Sulpiride

• Catalog No.: Bio-0717
• CAS Number: 15676-16-1
• M. F.: C15H23N3O4S
• M. W.: 341.42582

SYNONYMS

• IUPAC name: N-[(1-ethylpyrrolidin-2-yl)methyl]-2-methoxy-5-sulfamoylbenzamide
• IUPAC Traditional name: N-[(1-ethylpyrrolidin-2-yl)methyl]-2-methoxy-5-sulfamoylbenzamide
• Synonyms: Milsulvan; Mirbanil; Dogmatil; Dogmatyl; Eglonyl

DATABASE IDS

• CAS Number: 15676-16-1

PROPERTIES

• Application(s): Low acute toxicity
• Application(s): Antidepressant
• Application(s): Digestive aid
• Application(s): Antianxiety drug
• Application(s): Non-sedative major antipsychotic agent
• Application(s): Migraine therapeutic
• Mechanism of Action: Dopamine D2-receptor antagonist
• Mechanism of Action: In contrast to most other neuroleptics which block both dopamine D1 and D2 receptors, Sulpiride is more selective and acts primarily as a dopamine D2 antagonist
• Mechanism of Action: Sulpiride appears to lack effects on norepinephrine, acetylcholine, serotonin, histamine, or gamma-aminobutyric acid (GABA) receptors

REFERENCES

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