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N-[(3S,4R)-1-cyclohexanecarbonyl-4-(4-methylphenyl)pyrrolidin-3-yl]acetamide
1-{[3-(1-benzofuran-2-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}azetidin-3-ol
N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-2-(7-methyl-3-oxo-3,4-dihydro-2H-1,4-benzothiazin-4-yl)acetamide
1-{2-[methyl({[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl})amino]pyrimidin-4-yl}pyrrolidin-3-ol
5-(oxolan-2-yl)-N-{[4-(2-oxopyrrolidin-1-yl)phenyl]methyl}thiophene-2-carboxamide
N-methyl-2-oxo-N-(1H-pyrazol-3-ylmethyl)-1-[(1r,4r)-4-hydroxycyclohexyl]-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
2-(pyrimidin-2-ylsulfanyl)-N-({5-[3-(trifluoromethoxy)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methyl)acetamide
methyl 2-{3-[3-(pyridin-4-yl)phenyl]-1H-pyrazol-1-yl}butanoate
1-methanesulfonyl-N-[1-(3-methoxyphenyl)propan-2-yl]piperidin-4-amine
3-[1-(2,3-dihydro-1-benzofuran-7-carbonyl)piperidin-3-yl]-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
(5R)-5-[1-(2-methyl-1,3-benzothiazol-6-yl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]pyrrolidin-2-one
(2R,6R)-4-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
N-{2-[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
1-[4-(3-methylpyridin-2-yl)piperazin-1-yl]-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propan-1-one
5-(4-chlorophenoxy)-4-{5H,6H,7H,8H-imidazo[1,5-a]pyrazin-7-ylmethyl}-1,3-dimethyl-1H-pyrazole
N-(2-{7-[(5-methylfuran-2-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2-phenoxyacetamide
4-(4-chlorophenyl)-1-[4-(4-hydroxypiperidin-1-yl)piperidin-1-yl]butan-1-one
3-[2-methoxy-5-(4H-1,2,4-triazol-4-yl)phenyl]-1-methyl-1-[1-(4-methylpyridin-2-yl)propan-2-yl]urea
1-cyclooctyl-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
4-(cyclopentylamino)-N-[(3-fluorophenyl)methyl]-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
2-(pyridin-2-yl)-5-({spiro[indene-1,4'-piperidine]-1'-yl}carbonyl)pyrimidin-4-ol
N-{2-[7-(cyclohexylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}oxolane-2-carboxamide
1-{dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}-4-phenylazepane
3-[1-(dimethyl-1,3-thiazol-2-yl)propyl]-1-(4-methyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-7-yl)urea
2-[methyl(phenyl)amino]-1-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}ethan-1-one
N-(4-fluoro-2-methylphenyl)-3-[1-(thian-4-yl)piperidin-3-yl]propanamide
N-butyl-2-(1,4-dimethylpiperazin-2-yl)-N-[(3-methoxyphenyl)methyl]acetamide
N-[2-(6-oxo-3-phenyl-1,6-dihydropyridazin-1-yl)ethyl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-[(3-methoxyphenyl)methyl]-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-6-oxopiperidine-3-carboxamide
(1-{2-[(5-ethyl-1,3,4-oxadiazol-2-yl)amino]ethyl}piperidin-2-yl)methanol
2-{3-[(1R,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-3-oxopropyl}-2,3-dihydro-1H-isoindol-1-one
N-ethyl-1-[(2-fluorophenyl)methyl]-N-(4-hydroxybutyl)-6-oxopiperidine-3-carboxamide
1-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]ethan-1-one
N-{[5-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-3-yl]methyl}-1,9-dioxaspiro[5.5]undecan-4-amine
5-(3-{2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl}-3-oxopropyl)imidazolidine-2,4-dione
N-benzyl-1-methyl-5-(quinolin-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-(1-methyl-1H-pyrrole-2-carbonyl)-N-[4-(1H-pyrazol-5-yl)phenyl]piperidine-3-carboxamide
N-[3-methyl-1-(7-{[3-(trifluoromethyl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)butyl]furan-2-carboxamide
N-(1-cycloheptyl-5-oxopyrrolidin-3-yl)-3-(dimethylamino)benzamide
4-(5-methylpyridin-2-yl)-1-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}piperidin-4-ol
2-amino-6-(3,5-dimethylphenyl)-4-(oxolan-3-yl)pyridine-3-carbonitrile
2-[(2-methyl-1,3-oxazol-4-yl)methyl]-2-azatricyclo[6.3.1.04,12]dodeca-1(12),4,6,8,10-pentaen-3-one
2-phenyl-N-[1-(1-propyl-1H-1,2,4-triazol-5-yl)ethyl]imidazo[1,2-a]pyridine-6-carboxamide
1-{4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}-2-(1H-pyrazol-1-yl)butan-1-one
1-(4-chlorophenyl)-4-({3-[(3-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)piperazine
2-[5-(1-{[5-(propan-2-yl)-1,3,4-oxadiazol-2-yl]methyl}pyrrolidin-2-yl)-1,2,4-oxadiazol-3-yl]pyridine
(1R,5S,6S)-6-{[4-(3-methylphenoxy)piperidin-1-yl]methyl}-3-azabicyclo[3.1.0]hexane
3-(5-{[3-(2-phenylethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}thiophen-3-yl)prop-2-yn-1-ol
4-(1H-1,2,4-triazol-1-yl)-1-{3-[3-(trifluoromethyl)benzoyl]piperidin-1-yl}butan-1-one
3-[1-methyl-10-oxo-9-(prop-2-en-1-yl)-1,4,9-triazaspiro[5.6]dodecan-4-yl]propanamide