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2-(1-tert-butyl-1H-pyrazol-4-yl)-N,N-diethyl-3,6-dimethylquinoline-4-carboxamide
2-(2-oxo-1,3-oxazolidin-3-yl)-N-{[4-({[3-(trifluoromethyl)phenyl]methyl}amino)quinazolin-2-yl]methyl}acetamide
2-[(3S,4R)-3-(dimethylamino)-4-(4-methylphenyl)pyrrolidin-1-yl]-N-(5-methylpyridin-2-yl)acetamide
2-[9-(3-hydroxy-4-methylbenzoyl)-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl]acetamide
2-(5-chlorothiophen-2-yl)-1-[2-(propan-2-yloxy)ethyl]-1H-imidazole
3-{[3-cyclopropyl-1-(3-methylpyridin-2-yl)-1H-1,2,4-triazol-5-yl]methyl}-2-methyl-1H-indole
(3S,4R)-1-(2-chloro-6-methylbenzenesulfonyl)-N,N-dimethyl-4-(propan-2-yl)pyrrolidin-3-amine
(2S,5R)-1-{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2,5-dimethylpiperazine
{2-oxo-2-[7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decan-2-yl]ethyl}urea
3-methyl-1-(1-methyl-1H-1,2,3-benzotriazol-5-yl)-3-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}urea
N-[(5-methylpyrazin-2-yl)methyl]-5-(pyrrolidin-1-ylmethyl)furan-2-carboxamide
3-(1H-1,3-benzodiazole-2-carbonyl)-7-methyl-3,7,11-triazaspiro[5.6]dodecan-12-one
1-(5-propyl-1,3,4-oxadiazol-2-yl)-4-(pyrrolidine-1-sulfonyl)-1,4-diazepane
(1-{2-[5-(3-methyl-1H-pyrazol-5-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}piperidin-3-yl)methanol
4-(4-chlorophenyl)-N-[2-(6-hydroxy-2-methylpyrimidin-4-yl)ethyl]butanamide
1-(3-fluorophenyl)-3-(1-{1-[3-(1H-pyrazol-1-yl)propanoyl]piperidin-4-yl}-1H-pyrazol-5-yl)urea
1-(5-acetyl-2-ethoxyphenyl)-3-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}urea
1-[6-methyl-5-(5-{[methyl(propan-2-yl)amino]methyl}-1,2,4-oxadiazol-3-yl)-1,2,3,4-tetrahydro-2,7-naphthyridin-2-yl]-2-(methylsulfanyl)ethan-1-one
3-{2-[2-(2-chloro-3,4-dimethoxyphenyl)-1H-imidazol-1-yl]ethyl}-5-methyl-1,2,4-oxadiazole
7-[2-(methylamino)pyridine-3-carbonyl]-2-phenyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-[(3S,5S)-5-(ethylcarbamoyl)-1-[(1-methyl-1H-imidazol-2-yl)methyl]pyrrolidin-3-yl]-4-methyl-1,2,3-thiadiazole-5-carboxamide
2-(1-benzofuran-2-yl)-4-(2,6-dimethylpyridin-3-yl)pyrimidine
2-(1-{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}pyrrolidin-2-yl)-5-fluoro-1H-1,3-benzodiazole
2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]-N-({8-methylimidazo[1,2-a]pyridin-3-yl}methyl)acetamide
7-[3-(2,3-dihydro-1H-isoindol-2-yl)benzoyl]-2,7-diazaspiro[4.4]nonane-1,3-dione
2-methyl-5-({3-[2-(methylsulfanyl)ethyl]-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl}methyl)-1H-1,3-benzodiazole
2-({[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl](methyl)amino}methyl)-3,4-dihydroquinazolin-4-one
2-{[3-(4-ethyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}benzonitrile
[1-(1,5-dimethyl-1H-pyrazol-4-yl)ethyl]({[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl})amine
2-[(4-benzylpiperazin-1-yl)methyl]-N-methyl-N-(3-methylbutyl)-1,3-oxazole-4-carboxamide
{[7-methoxy-2-(thiophen-3-yl)quinolin-3-yl]methyl}(propan-2-yl)amine
(3aS,6aS)-2-ethyl-5-{2-[4-(hydroxymethyl)phenyl]acetyl}-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-[(3,4-dimethoxyphenyl)methyl]-N-(2-methoxyethyl)-1,3-benzoxazole-6-carboxamide
6-fluoro-N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-2-[1-(propan-2-yl)-1H-pyrazol-4-yl]quinoline-4-carboxamide
N-[(3-chloro-1-benzothiophen-2-yl)methyl]-N-methyl-2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetamide
N-[3-(2-methyl-1H-imidazol-1-yl)-1-phenylpropyl]-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
7-acetamido-1-[(4-fluorophenyl)methyl]-N-(oxolan-2-ylmethyl)-N-propyl-1H-1,3-benzodiazole-5-carboxamide
5-{2-[(2-chlorophenyl)methyl]morpholine-4-carbonyl}-2-(propan-2-yl)-3,4-dihydropyrimidin-4-one
2-(4-{[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl)ethan-1-ol
N4-[2-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]morpholine-2,4-dicarboxamide
ethyl 1-{[4-chloro-2-(dimethylamino)-1,3-thiazol-5-yl]methyl}-3-(2-methoxyethyl)piperidine-3-carboxylate
2-tert-butyl-4-hydroxy-N-[3-(pyridin-3-yloxy)propyl]pyrimidine-5-carboxamide
7-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}acetyl)-N,N,2-trimethyl-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
4-(4-fluorophenyl)-1-[3-(1H-1,2,4-triazol-3-yl)benzoyl]-1,2,3,6-tetrahydropyridine
5-{3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-2-methylbenzene-1,3-diol
4-[(2S,4R)-1-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]-4-[(4-fluorophenyl)sulfanyl]pyrrolidine-2-carbonyl]morpholine
N-(2-methoxyethyl)-3-{methyl[2-(pyridin-2-yl)ethyl]sulfamoyl}benzamide
3-[(dimethylamino)methyl]-1-{[3-(4-methoxyphenoxy)phenyl]methyl}pyrrolidin-3-ol
5-[9-hydroxy-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl]-3,4-dihydropyrimidin-4-one
3-{[(2S,5R)-5-({[2-(dimethylamino)ethyl](methyl)amino}methyl)oxolan-2-yl]methyl}-N,N-dimethylbenzamide