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N-(oxolan-3-yl)-4-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butanamide
N-cyclopropyl-2-fluoro-5-sulfamoyl-N-(thiophen-3-ylmethyl)benzamide
3-methyl-N-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)-3H-[1,2,3]triazolo[4,5-b]pyridine-6-carboxamide
6-(2-methoxyphenyl)-N-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)pyridazin-3-amine
1-(carbamoylmethyl)-N-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)piperidine-3-carboxamide
N-{[5-(2-acetylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(3-methylphenyl)acetamide
2-(2,4-dimethyl-6-oxo-1,6-dihydropyrimidin-5-yl)-N-[1-(thiophen-2-yl)propyl]acetamide
N5-{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}-N2,N2-dimethyl-5,6,7,8-tetrahydroquinazoline-2,5-diamine
3-[(3R,4S)-4-(morpholin-4-yl)-1-(2,4,5-trimethylbenzoyl)piperidin-3-yl]propan-1-ol
N-ethyl-3,5-difluoro-N-[2-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]pyridine-2-carboxamide
3-bromo-5-[(pyridin-3-ylmethyl)sulfamoyl]benzoic acid
3-(1H-imidazol-2-yl)-1-[7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carbonyl]piperidine
4-[3-(2,6-dimethylphenoxy)azetidin-1-yl]-5-methylpyrimidin-2-amine
2-[1-(5-chloropyridine-2-carbonyl)pyrrolidin-2-yl]-5-fluoro-1H-1,3-benzodiazole
1-[(4-fluorophenyl)methyl]-4-[5-oxo-1-(propan-2-yl)pyrrolidine-3-carbonyl]piperazin-2-one
4-[(7-chloro-2-methylquinolin-4-yl)formamido]-N-methylbutanamide
N-[4-(1H-1,3-benzodiazol-2-yl)phenyl]-1-(2-hydroxyacetyl)piperidine-4-carboxamide
8-(2,6-dimethylbenzoyl)-2-(3-methoxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
N-cyclopentyl-2-(methylsulfanyl)-N-(3-phenylprop-2-yn-1-yl)acetamide
N-[(3S,4R)-1-[2-(2-fluorophenyl)benzoyl]-4-propylpyrrolidin-3-yl]acetamide
N-(pyridin-3-yl)-3-({1-[2-(trifluoromethyl)phenyl]ethyl}amino)propanamide
7-[4-(pyridin-2-ylmethyl)-1,4-diazepane-1-carbonyl]-1,2,3,4-tetrahydroquinoxalin-2-one
1-[cyclohexyl(methyl)amino]-3-(3-{[ethyl(pyridin-4-ylmethyl)amino]methyl}phenoxy)propan-2-ol
N-(1-benzylpiperidin-3-yl)-1-[4-(furan-2-yl)pyrimidin-2-yl]-5-(methoxymethyl)-1H-pyrazole-4-carboxamide
N,N-dimethyl-1-(prop-2-en-1-yl)-5-{[2-(thiophen-2-yl)ethyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
7-(2-cyclohexylethyl)-2-(2-methoxyacetyl)-2,7-diazaspiro[4.5]decan-6-one
2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(3-methylbutyl)acetamide
N-(furan-2-ylmethyl)-N-{[2-(4-hydroxypiperidin-1-yl)-7-(methylsulfanyl)quinolin-3-yl]methyl}-4-(1H-pyrazol-1-yl)benzamide
4-(furan-2-yl)-N-methyl-N-[(1-methylpyrrolidin-2-yl)methyl]benzamide
N-[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]-5-ethyl-N,2,3-trimethylpyrazolo[1,5-a]pyrimidin-7-amine
4-(2,3-dimethoxybenzoyl)-1-(2-methylphenyl)piperazin-2-one
(2R)-2-[4-phenyl-5-(2,3,4-trimethoxyphenyl)-1H-imidazol-1-yl]propanamide
7-(2-ethoxyethoxy)-4-[4-(propan-2-yl)-1,3-thiazol-2-yl]-1,2,3,4-tetrahydroquinolin-2-one
4-[4-(4-ethyl-1H-pyrazol-5-yl)piperidin-1-yl]-2-methyl-5-propylpyrimidine
N-[(8-methoxyquinolin-5-yl)methyl]-N-methyl-1,4-dithiepan-6-amine
4-[1-(furan-3-ylmethyl)-4-phenyl-1H-imidazol-5-yl]phenol
N-[2-(1H-imidazol-1-yl)ethyl]-5-[3-(trifluoromethyl)phenyl]-1,2,4-triazin-3-amine
N-(4-methoxy-3-propanamidophenyl)-2-methyl-4-oxo-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carboxamide
methyl({[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}){[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
N-[(5-methyl-1,2-oxazol-3-yl)methyl]-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]acetamide
1-methyl-N-{1-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl}-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
(3S,4S)-4-cyclopropyl-1-[2-(4-methanesulfonylphenyl)acetyl]pyrrolidine-3-carboxylic acid
N-(6-methoxy-2H-1,3-benzodioxol-5-yl)-3-methyl-2-oxo-1-oxa-3,8-diazaspiro[4.5]decane-8-carboxamide
ethyl 1-(1H-imidazol-4-ylmethyl)-3-[(3-methoxyphenyl)methyl]piperidine-3-carboxylate
4-phenyl-N-{1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}butanamide
2-cyclopropyl-N-[3-(6-methyl-1,3-benzoxazol-2-yl)propyl]-6-oxo-1,6-dihydropyrimidine-5-carboxamide
3-benzyl-8-(furan-3-ylmethyl)-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[2-(5-{[(3-chlorophenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-3,4,5-trimethoxybenzamide
3-phenyl-N-{1-[1-(1,3-thiazol-2-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}propanamide
3-[(7-methanesulfonyl-4-methylquinazolin-2-yl)(methyl)amino]propane-1,2-diol