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(2S,4S)-4-amino-1-[2-(2,5-dimethoxyphenyl)acetyl]-N-ethylpyrrolidine-2-carboxamide
(2S,4S)-1-{[4-(diethylamino)phenyl]methyl}-4-{[(2,5-dimethylphenyl)methyl]amino}-N-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
2-ethoxy-3-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidine-1-carbonyl}pyridine
(2S,4S)-N-[2-(2-methoxyphenyl)ethyl]-1-[(4-phenylphenyl)methyl]-4-(1H-1,2,3,4-tetrazol-1-yl)pyrrolidine-2-carboxamide
N-cycloheptyl-3-{[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]amino}propanamide
N-(1-{7-[(3-fluorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-3-methylbutyl)furan-2-carboxamide
ethyl 1-(dimethyl-1,3-thiazole-5-carbonyl)-3-[(2E)-3-phenylprop-2-en-1-yl]piperidine-3-carboxylate
N-[2-(4-chlorophenyl)ethyl]-3-(2-phenylethyl)-1,2-oxazole-5-carboxamide
N,N-diethyl-1-[(1s,4s)-4-[3-(2H-1,3-benzodioxol-5-yl)propanamido]cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
3-(but-2-yn-1-yl)-5-(2-phenylethyl)-5-(1-{[4-(pyrrolidin-1-yl)phenyl]methyl}piperidin-4-yl)imidazolidine-2,4-dione
3-(5-methylthiophen-2-yl)-N-(3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}propyl)-1H-pyrazole-5-carboxamide
4-[(1R,2R,6S,7S)-4-azatricyclo[5.2.1.02,6]decane-4-carbonyl]-6-(2-methylpropyl)pyrimidin-2-amine
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-6-(4-fluorophenyl)-N-methylimidazo[2,1-b][1,3]thiazole-3-carboxamide
1-[3-(4-fluorophenoxy)azetidin-1-yl]-2-(1-propylpiperidin-4-yl)ethan-1-one
N-(4-methoxyphenyl)-1-(6-methylpyridine-3-carbonyl)piperidin-3-amine
N-[2-(5-methylfuran-2-yl)ethyl]-6-oxo-1-(3-phenylpropyl)piperidine-3-carboxamide
ethyl 3-{[3-(thiophene-2-sulfonamidomethyl)piperidine-1-carbonyl]amino}propanoate
N-(5-chloro-2-methoxyphenyl)-3-[1-(pyridazine-4-carbonyl)piperidin-3-yl]propanamide
8-({3-[2-(1-methyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-1,2-oxazol-5-yl}methoxy)quinoline
N-{1-[2-(azocan-1-yl)-4-methylpyrimidin-5-yl]ethyl}-2-acetamidoacetamide
5-(4-chlorophenyl)-3-(3-methylpiperidin-1-yl)-1,2,4-triazine
[(3R,4R)-4-(azepan-1-ylmethyl)-1-(2,3-dihydro-1H-indene-5-carbonyl)pyrrolidin-3-yl]methanol
(4aS,8aR)-1-[2-(1H-imidazol-4-yl)ethyl]-6-(thiophene-2-carbonyl)-decahydro-1,6-naphthyridin-2-one
1-[2-(4-methoxyphenyl)ethyl]-6-oxo-N-(pyridin-4-ylmethyl)piperidine-3-carboxamide
1-[(1,2-dimethyl-1H-imidazol-5-yl)methyl]-4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-5-one
1-[(3S,4R)-3-(dimethylamino)-4-(4-methoxyphenyl)pyrrolidin-1-yl]-3-(pyridin-3-yl)propan-1-one
(3R)-3-cyclopropyl-4,4-dimethyl-1-(2-methyl-4,5,6,7-tetrahydro-2H-indazole-3-carbonyl)pyrrolidin-3-ol
1-(1-methyl-3-phenyl-1H-pyrazole-5-carbonyl)-4-(4-methylphenoxy)piperidine
N-methyl-N-{[2-(methylamino)pyrimidin-5-yl]methyl}-1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
4-[(2-{4-[(dimethylamino)methyl]phenyl}piperidin-1-yl)methyl]-N-methyl-1,3-thiazol-2-amine
4-(hydroxymethyl)-N-[4-(methylsulfanyl)phenyl]-4-(2-phenoxyethyl)piperidine-1-carboxamide
4-(2-chlorophenoxy)-1-[(1-ethyl-1H-pyrazol-4-yl)methyl]piperidine
2-(4-{[2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-1-yl)pyrimidine
1-[(2-aminopyridin-3-yl)methyl]-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
2-amino-4-(2-methoxypyrimidin-5-yl)-6-(4-methyl-1,3-thiazol-5-yl)pyridine-3-carbonitrile
N-{[2-(azepan-1-yl)-6-methylquinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)furan-2-carboxamide
N-[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]-1-{8-methoxy-5H,6H-benzo[h]quinazolin-2-yl}-5-methyl-1H-pyrazole-4-carboxamide
4-{1-[1-(3-methylpyrazin-2-yl)piperidin-4-yl]piperidine-3-carbonyl}morpholine
4-{[5-(2-ethyl-4-methyl-1,3-oxazol-5-yl)-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-3-yl]methyl}-1-methylpiperidine
1-(2-methoxy-6-{[(prop-2-en-1-yl)(prop-2-yn-1-yl)amino]methyl}phenoxy)-3-(morpholin-4-yl)propan-2-ol
2-(1-benzofuran-2-yl)-6,7-dimethoxyquinazolin-4-amine
(1R,6S)-6-({1-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]piperidin-4-yl}amino)cyclohex-3-ene-1-carboxamide
5-[1-(2-aminoacetyl)pyrrolidin-2-yl]-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]thiophene-2-carboxamide
methyl 4-{3-[(4aR,7aS)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]propanamido}benzoate
4-[3-(pyridin-4-yl)-1H-pyrazole-5-carbonyl]-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
N-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}imidazo[2,1-b][1,3]thiazole-6-carboxamide
4-methyl-N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}-1H-imidazole-2-carboxamide
7-chloro-4-[1-ethyl-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-(3,5-dimethylphenyl)-3-{1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}-3-oxopropanamide
1-benzyl-N3-cyclopropyl-4-oxo-N5-[2,2,2-trifluoro-1-(furan-2-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide