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2-[1-(2,3-dihydro-1H-inden-2-yl)-3-oxopiperazin-2-yl]-N-ethyl-N-(pentan-3-yl)acetamide
{[4-cyclopropyl-5-(1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidin-4-yl)-4H-1,2,4-triazol-3-yl]methyl}dimethylamine
N-({3-methoxy-4-[2-(pyridin-2-yl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]naphthalene-1-sulfonamide
2-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-4-phenyl-1,2-dihydrophthalazin-1-one
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-{3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}piperidin-3-ol
N-(2,2-diethyl-3-hydroxypropyl)-N,1-dimethyl-3-propyl-1H-pyrazole-5-carboxamide
2-ethoxy-5-(2-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}pyrimidin-4-yl)benzoic acid
1-methyl-N-({2-[4-(2-methylphenyl)piperazin-1-yl]pyridin-3-yl}methyl)piperidine-2-carboxamide
(2S,4R)-4-(2,4-difluorobenzamido)-N-(1H-indol-4-ylmethyl)pyrrolidine-2-carboxamide
1-[4-(2H-1,3-benzodioxol-5-yl)pyrimidin-2-yl]-N-benzyl-5-cyclopropyl-N-(2-hydroxyethyl)-1H-pyrazole-4-carboxamide
(4aS,8aR)-6-(2-amino-6-methylpyrimidin-4-yl)-1-[2-(thiophen-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
N-methyl-N-{1-[1-(6-oxo-1,4,5,6-tetrahydropyridazine-3-carbonyl)piperidin-4-yl]-2-phenylethyl}thiophene-2-carboxamide
(4aR,7aS)-N,N-dimethyl-6,6-dioxo-4-(pyridazine-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
6-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidine-1-carbonyl]-2,3-dihydropyridazin-3-one
N,N-dimethyl-2-{3-[1-(pyridin-3-ylmethyl)-1H-pyrazol-3-yl]phenyl}benzamide
6-{3-[(2,4-difluorophenyl)methyl]-3-(hydroxymethyl)piperidin-1-yl}pyridine-3-carbonitrile
(1-{3-[1-(furan-3-ylmethyl)-1H-imidazol-2-yl]phenyl}ethyl)dimethylamine
2-(4-{[2-(2,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-1-yl)-N-(propan-2-yl)acetamide
N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)piperidin-4-yl]methyl}-2-(methylamino)pyrimidine-5-carboxamide
1-(2-{2-benzyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carbonyl}phenyl)ethan-1-one
5-{[1-(4-methyl-1,4-diazepan-1-yl)hex-5-en-2-yl]oxy}pyridine-2-carbonitrile
4-({4-[1-(4-methylpiperazin-1-yl)ethyl]piperidin-1-yl}methyl)phenol
1-({3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)piperidine-4-carboxamide
1-(6-{[2-methyl-2-(morpholin-4-yl)propyl]amino}pyridin-3-yl)ethan-1-one
5-methyl-1-[4-(5-methylfuran-2-yl)pyrimidin-2-yl]-N-[(1-methylpiperidin-3-yl)methyl]-1H-pyrazole-4-carboxamide
4-benzyl-3-ethyl-1-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)-1,4-diazepan-5-one
2-(1-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-1H-1,2,3-triazol-4-yl)benzoic acid
7-fluoro-2-(pyrimidin-5-yl)-4-[(2S)-2-(pyrrolidin-1-ylmethyl)pyrrolidine-1-carbonyl]quinoline
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2-[4-(pyrimidin-2-yl)piperazin-1-yl]acetamide
6-[(2E)-3-(3,4-dimethoxyphenyl)prop-2-enoyl]-N-[3-(pyridin-4-yl)propyl]-6-azaspiro[2.5]octane-1-carboxamide
3-[(4-methoxyphenyl)methyl]-1-(3-methoxypropyl)-8-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-benzyl-7-(furan-2-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
1-(3-chloro-2,6-dimethylphenyl)-3-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]urea
3-(1,3-dihydro-2-benzofuran-5-yl)-1-(oxolan-2-ylmethyl)-1-(pyridin-2-ylmethyl)urea
13-(2,1,3-benzothiadiazol-4-yl)-5-thia-2,7,10-triazatricyclo[6.5.0.02,6]trideca-1(8),3,6-trien-11-one
1-(3-hydroxypropyl)-N-[3-(3-methoxyphenyl)phenyl]piperidine-2-carboxamide
3-[1-(2,1,3-benzoxadiazol-5-ylmethyl)piperidin-3-yl]-N-[(2,4-dimethoxyphenyl)methyl]propanamide
5-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]-N-[2-(1-methylpyrrolidin-2-yl)ethyl]pyridin-2-amine
2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-{2-[2-(propan-2-yl)-1,3-thiazol-4-yl]ethyl}acetamide
4-chloro-N-(2-hydroxy-2-phenylethyl)-1,5-dimethyl-N-(pyridin-4-ylmethyl)-1H-pyrazole-3-carboxamide
5-(cycloheptylamino)-1-ethyl-N-(furan-3-ylmethyl)-N-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-[(2,3-difluorophenyl)methyl]-3-hydroxy-3-({[(6-methylpyridin-2-yl)methyl]amino}methyl)piperidin-2-one
5-{2-[2-(1H-1,3-benzodiazol-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl]-2-oxoethyl}pyrrolidin-2-one
2-(2-{1-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]piperidin-4-yl}-1H-imidazol-1-yl)acetamide
1-[4-(4-methoxybenzoyl)piperazin-1-yl]-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
3-(2,4-dichloro-3-methylphenyl)-1-{3-[3-(hydroxymethyl)piperidin-1-yl]propyl}urea
1-[1-(4-methoxyphenyl)-2,2-dimethylcyclopropanecarbonyl]azetidin-3-ol
N-methyl-2-(methylsulfanyl)-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}benzamide
4,4,4-trifluoro-N-[(1-methylpyrrolidin-3-yl)methyl]butanamide
2-(2-{[(3-methoxyphenyl)methyl](methyl)amino}pyrimidin-4-yl)pyridine-4-carboxylic acid