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N-butyl-7-[(3-methylphenyl)methyl]-6-oxo-2,7-diazaspiro[4.5]decane-2-carboxamide
N-[(2-benzyl-1,3-thiazol-4-yl)methyl]-3-propyl-1H-pyrazole-5-carboxamide
N-benzyl-2-(1H-1,2,4-triazol-3-yl)-N-(2,2,2-trifluoroethyl)benzamide
2-[3-(4-phenyl-1H-imidazol-1-yl)phenoxy]acetamide
1-(4-{[4-(aminomethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)-2-(phenylsulfanyl)ethan-1-one
1-(2-methylphenyl)-4-{1-[(2E)-3-phenylprop-2-en-1-yl]piperidin-3-yl}piperazine
N-[(2-methoxyphenyl)methyl]-3-(1,2-oxazolidin-2-yl)-N-(pyridin-3-ylmethyl)propanamide
(1S,5R)-3-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[3-(2-ethoxyethoxy)phenyl]-2-(2-hydroxyethyl)-3-oxopiperazine-1-carboxamide
(2S,4S)-4-amino-1-[(6,8-dimethyl-2-oxo-1,2-dihydroquinolin-3-yl)methyl]-N-methylpyrrolidine-2-carboxamide
1-[1,3-dioxo-2-(pyridin-2-ylmethyl)-2,3-dihydro-1H-isoindol-4-yl]-N-[(4-methoxyphenyl)methyl]piperidine-3-carboxamide
N-cyclopropyl-3-{1-[2-(4-methylphenoxy)acetyl]piperidin-3-yl}propanamide
1-{4-[(2,2-dimethylmorpholin-4-yl)methyl]-2-methoxyphenoxy}-3-[methyl(propan-2-yl)amino]propan-2-ol
(1S,4S)-2-(2-methoxy-5-phenylphenyl)-5-(6-methylpyrimidin-4-yl)-2,5-diazabicyclo[2.2.1]heptan-3-one
N-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-2-{1-[(2-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-methylacetamide
7-methyl-3-(3-phenylbutyl)-3,7,11-triazaspiro[5.6]dodecan-12-one
3-(3,4-dimethyl-1H-pyrazol-5-yl)-N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}propanamide
3-({methyl[2-(oxan-2-yl)ethyl]amino}methyl)pyridin-2-amine
6-(4-tert-butylbenzoyl)-N-[2-(pyridin-2-yl)ethyl]-6-azaspiro[2.5]octane-1-carboxamide
2-(6-methoxy-2H-1,3-benzodioxol-5-yl)-1H-1,3-benzodiazole-5-carbonitrile
3-(2-fluorophenyl)-1-(2-methoxyethyl)-3-{2-[3-(2-methylphenoxymethyl)piperidin-1-yl]-2-oxoethyl}pyrrolidine-2,5-dione
5-[(1-benzylpiperidin-4-yl)amino]-1-ethyl-N-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-[(3R,5S)-5-(diethylcarbamoyl)-1-(2-methoxyacetyl)pyrrolidin-3-yl]-1H-pyrrole-3-carboxamide
(3S,4S)-1-(2-ethylpyrimidine-5-carbonyl)-4-(naphthalen-2-yl)piperidin-3-ol
2-ethoxy-4-{[({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)(2-methoxyethyl)amino]methyl}phenol
3-methoxy-N-(1-{7-[(2-methoxynaphthalen-1-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)benzamide
1-[2-(4-chlorophenyl)ethyl]-6-oxo-N-(pentan-3-yl)piperidine-3-carboxamide
N-{[3-(3,4-difluorophenyl)phenyl]methyl}propanamide
methyl 2-[(3aR,7aS)-5-methyl-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-yl]-3-ethyl-3H-imidazo[4,5-b]pyridine-6-carboxylate
5-(2H-1,3-benzodioxol-5-ylmethyl)-5-methyl-1-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]piperidin-2-one
[(4-chloro-3-fluorophenyl)methyl](ethyl){[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}amine
{4-[4-(trifluoromethyl)pyridin-2-yl]phenyl}methanol
3-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methylpropanamide
{5-[1-(1H-indol-4-ylmethyl)-4-phenyl-1H-imidazol-5-yl]furan-2-yl}methanol
(3E)-2-{[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl](methyl)amino}-5,5-dimethylhex-3-enoic acid
1-cyclobutyl-4-{4-[(3,3-diethylpyrrolidin-1-yl)methyl]-1H-1,2,3-triazol-1-yl}piperidine
2,6-dihydroxy-N-[(2-propyl-1,3-thiazol-4-yl)methyl]benzamide
1-[(1-cyclopropyl-1H-imidazol-2-yl)methyl]-1,2-dihydroquinoxalin-2-one
ethyl 4-benzyl-1-[(1-ethyl-1H-pyrazol-4-yl)methyl]piperidine-4-carboxylate
N-[(1-{[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}piperidin-3-yl)methyl]acetamide
3-(2-chloro-4-fluoro-5-methylphenyl)-1-[(2-ethoxyphenyl)methyl]-1-(2-hydroxyethyl)urea
2-{1-[(2-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-{[1-(hydroxymethyl)cyclobutyl]methyl}-N-methylacetamide
2-(2-aminoethyl)-N-[3-(oxolan-3-yl)propyl]quinazolin-4-amine
4-(1-{2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]ethyl}-1H-imidazol-2-yl)-3-methoxyphenol
2-methoxyethyl 3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carboxylate
N-(2-{[5-(1,5-dimethyl-1H-pyrazol-4-yl)-1,2-oxazol-3-yl]formamido}ethyl)-4-fluorobenzamide
3-[1-(1-methylcyclohexanecarbonyl)piperidin-3-yl]-1-[4-(pyridin-2-yl)piperazin-1-yl]propan-1-one
3-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[3-(1H-indazol-1-yl)propyl]-2-(6-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)acetamide
(5S,9aS,9bS)-5-(4-fluoro-3-methoxyphenyl)-2-[(5-methylfuran-2-yl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one