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1-methyl-4-(oxane-4-carbonyl)-9-(prop-2-en-1-yl)-1,4,9-triazaspiro[5.6]dodecan-10-one
3-{4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}pyridine
(isoquinolin-5-ylmethyl)[2-(4-methoxyphenyl)ethyl][(1-methylpiperidin-4-yl)methyl]amine
N-methyl-4-[5-(piperazin-1-ylmethyl)thiophen-3-yl]-1H-pyrrolo[2,3-b]pyridin-6-amine
5-(3-acetylphenoxymethyl)-N-methyl-N-[2-(oxan-2-yl)ethyl]-1,2-oxazole-3-carboxamide
{[3-(3-chlorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl}(methyl)[(1-methylpyrrolidin-2-yl)methyl]amine
2-{3-[2-(4-ethylphenyl)-1H-imidazol-1-yl]piperidin-1-yl}pyrimidine
N-{2-[(4-chlorophenyl)methoxy]ethyl}-3-fluoro-7-methylimidazo[1,2-a]pyridine-2-carboxamide
N-{[2-(1H-imidazol-1-yl)phenyl]methyl}-2-{2-methylimidazo[1,2-a]pyridin-3-yl}acetamide
ethyl 4-(2-phenoxyethyl)piperidine-4-carboxylate
2-(5-amino-1H-1,2,3,4-tetrazol-1-yl)-1-[7-(hydroxymethyl)-3,9-diazaspiro[5.5]undecan-3-yl]ethan-1-one
2-(aminomethyl)-N-(4-methoxy-3,5-dimethylphenyl)piperidine-1-carboxamide
2-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-7-methyl-4H-chromen-4-one
2-(5-amino-1,3,4-thiadiazol-2-yl)-N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]acetamide
3-(4-hydroxy-2-methylquinolin-3-yl)-N-[4-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]propanamide
2-{[1-ethyl-3-(2-methylpropyl)-1H-pyrazol-5-yl]formamido}-2-(2-fluorophenyl)acetic acid
3-[1-(3-methylbutyl)-3-(morpholine-4-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-4,5,6,7-tetrahydro-1,2-benzoxazole
1-({3-[3-(morpholin-4-yl)azetidine-1-carbonyl]-1H-pyrazol-5-yl}methyl)-1H-indole
(5S)-5-{[(pyridin-2-ylmethyl)[(3-{[3-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)methyl]amino]methyl}pyrrolidin-2-one
6-methyl-N-[2-(2-methyl-1H-indol-1-yl)ethyl]imidazo[1,2-a]pyridine-2-carboxamide
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-6-[(3-hydroxypropyl)amino]-N-methylpyridine-3-carboxamide
N'-(1-cyclopropanecarbonylpiperidin-3-yl)-N-(2,4-dimethylphenyl)propanediamide
2-(3,6-dioxo-1,2,3,6-tetrahydropyridazin-1-yl)-N-ethyl-N-{[2-(prop-2-en-1-yloxy)phenyl]methyl}acetamide
1-methyl-N-{[4-(methylsulfanyl)phenyl]methyl}-N-propyl-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
N-(3-{1-azabicyclo[3.2.1]octan-5-yloxy}phenyl)-4,6-dimethylpyrimidin-2-amine
6-[3-fluoro-5-(2-methylpropoxy)phenyl]quinazolin-4-amine
N-{[7-(5-acetyl-2-fluorophenyl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methyl}-4,4,4-trifluorobutanamide
N-(2-{[4-methyl-3-(2-oxoimidazolidin-1-yl)phenyl]formamido}ethyl)pyridine-3-carboxamide
2-(2H-1,3-benzodioxol-5-yl)-1-{2-[2-(3-{[4-(3-chlorophenyl)piperazin-1-yl]methyl}phenoxy)ethyl]piperidin-1-yl}ethan-1-one
2-[6-(cyclopentylamino)-1H-pyrrolo[2,3-b]pyridin-4-yl]pyridin-3-ol
(3aR,6aR)-2-[(3-chlorophenyl)methyl]-5-(cyclobutylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-(methanesulfonylmethyl)-1-[(2-phenyl-1,3-oxazol-4-yl)methyl]piperidine
N-benzyl-2-(1-methyl-1H-pyrazol-3-yl)piperidine-1-sulfonamide
[(3R,4S)-1-[(5-fluoro-1-methyl-1H-indol-2-yl)methyl]-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
2-{4-[2-(2-methyl-1H-imidazol-1-yl)propyl]piperazin-1-yl}pyrimidine
N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-N,5-dimethyl-1-propyl-1H-pyrazole-4-carboxamide
3-methoxy-1-(2-{9-oxa-2-azaspiro[5.5]undecan-2-yl}-2-oxoethyl)-1,2-dihydropyridin-2-one
3-({[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}(oxolan-2-ylmethyl)amino)propan-1-ol
7-(cyclopropylmethyl)-6-(4-methoxyphenyl)-N-methyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
8-(1H-indol-3-ylmethyl)-1-[2-(4-methoxyphenyl)ethyl]-3-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(3-{[3-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)-2-(3-methyl-1H-1,2,4-triazol-5-yl)ethan-1-one
(1S,5R)-3-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
3-(2-fluorophenyl)-N-[2-(2-oxopiperidin-1-yl)ethyl]-3-phenylpropanamide
4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]-1-[(3-methoxyphenyl)methyl]piperidine
N-{2-[({5-[(dimethylamino)methyl]furan-2-yl}methyl)sulfanyl]ethyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2-(5-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepine-8-sulfonyl}thiophen-2-yl)pyridine
N-methyl-3-(1,2-oxazolidin-2-yl)-N-(quinolin-4-ylmethyl)propanamide
N-[2-(dimethylamino)-2-(3-methylthiophen-2-yl)ethyl]-2-(piperidin-4-yl)acetamide
methyl 2-{2-[(3,5-difluorophenyl)methyl]-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}propanoate
N-{2-[methyl(phenyl)amino]propyl}-6-(4H-1,2,4-triazol-4-yl)pyridine-2-carboxamide