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1-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-(phenoxymethyl)-5-(pyrrolidin-3-yl)-1H-1,2,4-triazole
5-{3-[2-(3-methoxyphenyl)ethyl]piperidine-1-carbonyl}quinoxaline
1-[2-(phenylsulfanyl)ethyl]-4-(pyridin-3-ylmethyl)-1,4-diazepane
4-({[2-(2-ethylphenoxy)ethyl](methyl)carbamoyl}amino)-3-methylbenzamide
4-[({2,3-dimethyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]benzene-1,3-diol
2-(4-fluorophenyl)-N-[1-(1H-1,2,3,4-tetrazol-5-yl)ethyl]imidazo[1,2-a]pyridine-6-carboxamide
5-{[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-2-methyl-1H-pyrrole-3-carbonitrile
1-tert-butyl-4-(3-propyl-1,2,4-oxadiazol-5-yl)pyrrolidin-2-one
N-[2-(1H-imidazol-1-yl)propyl]-2-(pyridin-2-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
5-{2-[(1H-1,3-benzodiazol-2-ylmethyl)amino]pyrimidin-4-yl}-2-ethoxybenzoic acid
1-[2-methoxy-4-({[2-(4-methylphenyl)ethyl]amino}methyl)phenoxy]-3-(pyrrolidin-1-yl)propan-2-ol
3-chloro-N-[(3S,4S)-4-ethoxy-1-methylpyrrolidin-3-yl]-4-fluoro-1-benzothiophene-2-carboxamide
N-(2-{1-[(3-hydroxyphenyl)methyl]piperidin-3-yl}ethyl)ethane-1-sulfonamide
4-(1-methyl-1H-pyrazole-3-carbonyl)-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-({1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]piperidin-3-yl}methyl)-2-hydroxypyridine-3-carboxamide
1-[5-(3-chlorothiophene-2-carbonyl)-1-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]-4-phenylpiperazine
2-(1-{[2-(3,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1H-pyrazol-4-yl)ethan-1-ol
(3S,4S)-4-cyclopropyl-1-{[(4-methoxyphenyl)methyl]carbamoyl}pyrrolidine-3-carboxylic acid
N'1-[(3R,4S)-4-cyclopropyl-1-[(trimethyl-1H-imidazol-2-yl)methyl]pyrrolidin-3-yl]cyclopropane-1,1-dicarboxamide
3-(2-benzyl-5-oxopyrrolidin-2-yl)-N-(2,3-dihydro-1-benzofuran-2-ylmethyl)-N-methylpropanamide
1-[5-(2-fluoro-6-methoxyphenyl)thiophen-2-yl]propan-1-one
{[1-(2,4-difluorophenyl)-3-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}(2-methoxyethyl)methylamine
2-{6-hydroxy-4-[2-(3-methylphenyl)acetyl]-1,4-diazepan-1-yl}acetic acid
ethyl 2-[3-(1H-pyrazol-3-yl)phenyl]pyridine-3-carboxylate
4-{4-[4-(2,4-dimethylphenyl)piperazine-1-carbonyl]piperidin-1-yl}-2-(pyridin-3-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
N-methyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]-3-(pyridin-3-yl)propanamide
2,3-dimethyl-6-(3,4,7-trimethyl-1H-indole-2-carbonyl)-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
4-[4-(4-acetylpiperazin-1-yl)piperidin-1-yl]-N-(1-phenylethyl)benzamide
3-chloro-5-{2,3-dimethyl-4-oxo-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-7-carbonyl}-1,2-dihydropyridin-2-one
3-[({1-[2-(thiophen-2-yl)-1,3-thiazole-4-carbonyl]piperidin-4-yl}oxy)methyl]pyridine
1-(4-{4-[3-(3-hydroxypropyl)piperidine-1-carbonyl]phenoxy}piperidin-1-yl)-3-methoxypropan-1-one
N-cyclopentyl-4-(3-methylpyridin-4-yl)-1H-pyrrolo[2,3-b]pyridin-6-amine
N-(1-{1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]piperidin-4-yl}-1H-pyrazol-5-yl)-4-phenylbutanamide
1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-3-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidine
2-(2-{1-ethyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-1H-pyrrol-1-yl)pyridine
5-(2H-1,3-benzodioxol-5-ylmethyl)-5-[3-(7-chloro-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-3-oxopropyl]pyrrolidin-2-one
(2S,4R)-4-amino-1-[3-(1H-indol-3-yl)propanoyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
1-ethyl-4-{[1-(naphthalen-2-yl)-1H-pyrazol-4-yl]methyl}-1,4-diazepane
1-(2-methylphenyl)-4-{1-[2-(methylsulfanyl)pyridine-3-carbonyl]piperidin-3-yl}piperazine
4-(2H-1,3-benzodioxol-5-yl)-3-methyl-1-[2-(4-methyl-1,4-diazepan-1-yl)-2-oxoethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
methyl 6-{[methyl(1,2-oxazol-3-ylmethyl)amino]methyl}-3-(4-methylbenzamido)thieno[2,3-b]pyridine-2-carboxylate
{[2-(ethanesulfonyl)-1-(3-phenylpropyl)-1H-imidazol-5-yl]methyl}(methyl)[(4-methylphenyl)methyl]amine
N-(5-methyl-1,2-oxazol-3-yl)-N'-{[1-(piperidin-1-yl)cyclopentyl]methyl}ethanediamide
N-[4-({4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-1-yl}methyl)phenyl]acetamide
2-(2-fluorophenyl)-N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-N-(2-methylpropyl)acetamide
(1R,3S)-7-[1-(2-fluorophenyl)cyclopropanecarbonyl]-7-azaspiro[3.5]nonane-1,3-diol
(1R,5R)-N,N-dimethyl-6-{[3-(morpholin-4-yl)phenyl]methyl}-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
4-(2-methoxyphenoxy)-1-(3-methylpyrazin-2-yl)piperidine-4-carboxylic acid
7-(2-fluoro-6-methoxybenzoyl)-5H,6H,7H,8H-imidazo[1,5-a]pyrazine
1-methyl-N-[5-oxo-1-(2-phenylethyl)pyrrolidin-3-yl]cyclopropane-1-carboxamide