1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-N-(1,3-thiazol-2-ylmethyl)-1H-pyrazole-4-carboxamide
(4aR,7aS)-1-cyclobutanecarbonyl-4-[(2-methoxyphenyl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
[(1S)-1-{3-[(3,4-dimethoxyphenyl)methyl]-1-(1-methylpiperidin-4-yl)-1H-1,2,4-triazol-5-yl}ethyl](methyl)amine
1-[(4-ethyl-5-methylpyrimidin-2-yl)amino]-3-(4-methoxyphenoxy)propan-2-ol
5-(3-fluoro-4-methoxyphenyl)-1-[(5-methylfuran-2-yl)methyl]-1H,4H-pyrazolo[3,4-d]imidazole
1-(1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}piperidin-4-yl)azepane
2-(1-{1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}piperidin-4-yl)propan-2-ol