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2-(methylamino)-N-(2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}ethyl)pyridine-4-carboxamide
N-{[6-(dimethylamino)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}-N-[2-(dimethylamino)ethyl]oxolane-2-carboxamide
(3S,4R)-1-{[2-(methoxymethyl)pyrimidin-5-yl]methyl}-N,N-dimethyl-4-propylpyrrolidin-3-amine
N-[1-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N,2,6-trimethylquinoline-3-carboxamide
3-(1-benzofuran-2-yl)-5-methyl-2-(4H-1,2,4-triazol-4-yl)pyridine
N-(2-hydroxy-3-phenylpropyl)-5-(morpholin-4-ylmethyl)-1,2-oxazole-3-carboxamide
N-{[1-(methoxymethyl)cyclopentyl]methyl}-2,4-dioxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
N-[(3R,4S)-4-cyclopropyl-1-(furan-2-carbonyl)pyrrolidin-3-yl]pyrazolo[1,5-a]pyridine-3-carboxamide
N-[(1S,2R)-2-hydroxycyclopentyl]-2-(4-methyl-1,4-diazepan-1-yl)acetamide
4-methoxy-3-{3-methyl-2-oxo-1-oxa-3,7-diazaspiro[4.4]nonane-7-carbonyl}benzene-1-sulfonamide
(1S,5R)-3-[(4-methoxyphenyl)methyl]-6-{[5-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-3,6-diazabicyclo[3.2.2]nonane
(1-{3-[(5-methylpyrimidin-2-yl)amino]propyl}piperidin-2-yl)methanol
6-methyl-N-[(5-methyl-1H-1,3-benzodiazol-2-yl)methyl]-4-(4-methyl-1H-imidazol-5-yl)-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
N-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-4-(piperidin-3-yl)benzamide
3-{[3-(4-methoxy-2-methylbenzoyl)piperidin-1-yl]sulfonyl}pyridine
2-{4-[(2-ethylpyrimidin-4-yl)methyl]piperazin-1-yl}pyridine-3-carboxamide
methyl 1-[2-(1H-indol-3-yl)ethyl]-3-(3-methoxypropanamido)-5-[(pyridin-3-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
4-{2-cyclobutyl-3H-imidazo[4,5-b]pyridin-3-yl}-1-(oxolane-2-carbonyl)piperidine
N-[(4-methoxyphenyl)methyl]-5-oxo-N-propyl-1-(pyridin-4-ylmethyl)pyrrolidine-3-carboxamide
N,5,7-trimethyl-N-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]pyrazolo[1,5-a]pyrimidine-2-carboxamide
2-{[2-(2,4-difluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-5-methyl-1,3,4-oxadiazole
2-{4-[5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]morpholin-2-yl}ethan-1-amine
N-[(1,3-dimethylpyrrolidin-3-yl)methyl]-3-(5-methyl-2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)propanamide
11-[bis(prop-2-en-1-yl)amino]-4-(2,3-dihydro-1H-inden-2-yl)-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
{1-[1-(7-methoxy-4-methylquinazolin-2-yl)piperidine-3-carbonyl]piperidin-4-yl}(phenyl)methanol
3-methyl-5-{4-[(2-methylphenyl)sulfanyl]piperidine-1-carbonyl}pyridine
2-(3-chloro-4-hydroxyphenyl)-1-[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]ethan-1-one
3-{6-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}-1-methyl-1,2-dihydropyridin-2-one
1-(3-cyclohexyl-1H-pyrazole-4-carbonyl)-4-[(dimethylamino)methyl]azepan-4-ol
3-{2-[3-(1H-1,3-benzodiazol-2-ylmethyl)piperidin-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
5-(1-benzofuran-2-yl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
ethyl 3-{2-[(6-{[(4-fluorophenyl)methyl](methyl)amino}pyridazin-3-yl)oxy]acetamido}propanoate
1-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-N-[2-(dimethylamino)ethyl]-N-ethyl-1H-1,2,3-triazole-4-carboxamide
3-[1-(1-benzofuran-2-ylmethyl)piperidin-3-yl]-N-(2-fluorophenyl)propanamide
{[1-benzyl-2-(2-methylpropanesulfonyl)-1H-imidazol-5-yl]methyl}[(1-ethylpiperidin-3-yl)methyl]methylamine
3-[5-(2,6-dimethylphenyl)-1,2,4-oxadiazol-3-yl]-6-methylpyridazine
4-(2-methyl-1H-imidazol-1-yl)-1-(pyrrolidine-1-sulfonyl)piperidine-4-carboxylic acid
2-(1-{[4-(pyrrolidine-1-carbonyl)phenyl]methyl}-1H-1,2,3-triazol-4-yl)benzoic acid
N-[(3S,4R)-1-(4,5-dimethylthiophene-2-carbonyl)-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
4-{2-[3-butyl-5-oxo-4-(2-phenylethyl)-4,5-dihydro-1H-1,2,4-triazol-1-yl]acetyl}piperazin-2-one
2-(1-{[2-(1H-pyrazol-1-yl)phenyl]methyl}-1H-1,2,3-triazol-4-yl)benzoic acid
6-{1-[4-(3-hydroxypyrrolidin-1-yl)pyrimidin-2-yl]piperidin-4-yl}-2-methylpyrimidin-4-ol
N'-cycloheptyl-N-(3-methoxypropyl)-N-(1-methylpiperidin-4-yl)butanediamide
[(3R,4R)-1-{[2-(morpholin-4-yl)pyrimidin-5-yl]methyl}-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
3-{5-[(2-{[(3S)-3-fluoropyrrolidin-1-yl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl)methyl]furan-2-yl}-1H-pyrazole
2-[(4-{5-[(2-methoxyethyl)sulfanyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)methyl]pyridine
8-[5-(hydroxymethyl)furan-2-carbonyl]-2-(3-methylbut-2-en-1-yl)-2,8-diazaspiro[4.5]decan-3-one
2-(3,4-dimethylphenoxy)-1-[(1R,5R)-6-methyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-3-(5-methylthiophen-2-yl)-5-(morpholine-4-sulfonyl)benzamide
3-methyl-6-[5-(1-methylcyclohexyl)-1,2,4-oxadiazol-3-yl]pyridazine