Eprosartan

• Catalog No.: Bio-0035
• CAS Number: 133040-01-4
• M. F.: C23H24N2O4S
• M. W.: 424.51266

SYNONYMS

• IUPAC name: 4-({2-butyl-5-[(1E)-2-carboxy-2-(thiophen-2-ylmethyl)eth-1-en-1-yl]-1H-imidazol-1-yl}methyl)benzoic acid
• IUPAC Traditional name: 4-({2-butyl-5-[(1E)-2-carboxy-2-(thiophen-2-ylmethyl)eth-1-en-1-yl]-1H-imidazol-1-yl}methyl)benzoic acid
• Synonyms: Teveten

DATABASE IDS

• CAS Number: 133040-01-4

PROPERTIES

• Application(s): Antihypertensive agent
• Mechanism of Action: Angiotensin II AT 1 -receptor antagonist

REFERENCES

• Eur. Pat., 1990, SmithKline Beckman, 403 159; CA, 114, 207258h, (synth, pharmacol)
• Weinstock, J. et al., J. Med. Chem., 1991, 34, 1514; 1993, 36, 1880, (synth, pharmacol, pmr)
• Edwards, R.M. et al., J. Pharmacol. Exp. Ther., 1992, 260, 175, (pharmacol)
• Wittenberger, S.J. et al., Synth. Commun., 1993, 23, 3231, (synth, pmr, cmr)
• McLellan, K.J. et al., Drugs, 1998, 55, 713-718, (rev)
• Plosker, G.L. et al., Drugs, 2000, 60, 177-201, (rev)