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3-[({1-[4-(1H-pyrazol-3-yl)benzoyl]piperidin-4-yl}oxy)methyl]pyridine
4-[(2,6-difluorophenyl)methyl]-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N,5-dimethyl-N-[(3-methylpyridin-2-yl)methyl]pyrazine-2-carboxamide
5-cyclopropanecarbonyl-1'-(2,6-dimethylpyrimidine-4-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-[2-({4-[2-oxo-2-(piperidin-1-yl)ethyl]piperazin-1-yl}methyl)phenoxy]acetic acid
N-[3-(1H-indazol-1-yl)propyl]-7-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
4-(2-{[1-(4-methylpyrimidin-2-yl)piperidin-4-yl]amino}ethyl)benzene-1-sulfonamide
1-[2-(4-methoxyphenyl)ethyl]-N-methyl-6-oxo-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
3-(4,6-dimethoxypyrimidin-2-yl)-3,9-diazaspiro[5.6]dodecan-10-one
2-(2,1,3-benzoxadiazole-4-sulfonyl)-2,7-diazaspiro[4.5]decane
cyclohexyl[4-(furan-3-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methanol
2-(4-chlorophenyl)-4-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)morpholine
2-(3-{[(2S)-2-(hydroxymethyl)pyrrolidin-1-yl]methyl}phenyl)-6-(2-methyl-1,3-thiazol-4-yl)-3,4-dihydropyrimidin-4-one
4-({2-[1-(butane-1-sulfonyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
N-{2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}-4-(pyridin-4-yl)pyrimidin-2-amine
N,8-dimethyl-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}imidazo[1,2-a]pyridine-2-carboxamide
2-methanesulfonyl-N-methyl-N-[3-(pyrrolidin-1-yl)butyl]acetamide
1-(2-{4-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]piperazin-1-yl}ethyl)-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
N-(4-fluoro-3-{[methyl(oxan-2-ylmethyl)carbamoyl]amino}phenyl)propanamide
8-(1H-indol-3-ylmethyl)-1-(2-methylpropyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[7-(hydroxymethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
N-(4-fluoro-2-methylphenyl)-3-[1-(4-methylbenzoyl)piperidin-3-yl]propanamide
2-({[(3R,4R)-1-(2-chloro-5-fluorobenzoyl)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
1-cyclohexyl-4-(1-methyl-1H-pyrazole-5-carbonyl)-1,4-diazepan-6-ol
N-[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]-1,3-dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
2-({8-methyl-2,8-diazaspiro[4.5]decan-2-yl}sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
(1R,5S,6R)-N-(furan-2-ylmethyl)-3-(quinolin-4-ylmethyl)-3-azabicyclo[3.1.0]hexane-6-carboxamide
[(2-chlorophenyl)methyl]({[2-cyclopropylmethanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl})methylamine
N-{[5-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-3-yl]methyl}-5-ethyl-1,3,4-oxadiazol-2-amine
N-cyclopropyl-3-(6,7-dimethyl-1H-1,3-benzodiazol-2-yl)-N-[(2-methoxyphenyl)methyl]propanamide
2-[(oxolan-2-ylmethyl)(propyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
4-[5-(5-ethoxyfuran-2-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carbonyl]morpholine
N-[2-(3,6-dioxo-1,2,3,6-tetrahydropyridazin-1-yl)ethyl]-1-[(4-methylphenyl)amino]cyclopentane-1-carboxamide
methyl 2-{5-methyl-2-[(oxolan-3-ylformamido)methyl]-2,3-dihydro-1-benzofuran-7-yl}benzoate
N-[(3R,4R)-1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-3-hydroxypiperidin-4-yl]pyridine-2-carboxamide
3-(4,5-dimethyl-1H-pyrazol-3-yl)-1-[3-(2-phenylacetyl)piperidin-1-yl]propan-1-one
3-[(3S,7S,8aS)-3-[(4-methoxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(3-chloro-4-methylphenyl)urea
1-{3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-(1H-indazol-1-yl)ethan-1-one
1-cyclopentyl-3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]piperidine
[3-({cyclopropyl[(1-methyl-1H-imidazol-2-yl)methyl]amino}methyl)-2,4,6-trimethylphenyl]methanol
3-(methylsulfanyl)-1-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
2-(2-phenyl-1H-imidazol-1-yl)-1-[4-(pyridin-3-ylmethoxy)piperidin-1-yl]ethan-1-one
2-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-N-ethylpyrimidin-4-amine
1-(2-methylphenyl)-4-[2-(pyrrolidin-1-yl)acetyl]piperazin-2-one
4-[(3-chloro-4-hydroxyphenyl)methyl]-1-(4-methoxyphenyl)-3-methylpiperazin-2-one
N'-[(1R)-2-hydroxy-1-phenylethyl]-N-(2,4,6-trimethylphenyl)butanediamide
3-methoxy-N-methyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}pyrazin-2-amine
2-[(4-methoxyphenyl)methyl]-N-[1-(pyridin-3-yl)propan-2-yl]-1,3-benzoxazole-6-carboxamide
5-ethyl-4-(pyrrolidin-1-ylmethyl)-N-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]furan-2-carboxamide
N-(2,2-dimethyloxan-4-yl)-N-ethyl-5-(phenoxymethyl)-1H-pyrazole-3-carboxamide