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1,6-dimethyl-3-[3-(1-methyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-1,4-dihydroquinolin-4-one
1-cyclopropyl-4-[5-(2,3-dihydro-1,4-benzodioxin-6-yl)-1H-imidazol-2-yl]pyrrolidin-2-one
N-[1-methyl-3-(pyridin-2-yl)-1H-pyrazol-5-yl]-2-(4-phenyl-1H-imidazol-1-yl)acetamide
9-(2,6-difluoro-3-methylbenzoyl)-2-(2-methoxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-methyl-3-{4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazine-1-carbonyl}-2,8-diazaspiro[4.5]decane
5-{3-[(4-methoxyphenyl)methyl]-1,2,4-oxadiazol-5-yl}-N-[1-(1-methyl-1H-pyrazol-4-yl)ethyl]pyridin-2-amine
1-(2-cyclopropylphenyl)-3-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}urea
N-(4-chloro-3-fluorophenyl)-4-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidine-1-carboxamide
4-[(2-fluorophenyl)methyl]-1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-1,4-diazepan-5-one
3-[5-(6-methoxy-2,3-dihydro-1H-inden-5-yl)-4-phenyl-1H-imidazol-1-yl]propan-1-ol
1-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]-3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
N-ethyl-4-({methyl[(2-methyl-2,3-dihydro-1H-isoindol-5-yl)methyl]carbamoyl}amino)benzamide
7-[3-(hydroxymethyl)-3-(2-methoxyethyl)piperidine-1-carbonyl]-3,4-dihydro-2H-1,4-benzoxazin-3-one
2-(3-fluorophenyl)-N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(pyridin-3-ylmethyl)acetamide
5-chloro-2-{4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridine
9-(3-ethyl-1H-indole-2-carbonyl)-3-oxa-9-azaspiro[5.5]undecane
2-({2-[benzyl(methyl)amino]-2,3-dihydro-1H-inden-2-yl}formamido)acetamide
2-(dimethylamino)-N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N,4-dimethylpyrimidine-5-carboxamide
6-methyl-2-oxo-N-[(5-oxo-1-phenylpyrrolidin-3-yl)methyl]-1,2-dihydropyridine-4-carboxamide
(3R,4S)-4-[ethyl(3-phenylpropyl)amino]oxolan-3-ol
N-({4-benzyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)-4-methoxybenzamide
({4-[1-(2-ethyl-4-methyl-1,3-thiazole-5-carbonyl)piperidin-2-yl]phenyl}methyl)dimethylamine
1-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-4-(1H-1,2,3,4-tetrazol-1-yl)butan-1-one
N-[2-(4-amino-6-hydroxypyrimidin-2-yl)ethyl]-2-(dimethylamino)-2-(2-methylphenyl)acetamide
1-[(1S,5R)-3-benzoyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(3-methoxyphenyl)propan-1-one
N-[1-(4-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3,5-dimethyl-1,2-oxazole-4-carboxamide
1-(4-{4-[(dimethylamino)methyl]-4-hydroxypiperidin-1-yl}-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
1-ethyl-N-[2-(furan-2-yl)ethyl]-5-(2-methoxyacetamido)-2-(pyridin-3-yl)-1H-1,3-benzodiazole-7-carboxamide
3-(2-methoxyphenyl)-N-[2-(2-methylpyridin-4-yl)-1,2,3,4-tetrahydroisoquinolin-7-yl]propanamide
methyl 3-cyclobutaneamido-5-{[(3,5-difluorophenyl)methyl]amino}-1-[2-(pyridin-2-yl)ethyl]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
3-(2-{[3-(trifluoromethyl)phenyl]methyl}morpholin-4-yl)propan-1-ol
N-cyclohexyl-3-[methyl(quinolin-5-ylmethyl)amino]propanamide
5-methanesulfonyl-1'-(6-methylpyridazin-3-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
3-[2-(3,4-difluorophenyl)ethyl]-1-(1-propyl-1H-pyrazole-5-carbonyl)piperidine
1-(2-phenylethyl)-3-(pyridin-3-ylmethyl)-8-(pyridin-4-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}-2-(methylamino)acetamide
2-(dimethylamino)-N-{[4-(dimethylamino)oxan-4-yl]methyl}-2-(2-fluorophenyl)acetamide
N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepine-3-carboxamide
1-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-(2-methoxyethyl)-5-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-1H-1,2,4-triazole
2-methyl-2-[4-(morpholin-4-yl)-2-{[(1r,4r)-4-hydroxycyclohexyl]amino}pyrimidin-5-yl]propanoic acid
4-[2-(3-fluorophenyl)ethyl]-11-(morpholin-4-yl)-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
N-benzyl-N-methyl-3-{1-[(1R,2R)-2-phenylcyclopropanecarbonyl]piperidin-4-yl}propanamide
3-[(3R,4S)-1-(2,6-difluorobenzoyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
N-cyclopropyl-1-[1-(2-phenylethyl)piperidin-4-yl]piperidine-3-carboxamide
4-[2-(3-fluoro-4-hydroxyphenyl)acetyl]-5-methyl-1-(3-methylphenyl)piperazin-2-one
2-({4-[(3R,4S)-3-amino-4-(3-methoxyphenyl)pyrrolidine-1-carbonyl]phenyl}sulfanyl)ethan-1-ol
6-(2-chlorophenyl)-N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}imidazo[2,1-b][1,3]thiazole-3-carboxamide
4-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-1-(cyclopropylmethyl)-2-(propan-2-yl)-1,4-diazepane
(3S,4S)-4-cyclopropyl-1-[2-(dimethylamino)-4-methylpyrimidine-5-carbonyl]pyrrolidine-3-carboxylic acid
N-[(2-ethyl-3-methyl-1H-indol-5-yl)methyl]-6-(4H-1,2,4-triazol-4-yl)pyridine-3-carboxamide