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Darifenacin hydrobromide_Molecular_structure_CAS_133099-07-7)
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Darifenacin hydrobromide

Catalog No. Bio-0941 Name InterBioScreen
CAS Number 133099-07-7 Website http://www.ibscreen.com
M. F. C28H31BrN2O2 Telephone +7 49652 40091
M. W. 507.46194 Fax
Purity Email screen@ibscreen.chg.ru
Storage Chembase ID: 165412

SYNONYMS

IUPAC name
2-[(3S)-1-[2-(2,3-dihydro-1-benzofuran-5-yl)ethyl]pyrrolidin-3-yl]-2,2-diphenylacetamide hydrobromide
IUPAC Traditional name
2-[(3S)-1-[2-(2,3-dihydro-1-benzofuran-5-yl)ethyl]pyrrolidin-3-yl]-2,2-diphenylacetamide hydrobromide
Synonyms
Emselex
Enablex

DATABASE IDS

CAS Number 133099-07-7

PROPERTIES

Application(s) Used to treat urinary incontinence
Salt Data HBr
Mechanism of Action Works by blocking the M3 muscarinic acetylcholine receptor, which is primarily responsible for bladder muscle contractions

DETAILS

REFERENCES

  • Liver Physiol. 2010 Jul;299(1):G215-9. Epub 2010 Apr 15.
  • 3. Jha S, Parsons M: Treatment of overactive bladder in the aging population: focus on darifenacin. Clin Interv Aging. 2006;1(4):309-16.
  • 1. Bharucha AE, Ravi K, Zinsmeister AR: Comparison of selective M3 and nonselective muscarinic receptor antagonists on gastrointestinal transit and bowel habits in humans. Am J Physiol Gastrointest
  • 2. Bozkurt TE, Sahin-Erdemli I: M(1) and M(3) muscarinic receptors are involved in the release of urinary bladder-derived relaxant factor. Pharmacol Res. 2009 May;59(5):300-5. Epub 2009 Feb 5.