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2-[1-(2-methylpropyl)-4-(quinolin-5-ylmethyl)piperazin-2-yl]ethan-1-ol
3-(2-ethyl-1H-imidazol-1-yl)-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}propanamide
dimethyl({[4-(trimethylpyrimidin-4-yl)phenyl]methyl})amine
2-{1-[(2-chloro-4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[3-(propan-2-yloxy)propyl]acetamide
ethyl 3-[(2,4-difluorophenyl)methyl]-1-(2-methyl-1,3-thiazole-4-carbonyl)piperidine-3-carboxylate
ethyl 3-[(3-methoxyphenyl)methyl]-1-[3-(1,2-oxazolidin-2-yl)propanoyl]piperidine-3-carboxylate
5-methyl-1-(4-methylphenyl)-4-[2-(1H-1,2,4-triazol-3-yl)benzoyl]piperazin-2-one
1-methyl-4-{[6-(3-methylphenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}-1,4-diazepane
3-(piperidin-1-ylmethyl)-4-propyl-4,5-dihydro-1H-1,2,4-triazol-5-one
1-{4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-(methylsulfanyl)ethan-1-one
2-[(2-fluorophenyl)methyl]-N-[2-(pyridin-2-yl)ethyl]-1,3-benzoxazole-6-carboxamide
8-[2-(4-fluorophenyl)-2-hydroxyacetyl]-3-(3-methylbutyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-(6-methyl-2-propylpyrimidin-4-yl)-N-[1-(1,3-thiazol-2-yl)ethyl]piperidin-4-amine
1-{5-methanesulfonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
4-(hydroxymethyl)-4-(2-phenoxyethyl)-N-[4-(trifluoromethyl)phenyl]piperidine-1-carboxamide
2-{1-[(2,3-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-ethyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]acetamide
N-[4-(furan-2-yl)butan-2-yl]-4-(trifluoromethyl)pyrimidin-2-amine
7-methyl-3-[(4-methylpiperidin-1-yl)methyl]-1-(pyridin-2-ylmethyl)-1,2-dihydroquinolin-2-one
N-butyl-2-{1-[(4-methoxy-3-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
N-{3-oxo-3-[3-(4-phenyl-1H-pyrazol-5-yl)piperidin-1-yl]propyl}methanesulfonamide
4-(4-chlorophenoxy)-1-(4-methylpyrimidin-2-yl)piperidine-4-carboxylic acid
N-[2-(6,7-dimethyl-1H-1,3-benzodiazol-2-yl)ethyl]-1-(propan-2-yl)piperidine-4-carboxamide
1-(2-methoxyethyl)-3-[(3-methoxyphenyl)methyl]-8-[(2-methyl-1H-imidazol-4-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-{2-[(3R,4R)-4-ethyl-3,4-dihydroxypiperidin-1-yl]-2-oxoethyl}-5,6-dimethyl-2,3-dihydropyridazin-3-one
(9aR)-8-(4-chlorobenzoyl)-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-[2-(furan-2-yl)-2-(pyrrolidin-1-yl)ethyl]-2-(3-methylthiophen-2-yl)-1H-imidazole
2-amino-3-ethyl-N-[2-(3-methylthiophen-2-yl)ethyl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
N-{[7-(2,3-difluorobenzoyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-2-(thiophen-2-yl)acetamide
2-{4-[(4-ethylpiperazin-1-yl)methyl]phenyl}-5,6-dimethyl-3,4-dihydropyrimidin-4-one
(1R,5R)-N,N-dimethyl-6-[3-(1H-pyrazol-1-ylmethyl)benzoyl]-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
2-(2,3-dihydro-1,4-benzodioxin-2-yl)-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-[3-(dimethylamino)propyl]-N-methyl-7-(pyridine-3-carbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
(1R,5S,6S)-6-{[4-(2-methylphenyl)-1,4-diazepan-1-yl]methyl}-3-azabicyclo[3.1.0]hexane
2-[3-cyclopentyl-5-(oxolan-3-yl)-1H-1,2,4-triazol-1-yl]ethan-1-ol
3-(2-methyl-1H-imidazol-1-yl)-1-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
N-[1-(3-methoxyphenyl)ethyl]-7-oxo-7H-[1,3]thiazolo[3,2-a]pyrimidine-5-carboxamide
(2S,4S)-1-[(3-chloro-5-fluoro-4-methoxyphenyl)methyl]-4-acetamido-N-ethylpyrrolidine-2-carboxamide
7-[2-(3-phenylpyrrolidin-1-yl)acetyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-cyclopropanecarbonyl-8-[2-(pyridin-3-yl)acetyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-chloro-4-{[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepan-1-yl]methyl}phenol
N-{5H,6H,7H-cyclopenta[d]pyrimidin-2-ylmethyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
2-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[(3,5-difluorophenyl)methyl]-5-methoxybenzamide
2-[(3S,4R)-4-amino-1-(3,5-dimethyl-1H-indole-2-carbonyl)pyrrolidin-3-yl]ethan-1-ol
4-({2-[1-(furan-2-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
3-{[(4-fluorophenyl)methyl]sulfanyl}-N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}propanamide
methyl 4-{[2-(4-fluorophenyl)pyrrolidin-1-yl]methyl}-1H-pyrazole-3-carboxylate
2-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-2,3-dihydro-1,2-benzothiazol-3-one
(4S)-1-{[2-(benzylamino)pyrimidin-5-yl]methyl}-3,3,4-trimethylpiperidin-4-ol
5-[(1S,5R)-3-acetyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1-methyl-1,2-dihydropyridin-2-one
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-(2-oxopyrrolidin-1-yl)acetamide