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[2-(diethylamino)-2-(furan-2-yl)ethyl][(3,5-difluorophenyl)methyl]amine
2-cyclopropyl-8-{[2-(propan-2-yl)pyrimidin-5-yl]methyl}-2,8-diazaspiro[5.5]undecan-3-one
5-(1-{[(2-methyl-2H-1,2,3-triazol-4-yl)carbamoyl]methyl}-1H-pyrazol-4-yl)-N-propylfuran-2-carboxamide
2-{1-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]piperidin-2-yl}pyridine
(1S,5R)-6-benzyl-3-(5-hydroxypyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
7,7-dimethyl-2-{[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]methyl}-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
4-(3-{[2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]amino}propyl)piperazin-2-one
1-[4-(4-fluorophenoxy)piperidin-1-yl]-2-(thiophen-3-yl)ethan-1-one
2-[(7-chloro-4-methylquinolin-2-yl)amino]acetamide
6-methyl-N-[1-(2-phenylethyl)piperidin-3-yl]pyridazin-3-amine
(3R,4R)-4-[4-(2-fluorophenyl)piperazin-1-yl]-1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidin-3-ol
1-{[2-(3,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-propyl-1H-1,2,4-triazole
N-{2-[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidin-1-yl]-2-oxoethyl}benzamide
N-methyl-5-[(methylsulfanyl)methyl]-N-[1-(3-phenylpropyl)piperidin-3-yl]furan-2-carboxamide
5-methoxy-3-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}-1H-indazole
N-ethyl-N-methyl-6-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}pyrimidin-4-amine
[(2S)-1-{5-[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}pyrrolidin-2-yl]methanol
2-[9-oxo-8-(propan-2-yl)-2,8-diazaspiro[5.5]undecan-2-yl]-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
(3R,5S)-5-[(2,3-dihydro-1H-inden-5-yloxy)methyl]-N-(2-phenylethyl)piperidine-3-carboxamide
6-{4-oxo-2-phenyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl}-2,3,4,5-tetrahydropyridazin-3-one
4-(azetidine-1-carbonyl)-1-[1-(3-phenylpropyl)piperidin-4-yl]piperidine
N-[(1-butylpiperidin-4-yl)methyl]-3-cyclopropaneamido-4-methylbenzamide
3-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-(2-{4-methyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}ethyl)benzamide
(2S,3S)-2-[3-(4,5-dimethyl-1H-pyrazol-3-yl)propanamido]-3-methylpentanamide
2-[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]-N-cycloheptylacetamide
1-(6-ethoxy-4-methylquinazolin-2-yl)-N-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}pyrrolidine-2-carboxamide
N-[(4-fluorophenyl)methyl]-3-[5-(2-phenylethyl)-1,3,4-oxadiazol-2-yl]propanamide
N-[4-(2-methyl-1H-imidazol-1-yl)phenyl]-1-(6-methylpyridine-2-carbonyl)pyrrolidine-2-carboxamide
1-(azocan-1-yl)-3-[5-methoxy-2-({methyl[2-(1H-pyrazol-4-yl)ethyl]amino}methyl)phenoxy]propan-2-ol
4-methyl-2-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}-1,3-thiazole-5-carboxylic acid
N-{[4-(but-2-yn-1-yloxy)phenyl]methyl}-4-phenyl-N-(pyridin-3-ylmethyl)benzamide
1-[2-(5-amino-1H-1,2,4-triazol-3-yl)ethyl]-5-(2H-1,3-benzodioxol-5-ylmethyl)-5-methylpiperidin-2-one
N-{[2-(dimethylamino)-1,3-thiazol-4-yl]methyl}-2-(7-fluoro-2-methyl-1H-indol-3-yl)acetamide
(1R,5R)-6-(8-fluoroquinoline-2-carbonyl)-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
4-(2-methylquinolin-6-yl)-1-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]piperidin-4-ol
4-{1-cyclopentyl-3-methyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-5-methyl-1-propyl-1H-pyrazole
N-(1,2-oxazol-3-ylmethyl)-2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carboxamide
(3aS,6aS)-2-cyclohexyl-5-(ethanesulfonyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-amido]-1,2,3,4-tetrahydronaphthalene-1-carboxylic acid
methyl 3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidine-1-carboxylate
N-[(6-methylpyridin-2-yl)methyl]-4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}benzamide
N-methyl-2-(oxolane-3-carbonyl)-N-(propan-2-yl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
6-methoxy-N-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-(2-{[(4-hydroxy-6,8-dimethylquinolin-2-yl)methyl]amino}ethyl)pyridine-3-carboxamide
2-[3,5-dimethyl-4-({methyl[(5-propyl-1H-pyrazol-3-yl)methyl]amino}methyl)-1H-pyrazol-1-yl]ethan-1-ol
ethyl 4-{6-[3-(1,3-benzothiazol-2-yl)propanoyl]-6-azaspiro[2.5]octane-1-carbonyl}piperazine-1-carboxylate
N-[(1-methylpiperidin-3-yl)methyl]-2-(prop-2-en-1-ylsulfanyl)acetamide
N-[2-(1H-imidazol-4-yl)ethyl]-2-oxo-1-oxaspiro[4.5]decane-4-carboxamide
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}-N-(2-methoxyethyl)-4-methyl-1,2,5-oxadiazole-3-carboxamide
4-[5-({3-[3-(propan-2-yloxy)benzoyl]piperidin-1-yl}methyl)-1,3-thiazol-2-yl]morpholine