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4-[2-(4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-2,6-dimethylpyrimidine
(2S)-4-methyl-2-[4-(quinolin-4-yl)-1H-1,2,3-triazol-1-yl]pentan-1-ol
1-(2-fluorophenyl)-4-[(3-{[1-(furan-3-carbonyl)piperidin-3-yl]methoxy}phenyl)methyl]piperazine
9-[2-(4-hydroxyphenyl)acetyl]-2-(3-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
methyl 1-[1-(2-cyclohexylethyl)-1H-1,2,3-triazole-4-carbonyl]piperidine-4-carboxylate
2-[4-(2H-1,3-benzodioxol-4-ylmethyl)-1-(2,2-dimethylpropyl)piperazin-2-yl]ethan-1-ol
[(2S)-1-{[3-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]methyl}pyrrolidin-2-yl]methanol
2-(2,5-dimethoxyphenyl)-N-{[7-methoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}-N-[3-(2-oxopyrrolidin-1-yl)propyl]acetamide
{[1-benzyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}(methyl)[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amine
(2S)-2-[2-(2,4-dimethylbenzenesulfonamido)acetamido]-4-methylpentanamide
2-amino-1-[3-(naphthalen-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]ethan-1-one
N-[2-(cyclohex-1-en-1-yl)ethyl]-5-[(2S)-2-(hydroxymethyl)pyrrolidine-1-carbonyl]-1-[(2-methoxyphenyl)methyl]-4-oxo-1,4-dihydropyridine-3-carboxamide
2-[4-(dimethylamino)phenyl]-1-[4-(3-hydroxypiperidin-1-yl)piperidin-1-yl]ethan-1-one
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-[2-(4-methyl-1,2,5-oxadiazol-3-yl)acetyl]pyrrolidine-3-carboxylic acid
[(5-methoxy-1H-1,3-benzodiazol-2-yl)methyl](4-methoxy-4-methylpentan-2-yl)amine
(2S)-N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-2-hydroxy-3-phenylpropanamide
1-[4-(2-amino-4-phenylpyrimidine-5-carbonyl)-1,4-diazepan-1-yl]ethan-1-one
6-methyl-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-2-(pyridin-3-yl)pyrimidin-4-amine
2-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)-2-phenyl-1-[4-(pyridin-4-yl)piperidin-1-yl]ethan-1-one
N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
3-(azepane-1-carbonyl)-N-[(4-phenyloxan-4-yl)methyl]-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-[3-(1H-imidazol-1-yl)propyl]-6-methyl-2-[(2-methylphenyl)methyl]-4-oxo-1-(pyridin-2-ylmethyl)-1,4-dihydropyridine-3-carboxamide
N-[(1R,2S)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]-3-[(2-methylprop-2-en-1-yl)oxy]benzamide
N,5-dimethyl-2-(2-methylpropanamido)-N-[2-(2-oxopiperidin-1-yl)ethyl]benzamide
3-methyl-1-[2-oxo-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethyl]-4-(2-phenylethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[1-(6-methylpyridin-2-yl)propan-2-yl]benzamide
7-fluoro-3-(4H-1,2,4-triazol-4-ylmethyl)-1,2-dihydroquinolin-2-one
2-[2-(1-cyclobutyl-1H-imidazol-2-yl)phenoxy]ethan-1-ol
1'-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-5-methanesulfonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
6-[(2R,3R,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pyridine-3-carbonitrile
(3S,7S,8aS)-7-{[(2-chlorophenyl)methyl]amino}-3-(1H-indol-3-ylmethyl)-octahydropyrrolo[1,2-a]piperazine-1,4-dione
2-(dimethylamino)-N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N-methylbenzamide
7-methyl-2-(2-methyl-5-propylpyrimidin-4-yl)-2,7-diazaspiro[4.5]decan-6-one
N-(1-{1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-phenylacetamide
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-6-(2-hydroxyethyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
4-{1-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}morpholine
1-tert-butyl-3-[(3,4-dimethoxyphenyl)methyl]-5-(2-methyloxolan-2-yl)-1H-1,2,4-triazole
1-(2-methoxyphenyl)-N-[1-(thiophen-2-yl)propan-2-yl]-1H-pyrazole-4-carboxamide
2-(cyclopropylmethyl)-9-(1H-pyrazole-4-sulfonyl)-2,9-diazaspiro[5.5]undecan-3-one
1-{4-[({2-[4-(2-methylphenyl)piperazin-1-yl]pyridin-3-yl}methyl)amino]piperidin-1-yl}ethan-1-one
2-(5-acetylthiophen-3-yl)-N-(diphenylmethyl)acetamide
diethyl({2-[2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-1H-imidazol-1-yl]ethyl})amine
N-(2-chlorophenyl)-3-[(3-fluorophenyl)amino]piperidine-1-carboxamide
1-ethyl-2-(1-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}-1H-imidazol-2-yl)-1H-1,3-benzodiazole
[(2S)-1-({6-chloro-2-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]imidazo[1,2-a]pyridin-3-yl}methyl)pyrrolidin-2-yl]methanol
3-hydroxy-1-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}propan-1-one
1'-[2-(2,4-dimethyl-6-oxo-1,6-dihydropyrimidin-5-yl)acetyl]-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
2-{[3-(1-benzofuran-2-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}-7-methyl-2,7-diazaspiro[4.4]nonane
8-(6-aminohexanoyl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
4-(3-{[(3R)-3-methylpiperazin-1-yl]sulfonyl}benzoyl)thiomorpholine