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2,3,5,6-tetramethyl-N-({1-[(4-methylpiperazin-1-yl)methyl]cyclopropyl}methyl)benzamide
2-(2-{1-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)sulfonyl]piperidin-4-yl}-1H-imidazol-1-yl)acetamide
1-{4-[methyl(propyl)amino]piperidin-1-yl}ethan-1-one
6-amino-N-{[(1r,4r)-4-(methylcarbamoyl)cyclohexyl]methyl}pyridine-2-carboxamide
1-[2-(dimethylamino)-6-(3,6-dimethylpyrazin-2-yl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-4-yl]piperidin-4-ol
3-[5-(2H-1,3-benzodioxol-5-yl)-1,3,4-oxadiazol-2-yl]-1-[4-(benzyloxy)piperidin-1-yl]propan-1-one
2-(4-{[2-(hydroxymethyl)azepan-1-yl]methyl}phenoxy)ethan-1-ol
2-(4-ethylpiperazin-1-yl)-N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]-2,3-dihydro-1H-indene-2-carboxamide
3-[2-(5-ethylpyridin-2-yl)ethyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidin-1-yl]-2-(pyrrolidin-1-yl)ethane-1,2-dione
2-[(6-methyl-1H-1,3-benzodiazol-2-yl)methoxy]-N-{1-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]ethyl}acetamide
8-[3-(1H-1,3-benzodiazol-1-yl)propanoyl]-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
N-{4-[2-(1-methyl-1H-imidazol-2-yl)-1H-imidazol-1-yl]phenyl}pyridine-3-carboxamide
3-({2-amino-4H,5H,6H,7H-[1,3]thiazolo[5,4-c]pyridin-5-yl}methyl)-N-(5-methylpyridin-3-yl)benzamide
N-[3-(4-hydroxyphenyl)propyl]-5-oxo-1-(pyridin-4-ylmethyl)pyrrolidine-3-carboxamide
3-(furan-2-yl)-5-{2-[3-(2-methylpropyl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl]ethyl}-1,2,4-oxadiazole
1-[2-(oxolan-2-ylmethoxy)acetyl]-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
3-(3-fluorophenyl)-5-(5-methylthiophene-2-carbonyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
4,6-dimethyl-3-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
3-{[4-(cyclopropylmethyl)-5-oxo-3-(propan-2-yl)-1,4-diazepan-1-yl]methyl}-1,2-dihydroquinoxalin-2-one
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-N-methyl-2-(methylsulfanyl)-1,3-thiazole-4-carboxamide
4-(2H-1,3-benzodioxol-5-yloxy)-1-(2-methylpyrimidin-4-yl)piperidine-4-carboxylic acid
(5S,9aS,9bS)-5-{5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}-2-(2-phenylethyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-(2,3-dihydro-1,4-benzodioxine-2-carbonyl)-4-(4-ethyl-1H-pyrazol-5-yl)piperidine
6-methyl-2-{4-[4-(4-methylphenyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}pyridine-3-carboxamide
N-(4-{[methyl({[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl})amino]methyl}phenyl)acetamide
1-[(3R,4R)-4-{2-[3-(1H-pyrazol-1-yl)phenyl]-1H-imidazol-1-yl}oxolan-3-yl]piperidine
N-(2-fluoro-5-methylphenyl)-2-[4-(pyrrolidine-1-sulfonyl)morpholin-3-yl]acetamide
N-methyl-5-propyl-N-(quinolin-8-ylmethyl)-1,3,4-oxadiazole-2-carboxamide
5-benzamido-1-cyclopentyl-N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-1H-1,3-benzodiazole-7-carboxamide
3-[1-(2,1-benzoxazole-3-carbonyl)piperidin-3-yl]-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
1-(1-benzofuran-2-carbonyl)-N-(3,4-difluorophenyl)piperidin-3-amine
(2S,4S)-4-cyclopentaneamido-N,N-diethyl-1-[(5-methylfuran-2-yl)methyl]pyrrolidine-2-carboxamide
1-(2-methoxyacetyl)-N,4-dimethyl-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}piperazine-2-carboxamide
4-[5-(3-hydroxy-3-methylbut-1-yn-1-yl)thiophen-2-yl]-3-phenyl-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
[(3R,4R)-4-(azepan-1-ylmethyl)-1-[(1-methyl-1H-imidazol-2-yl)methyl]pyrrolidin-3-yl]methanol
(4aS,7aR)-1-(2-chlorobenzoyl)-4-(cyclopropylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
methyl (2S)-1-{2-[4-(4-{[2-(pyrazin-2-yl)ethyl]amino}piperidin-1-yl)phenyl]acetyl}pyrrolidine-2-carboxylate
5-methyl-4-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}pyrimidin-2-amine
1-{[3-(cyclopropylmethyl)-1,2,4-oxadiazol-5-yl]methyl}-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(dimethyl-1,3-oxazole-5-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
(3S)-1-[2-(4-ethylpiperazin-1-yl)-2,3-dihydro-1H-indene-2-carbonyl]pyrrolidin-3-ol
3-(4-cyclohexyl-1,4-diazepane-1-carbonyl)-N,N-dimethylaniline
methyl 1-[2-(1H-indol-3-yl)ethyl]-3-(3-methoxypropanamido)-5-[(oxan-4-yl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
5-(methoxymethyl)-N-({7-[(2-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)furan-2-carboxamide
2-(1-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}piperidin-3-yl)-1,2,3,4-tetrahydroisoquinoline
3-{4-[(1-methylpiperidin-4-yl)methyl]piperazin-1-yl}-1-(1,2,3,4-tetrahydroquinolin-1-yl)propan-1-one
2-cyclopentyl-N-(furan-2-ylmethyl)-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
N-[(2-ethoxy-3-methoxyphenyl)methyl]-N,1,3-trimethyl-1H-indole-2-carboxamide
1-[(4-fluoro-3-methylphenyl)methyl]-3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine