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N-methyl-N-{3-[2-(oxolan-3-yl)-1H-imidazol-1-yl]propyl}aniline
N-methyl-N-[1-(pyridin-3-yl)propyl]imidazo[2,1-b][1,3]thiazole-6-carboxamide
ethyl 4-({[3-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]methyl}amino)piperidine-1-carboxylate
5-(2-methoxyacetamido)-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-1-(2-phenylethyl)-1H-1,3-benzodiazole-7-carboxamide
1-butyl-3-cyclopropyl-5-[(1R,2R)-2-phenylcyclopropyl]-1H-1,2,4-triazole
(3S,4R)-3-cyclopropyl-4-[2-(2,4-dimethyl-6-oxo-1,6-dihydropyrimidin-5-yl)acetamido]-N,N-dimethylpyrrolidine-1-carboxamide
({5-[1-(2,1,3-benzoxadiazol-4-ylmethyl)piperidin-3-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
(2S,3R)-2-{[5-(3-acetylphenoxymethyl)-1H-pyrazol-3-yl]formamido}-3-hydroxybutanamide
N-[3-(1H-indol-1-yl)propyl]-3-{5-[2-(4-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}propanamide
2-(2-{[3-hydroxy-3-(hydroxymethyl)pyrrolidin-1-yl]methyl}phenoxy)-1-(piperidin-1-yl)ethan-1-one
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-4-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butanamide
3-[3-(naphthalen-1-yl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl]propanoic acid
N-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
3-[4-(2,4-difluorophenyl)-1H-pyrazol-5-yl]-1-[(2,3-difluorophenyl)methyl]piperidine
N-({5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl}methyl)furan-2-carboxamide
6-methoxy-3-({3-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}methyl)-1H-indazole
2-phenyl-1-(1-{pyrazolo[1,5-a]pyrimidine-3-carbonyl}piperidin-3-yl)ethan-1-one
N-[2-(1H-imidazol-1-yl)-1-phenylethyl]-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide
N-[(3R,4R)-4-hydroxypyrrolidin-3-yl]-2-(4-propanoylphenoxy)acetamide
N-({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N,1-dimethyl-1H-pyrazole-5-carboxamide
4-(3-chlorobenzoyl)-1-(3-chlorophenyl)piperazin-2-one
6-[(2-fluorophenyl)methoxy]-4-(furan-2-carbonyl)-1-[(4-methoxyphenyl)methyl]-1,4-diazepan-2-one
6-(2,8-dimethylquinoline-4-carbonyl)-2-methyl-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
N-[(5-methoxy-1,3-benzoxazol-2-yl)methyl]-3-(4-methyl-1,3-thiazol-5-yl)propanamide
1-cyclohexyl-5-[5-(methoxymethyl)furan-2-yl]-1H,4H-pyrazolo[3,4-d]imidazole
1-cyclohexyl-N3-cyclopropyl-N5-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
4-[(3-acetylphenyl)methyl]-1-[(4-methylphenyl)methyl]piperazin-2-one
1-(4,6-dimethylpyrimidin-2-yl)-N-{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}piperidin-4-amine
4-[3-cyclopropyl-5-(2,3-dihydro-1-benzofuran-2-yl)-1H-1,2,4-triazol-1-yl]-2-methylpyridine
3-(6-oxo-1,4,5,6-tetrahydropyridazin-3-yl)-N-[1-(2-phenylethyl)piperidin-3-yl]propanamide
N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-amine
4-[2-(1H-1,3-benzodiazol-1-yl)propanoyl]-1-(4-methylphenyl)piperazin-2-one
1-[4-(4-fluorophenyl)-1,2,3,6-tetrahydropyridin-1-yl]-4-(1H-pyrazol-4-yl)butan-1-one
N-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-N,5,6-trimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
5-[9-hydroxy-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl]-1-methyl-1,2-dihydropyridin-2-one
4'-(2-methoxyethyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
6-{[(2-aminopyrimidin-5-yl)methyl](methyl)amino}-N-[3-(pyridin-2-yl)propyl]pyridine-3-carboxamide
3-butyl-1-methyl-4-(pyridin-4-ylmethyl)piperazin-2-one
4-(2-{4-[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]-1H-1,2,3-triazol-1-yl}ethyl)morpholine
2-methyl-6-{1-[3-(1H-pyrazol-1-yl)benzoyl]piperidin-4-yl}pyrimidin-4-ol
2-[1-(cyclohexylmethyl)-4-[(1-methyl-1H-pyrazol-4-yl)methyl]piperazin-2-yl]ethan-1-ol
3-[3-(4-phenoxybenzoyl)piperidine-1-carbonyl]pyridine
N,1-dimethyl-N-{2-phenyl-1-[1-(quinoxaline-6-carbonyl)piperidin-4-yl]ethyl}-1H-pyrazole-3-carboxamide
N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
(1S,5R)-6-(3,5-dimethyl-1-benzofuran-2-carbonyl)-3-methyl-3,6-diazabicyclo[3.2.2]nonane
N-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]acetamide
N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}-2-(2,5,7-trimethyl-1H-indol-3-yl)acetamide
1-(1-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-yl)-3-(pyrrolidine-1-carbonyl)piperidine
N-({1-[2-(1H-imidazol-4-yl)acetyl]piperidin-3-yl}methyl)-4-phenylbenzamide
(4aR,8aR)-4a-hydroxy-N,N-dimethyl-7-(quinoxaline-6-carbonyl)-decahydro-2,7-naphthyridine-2-carboxamide