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1-[4-(dimethylamino)-5-methylpyrimidin-2-yl]-4-phenylpiperidine-4-carbonitrile
2-(2-fluoro-4-methylphenyl)-2-{methyl[2-(4-methyl-1,3-thiazol-5-yl)ethyl]amino}acetic acid
3-(2-chlorophenyl)-1-cyclopentyl-3-{2-[3-(4-fluorophenyl)pyrrolidin-1-yl]-2-oxoethyl}pyrrolidine-2,5-dione
methyl 3-{[(2R,3R)-2-ethoxy-3-propanamido-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]carbonyl}benzoate
1-{4-[4-(3-hydroxypiperidine-1-carbonyl)phenoxy]piperidin-1-yl}-3-methoxypropan-1-one
9-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
4-(pyridin-2-yl)-N-{2-[2-(pyridin-3-yl)-1,3-thiazol-4-yl]ethyl}pyrimidin-2-amine
2-{2-[3-(2-methoxybenzoyl)piperidin-1-yl]-2-oxoethyl}-2,3-dihydro-1H-isoindole-1,3-dione
N-benzyl-2-[2-(2-methylpropyl)-3-oxo-2,8-diazaspiro[4.5]decan-8-yl]propanamide
2-{4-[1-(3-chloropyridin-2-yl)piperidin-4-yl]piperazin-1-yl}ethan-1-ol
N-[4-(difluoromethoxy)-2-methylphenyl]-4-methyl-1,2,3,6-tetrahydropyridine-1-carboxamide
2-[(4-benzylpiperazin-1-yl)methyl]-N-[4-(1H-pyrazol-1-yl)butan-2-yl]-1,3-oxazole-4-carboxamide
{[3-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-5-yl]methyl}(methyl)[2-(pyridin-2-yl)ethyl]amine
(2S)-2-{[6-(2-aminoethyl)pyrimidin-4-yl]amino}-3-methylbutan-1-ol
1-{2-[4-(quinolin-2-yl)-1H-1,2,3-triazol-1-yl]ethyl}piperidine-3-carboxamide
2-(4-fluoro-2-methylphenyl)-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]acetamide
2-{1-[5-(2-methoxyphenoxymethyl)-1H-pyrazol-3-yl]-N-methylformamido}-N,2-dimethylpropanamide
(2S)-1-[2-(2,6-dimethoxyphenoxy)ethyl]-2-(pyrrolidin-1-ylmethyl)pyrrolidine
N-[4-(4-{[2-(morpholin-4-yl)ethyl]amino}piperidin-1-yl)phenyl]benzenesulfonamide
N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}-5-(oxolan-2-yl)thiophene-2-carboxamide
9-(propane-2-sulfonyl)-3,9-diazaspiro[5.6]dodecane
3-(3-chlorobenzoyl)-1-(3-methylthiophene-2-carbonyl)piperidine
N-[(3S,5S)-5-(diethylcarbamoyl)-1-methylpyrrolidin-3-yl]-1-methyl-1H-1,3-benzodiazole-5-carboxamide
7-(1H-1,3-benzodiazole-5-carbonyl)-2-(pyridin-2-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
4-hydroxy-N-[(5-methylpyrazin-2-yl)methyl]-2-(pyridin-2-yl)pyrimidine-5-carboxamide
ethyl 1-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-3-[(2-fluorophenyl)methyl]piperidine-3-carboxylate
8-{[2,5-dimethoxy-4-(methylsulfanyl)phenyl]methyl}-3-ethyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-ethyl-4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)-N-(2,2,2-trifluoroethyl)benzamide
4-({3-[5-(2-methylpropyl)-1H-1,2,4-triazol-3-yl]phenyl}methyl)morpholine
5-(2,4-difluorophenoxymethyl)-N-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-N-methyl-1,2-oxazole-3-carboxamide
2-cyano-N-{2-[4-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)morpholin-2-yl]ethyl}benzene-1-sulfonamide
4-hydroxy-1-methyl-N-[1-(5,6,7,8-tetrahydronaphthalen-2-yl)ethyl]piperidine-4-carboxamide
N'-cyclooctyl-N-(1-methoxybutan-2-yl)butanediamide
9-[1-(2-hydroxyethyl)-1H-1,3-benzodiazol-2-yl]-1-oxa-9-azaspiro[5.5]undecan-5-ol
2-phenyl-1-[4-(pyridin-4-ylmethyl)-1,8-dioxa-4,11-diazaspiro[5.6]dodecan-11-yl]ethan-1-one
5-ethyl-N-({2-[4-(2-methylphenyl)piperazin-1-yl]pyridin-3-yl}methyl)pyrimidin-2-amine
2-[(3R,4S)-4-(dimethylamino)-3-(3-hydroxypropyl)piperidine-1-carbonyl]-5-methylphenol
3-(1H-imidazol-2-ylmethyl)-9-methoxy-N-[(2-methoxyphenyl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
3-(furan-2-yl)-N-{1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl}propanamide
2-{3-[(pyridin-2-ylmethyl)carbamoyl]piperazin-1-yl}-1,3-oxazole-4-carboxylic acid
1-{[(3-hydroxy-2-oxo-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-3-yl)methyl]amino}cyclopentane-1-carboxamide
1-(2-{4-[1-(2-methylphenyl)-1H-pyrazol-4-yl]-1,2,3,6-tetrahydropyridin-1-yl}ethyl)pyrrolidin-2-one
1-[(1R,3S)-1-hydroxy-3-(2-hydroxyethoxy)-7-azaspiro[3.5]nonan-7-yl]-2-(1,3-thiazol-4-yl)ethan-1-one
1-({5-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-ylmethyl]-1,2,4-oxadiazol-3-yl}methyl)-4-methylpiperazine
3-methyl-2-{4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine
1-{[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-ol
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-5-(pyrrolidin-2-yl)thiophene-2-carboxamide
(3S,4S)-4-(pyridin-2-yl)-1-{thieno[2,3-d]pyrimidin-4-yl}pyrrolidine-3-carboxylic acid
ethyl 2-[(2-{[(3-phenyl-1H-pyrazol-4-yl)methyl]carbamoyl}phenyl)amino]acetate
N-[2-(2-amino-1,3-thiazol-4-yl)ethyl]-2,6,8-trimethylquinoline-4-carboxamide