Sulfamethoxypyridazine

• Catalog No.: Bio-0764
• CAS Number: 80-35-3
• M. F.: C11H12N4O3S
• M. W.: 280.30298

SYNONYMS

• IUPAC name: 4-amino-N-(6-methoxypyridazin-3-yl)benzene-1-sulfonamide
• IUPAC Traditional name: 4-amino-N-(6-methoxypyridazin-3-yl)benzene-1-sulfonamide
• Synonyms: Lederkyn; Kynex; Sulfalex; Midicel; Sulphamethoxypyridazine; Exazol

DATABASE IDS

• CAS Number: 80-35-3

PROPERTIES

• Application(s): Antiseptic
• Application(s): Long-acting sulfonamide used for treatment of systemic infections.
• Application(s): Low acute toxicity
• Mechanism of Action: Dihydrofolate reductase inhibitor
• Mechanism of Action: Folate antagonist

REFERENCES

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• Kracmar, J. et al., Pharmazie, 1975, 30, 447, (uv)
• Grechishkin, V.S. et al., J. Mol. Struct., 1982, 83, 345, (nqr, nmr)
• Bult, A., Pharm. Weekbl., Sci. Ed., 1983, 5, 77, (cmr)
• Basak, A.K. et al., Acta Cryst. C, 1987, 43, 735, (cryst struct)
• Negwer, M., Organic-Chemical Drugs and their Synonyms, 6th edn., Akademie-Verlag, 1987, 1932; 2752
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• Martindale, The Extra Pharmacopoeia, 30th edn., Pharmaceutical Press, 1993, 210
• Lewis, R.J., Sax's Dangerous Properties of Industrial Materials, 8th edn., Van Nostrand Reinhold, 1992, AKO500