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9-({4-amino-6-[(3-methylphenyl)amino]-1,3,5-triazin-2-yl}methyl)-1-oxa-9-azaspiro[5.5]undecan-5-ol
2-methyl-N-(2-phenoxyethyl)-3-[(pyridin-2-ylmethyl)amino]benzamide
ethyl 2-{7-methyl-12-oxo-3,7,11-triazaspiro[5.6]dodecan-3-yl}acetate
N-({7-[3-(1,3-benzothiazol-2-yl)propanoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-3-methylthiophene-2-carboxamide
(4-{[4-(piperidin-3-yl)-1H-1,2,3-triazol-1-yl]methyl}phenyl)methanol
1-[2-(1H-imidazol-4-yl)ethyl]-4-{8-oxatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-6-yl}-1H-1,2,3-triazole
7-methyl-3-{[1-(2-phenylethyl)piperidin-3-yl]methyl}-3H,4H-thieno[3,2-d]pyrimidin-4-one
1-[3-(1-methyl-1H-imidazole-2-carbonyl)piperidin-1-yl]-2-(pyridin-2-ylsulfanyl)ethan-1-one
4-{[1-(dimethylsulfamoyl)piperidin-4-yl]oxy}-N-(2-methoxyethyl)benzamide
1-methyl-N-[1-(methylcarbamoyl)cyclohexyl]-3-phenyl-1H-pyrazole-5-carboxamide
3-[(3R,4S)-1-(6-methylpyridazin-3-yl)-4-(morpholin-4-yl)piperidin-3-yl]propan-1-ol
4,5-dimethyl-6-[4-(1H-pyrazole-4-carbonyl)piperazin-1-yl]pyrimidine
4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-N-ethylpiperidine-1-carboxamide
3-(4-methyl-1H-pyrazol-1-yl)-1-{4-[4-methyl-5-(morpholin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}propan-1-one
N,N-dimethyl-5-{[4-(3-methylpyridin-4-yl)-1,4-diazepan-1-yl]methyl}pyridin-2-amine
N-methyl-5-(propan-2-yl)-N-{[2-(1H-pyrazol-1-yl)phenyl]methyl}-1,2-oxazole-3-carboxamide
4-methyl-N-{3-[methyl(phenyl)amino]propyl}pyrimidine-5-carboxamide
1-({4-[2-hydroxy-3-(morpholin-4-yl)propoxy]-3-methoxyphenyl}methyl)piperidine-4-carbonitrile
ethyl 1-[1-(1-methyl-1H-pyrazol-4-yl)ethyl]-4-oxo-5-phenoxy-1,4-dihydropyridine-3-carboxylate
N-[3-(5-amino-1,3,4-thiadiazol-2-yl)propyl]-3-[(2-fluorophenyl)formamido]propanamide
5-[(cyclopropylmethyl)(propyl)amino]-N-(furan-2-ylmethyl)-N,1-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
(3S,4S)-1-[(2-butoxy-3-methoxyphenyl)methyl]-4-(4-methylpiperazin-1-yl)pyrrolidin-3-ol
N-[(6-chloro-1H-1,3-benzodiazol-2-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-amine
ethyl({5-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)(2-methylprop-2-en-1-yl)amine
3-(3,4-dimethoxybenzoyl)-1-[(3,5-dimethoxyphenyl)methyl]piperidine
ethyl 1-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-4-{[2-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
2-(2-{[(1-ethyl-1H-imidazol-2-yl)methyl](methyl)amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
N-(3-methoxypropyl)-N-methyl-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
2-(6-chloroquinolin-2-yl)-N,N-dimethylbenzamide
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N-methyl-3-(4H-1,2,4-triazol-4-yl)benzamide
1-methyl-6-(pyridin-4-yl)-N-[(2R)-1,1,1-trifluoro-3-methylbutan-2-yl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-[(1-ethyl-1H-pyrazol-4-yl)methyl]pyrrolidine-3-carboxylic acid
6-chloro-N-{5-[(2-methylphenyl)methyl]-1,3,4-thiadiazol-2-yl}pyridine-2-carboxamide
N-{1-[1-(2,3-dihydro-1-benzofuran-5-ylmethyl)piperidin-4-yl]-2-phenylethyl}-N,2-dimethylfuran-3-carboxamide
N-{[2-(dimethylamino)-5,6,7-trimethoxyquinolin-3-yl]methyl}-4-acetamido-N-[2-(4-fluorophenyl)ethyl]benzamide
N-[4-(difluoromethoxy)phenyl]-2-(pyrrolidin-1-ylmethyl)-1,4-oxazepane-4-carboxamide
2-(2-methyl-6-{2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidin-1-yl}pyrimidin-4-yl)ethan-1-amine
2-{4-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]piperazin-1-yl}-N-ethylacetamide
7-[(4-methylpiperazin-1-yl)sulfonyl]-N-propyl-1,2,3,4-tetrahydroisoquinoline-2-carboxamide
[(2-butyl-1H-imidazol-4-yl)methyl][2-(4-methoxyphenyl)ethyl][(1-methylpiperidin-4-yl)methyl]amine
1-(3-chloro-4-fluorobenzoyl)-4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine
N-cyclopropyl-3-(2,5-dioxoimidazolidin-4-yl)-N-(1H-indol-5-ylmethyl)propanamide
1-[6-(2,5-difluorophenyl)pyridin-2-yl]piperazine
N-(2H-1,3-benzodioxol-5-yl)-1-[(3-cyclohexyl-1H-pyrazol-4-yl)methyl]piperidin-3-amine
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
1-(2-phenoxyethyl)-4-{[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}piperazine
4-[2-(1H-indol-3-yl)acetyl]piperazine-2-carboxylic acid
{[3-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-5-yl]methyl}(2,1,3-benzothiadiazol-5-ylmethyl)methylamine
(3aS,6aS)-2-cyclobutanecarbonyl-5-[2-(phenylsulfanyl)ethyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-{[2-(4-methoxy-2,5-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1-methyl-2-phenylpiperazine