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1-{[3-(furan-2-yl)phenyl]methyl}-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
2-(2-{[(3R,4R)-4-cyclopropyl-4-hydroxy-3-methylpiperidin-1-yl]methyl}phenoxy)acetic acid
2,5-dimethoxy-N-({4-[(3-phenylpropyl)amino]quinazolin-2-yl}methyl)benzene-1-sulfonamide
N-propyl-7-[(pyridin-3-yl)sulfamoyl]-1,2,3,4-tetrahydroisoquinoline-2-carboxamide
N-[2-(dimethylamino)-2-(4-fluorophenyl)ethyl]-3-(3-hydroxy-3-methylbutyl)benzamide
1-[(4-fluorophenyl)methyl]-N-[1-(2-methoxyphenyl)propan-2-yl]-N-methyl-1H-1,2,3-triazole-4-carboxamide
1-{6-[3-(morpholin-4-ylmethyl)phenyl]-1,2,3,4-tetrahydroquinolin-1-yl}ethan-1-one
3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-N-propylpiperidine-1-carboxamide
(2S,4R)-4-(5-methoxyfuran-2-amido)-N-methyl-1-[(3-methylthiophen-2-yl)methyl]pyrrolidine-2-carboxamide
(3R,4S)-1-(6,7-diethoxy-3-methyl-1-benzofuran-2-carbonyl)-3,4-dimethylpiperidin-4-ol
2-(2-aminoacetyl)-N-[(4-chlorophenyl)methyl]-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
5-(4-hydroxy-1-{[2-(prop-2-en-1-yloxy)phenyl]methyl}piperidin-4-yl)-N-(pyridin-2-ylmethyl)-1-benzofuran-2-carboxamide
1-methyl-3-[5-(4-methylphenyl)-1,3,4-thiadiazol-2-yl]-1-[(2-methylphenyl)methyl]urea
N,2,7-trimethyl-N-[1-(pyridin-3-yl)propyl]imidazo[1,2-a]pyridine-3-carboxamide
2-(dimethylamino)-2-(4-fluorophenyl)-N-[1-(morpholin-4-ylmethyl)cyclopentyl]acetamide
1-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}-4-[(2-methyl-1H-imidazol-1-yl)methyl]piperidine
2-methanesulfonyl-N-(pentan-3-yl)-N-(2-phenylethyl)acetamide
4-[1-(1-{5-methyl-1-[4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carbonyl}piperidin-4-yl)ethyl]morpholine
5-{[2-(2-chlorophenyl)ethyl]amino}-N,N-dimethyl-1-(2-methylpropyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
5-(2-chloro-4-methoxyphenoxymethyl)-N-(1H-imidazol-2-ylmethyl)-N-methyl-1,2-oxazole-3-carboxamide
3-({[(4-chlorophenyl)(phenyl)methyl]amino}methyl)-7-fluoro-1-methyl-1,2-dihydroquinolin-2-one
6-chloro-N-(2-hydroxyethyl)-N-[(2-methoxyphenyl)methyl]-2-methylquinoline-4-carboxamide
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-1-[(3-methoxyphenyl)methyl]-6-oxopiperidine-3-carboxamide
3-(3,4-dimethyl-1H-pyrazol-5-yl)-1-[2-(naphthalen-1-ylmethyl)morpholin-4-yl]propan-1-one
2-methyl-2-phenyl-N-{2-[4-(pyrimidin-2-yl)piperazin-1-yl]ethyl}propanamide
N-(4,6-dimethylpyridin-2-yl)-4-({methyl[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]amino}methyl)benzamide
3-phenyl-N-{[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl}-1H-pyrazole-4-carboxamide
1-{[3-(2,5-dimethylthiophen-3-yl)-1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}-4-ethylpiperazine
2-(3,5-dimethyl-4-phenyl-1H-pyrazol-1-yl)-N-(1-phenyl-1H-pyrazol-5-yl)acetamide
7-fluoro-N-[2-(morpholin-4-yl)ethyl]-2-oxo-1,2-dihydroquinoline-4-carboxamide
(3S,4S)-1-{[2-(methylamino)-1,3-thiazol-4-yl]methyl}-4-(pyridin-2-yl)pyrrolidine-3-carboxylic acid
N-[2-(dimethylamino)ethyl]-4-(thiophen-3-yl)-1H-pyrrolo[2,3-b]pyridin-6-amine
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-{[2-(morpholin-4-yl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}furan-2-carboxamide
6-[(3-methoxyphenyl)methoxy]-1-(2-methylpropyl)-4-[3-(1H-1,2,4-triazol-1-yl)propanoyl]-1,4-diazepan-2-one
N-(2-{[3-(3-acetylphenyl)-1-methyl-2-oxo-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-6-yl]methyl}quinolin-6-yl)acetamide
N-tert-butyl-2-methyl-3-({[1-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]carbamoyl}amino)benzamide
1-(4-cyclopentyl-1,4-diazepan-1-yl)-3-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]propan-1-one
1-[2-(1H-pyrazol-1-ylmethyl)pyrrolidin-1-yl]-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propan-1-one
1-ethyl-N-[(1-ethyl-1H-indazol-3-yl)methyl]-6-oxopiperidine-3-carboxamide
2-[5-(3,4-difluorophenyl)-1H-indazol-1-yl]-N-(1,3-dimethyl-1H-pyrazol-5-yl)acetamide
1-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-3-(1-methyl-1H-imidazol-2-yl)piperidine
4-{[7-chloro-2-(2-methoxyphenyl)quinolin-3-yl]methyl}piperazin-2-one
3-(dimethyl-1,2-oxazol-4-yl)-N-[2-(pyridin-2-ylsulfanyl)ethyl]propanamide
2-[5-(4-ethyl-2-methyl-1,3-thiazol-5-yl)-3-[(1-methylpiperidin-4-yl)methyl]-1H-1,2,4-triazol-1-yl]acetic acid
4-{5-[(6-methyl-2H-1,3-benzodioxol-5-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonyl}morpholine
3,3-dimethyl-1-[(5-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl)methyl]urea
methyl({[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}){[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}amine
2-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}-1,2,3,4-tetrahydroisoquinolin-4-ol
N,2-dimethyl-N-{2-phenyl-1-[1-(4,5,6,7-tetrahydro-2H-indazole-3-carbonyl)piperidin-4-yl]ethyl}furan-3-carboxamide
N-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-1-ethyl-5-oxopyrrolidine-3-carboxamide