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(4aR,7aS)-1-(2-methoxyethyl)-4-(1-methyl-1H-pyrrole-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-(2-methanesulfonylethyl)-5-(propan-2-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
6-(2-hydroxyethyl)-N-[(2E)-3-phenylprop-2-en-1-yl]-N-propylpyrazolo[1,5-a]pyrimidine-2-carboxamide
8-[(2-chloro-6-fluoro-3-methylphenyl)methyl]-2-cyclopropyl-2,8-diazaspiro[5.5]undecan-3-one
3,8-dibenzyl-1-(3-methoxypropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(4-chlorophenyl)-5-methyl-4-[2-(pyridin-3-yl)acetyl]piperazin-2-one
1-(7-{[4-(benzyloxy)piperidin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-4-(1H-1,2,4-triazol-1-yl)butan-1-one
1-(4-fluorobenzoyl)-4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine
N-(isoquinolin-5-ylmethyl)-N,4-dimethyl-2-(propan-2-yl)pyrimidine-5-carboxamide
N-[4-(1-ethyl-1H-1,2,4-triazol-5-yl)-7-methoxy-2-oxo-1,2,3,4-tetrahydroquinolin-6-yl]methanesulfonamide
1-benzyl-4-[2-(2-hydroxyethoxy)ethyl]-1,4-diazepan-6-ol
2-amino-4-methyl-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-1,3-benzothiazole-6-carboxamide
methyl 2-(5-{1-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]piperidin-4-yl}-1H-pyrazol-3-yl)acetate
6-(1,4-oxazepan-4-yl)-N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}pyridine-3-carboxamide
6-[(1R,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-9H-purine
2-{[1-(4-ethoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1,3-thiazole
(1S,9aR)-1-{[4-(2,6-dimethylpyridin-4-yl)piperazin-1-yl]methyl}-octahydro-1H-quinolizine
2-(2H-1,3-benzodioxol-5-yl)-N-[1-(5-{[(2-fluorophenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)-2-phenylethyl]acetamide
N-({1-[(2-butyl-1H-imidazol-4-yl)methyl]piperidin-3-yl}methyl)-2-(2-methoxyphenoxy)acetamide
2-[1-(4-chlorophenyl)-5-oxo-3-propyl-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-(propan-2-yl)acetamide
N-cyclopentyl-3-(4-hydroxyphenyl)-N-[(2-methylphenyl)methyl]-1H-pyrazole-5-carboxamide
N-butyl-2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
4-cyclobutyl-6-methyl-2-[3-(1H-pyrazol-1-yl)azetidin-1-yl]pyrimidine
1-(pyrrolidin-1-yl)-3-{1-[(2,3,6-trifluorophenyl)methyl]piperidin-3-yl}propan-1-one
3-[methyl({[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]methyl})amino]-1λ6-thiolane-1,1-dione
(4aR,7aS)-1-(1H-imidazol-2-ylmethyl)-4-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-cyclopropyl-1-(4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)ethan-1-one
(2S,4S)-1-[(2E)-3-phenylprop-2-en-1-yl]-4-({[4-(propan-2-yl)phenyl]methyl}amino)-N-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
2-[2-(1-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}piperidin-3-yl)-1H-imidazol-1-yl]acetamide
N-methyl-4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}benzamide
(3R,5S)-5-[4-(4-fluorophenoxy)piperidine-1-carbonyl]pyrrolidin-3-ol
2-{[5-(4-phenylazepane-1-carbonyl)pyridin-2-yl]amino}ethan-1-ol
3-{5-[(methylsulfanyl)methyl]-3-(oxan-4-yl)-1H-1,2,4-triazol-1-yl}pyridine
4-methyl-N-[2-(3-phenylpyrrolidin-1-yl)ethyl]-1,2,3-thiadiazole-5-carboxamide
N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]-2-(3-oxo-2,3-dihydro-1,2-benzothiazol-2-yl)acetamide
2-{[4-(2-chlorophenyl)-5-(2-methylpropyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-6-oxo-1-(3-phenylpropyl)piperidine-3-carboxamide
N-benzyl-N-methyl-3-{1-[2-(pyridin-2-ylsulfanyl)acetyl]piperidin-4-yl}propanamide
8-(2,1,3-benzoxadiazol-4-ylmethyl)-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
1-(carbamoylmethyl)-N-[(4-methyl-1H-1,3-benzodiazol-2-yl)methyl]piperidine-4-carboxamide
1-cyclopentyl-N-[4-(3-methoxyphenyl)phenyl]piperidine-3-carboxamide
methyl[(4-{[4-(propan-2-yloxy)phenyl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)methyl][2-(pyridin-2-yl)ethyl]amine
N-[(3S,4R)-4-(5-methylfuran-2-yl)-1-{2-methylthieno[3,2-d]pyrimidin-4-yl}pyrrolidin-3-yl]acetamide
1-[2-(4-methyl-1,2,5-oxadiazol-3-yl)pyrrolidin-1-yl]-2-(2-phenyl-1H-imidazol-1-yl)ethan-1-one
N-(pyridin-3-ylmethyl)-N-(thiophen-3-ylmethyl)-3-(4H-1,2,4-triazol-4-yl)benzamide
3-[({[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}amino)methyl]piperidin-3-ol
7-chloro-4-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}quinoline
1-(4-acetyl-1,4-diazepan-1-yl)-3-(4-chlorophenyl)-3-phenylpropan-1-one
N-(2-methyl-1-{7-[(3,4,5-trimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}propyl)furan-3-carboxamide
[(3R,4S)-1-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol