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N-(3-fluoro-2-methylphenyl)-2-{[(3S,4R)-4-methoxyoxolan-3-yl]amino}acetamide
3-fluoro-N-{1-[1-(2-methoxy-2-methylpropanoyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
N-[(3R,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2,4,5-trifluorobenzamide
2-({6-[2-(aminomethyl)-4-fluorophenyl]quinazolin-4-yl}amino)ethan-1-ol
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-2-[(2-ethyl-6-methylpyridin-3-yl)oxy]acetamide
5-{[benzyl(methyl)amino]methyl}-N-[2-(1H-imidazol-1-yl)ethyl]-1,2-oxazole-3-carboxamide
8-{[5-methyl-2-(naphthalen-2-yl)-1,3-oxazol-4-yl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
3,7-dimethyl-11-(4-methylnaphthalene-1-carbonyl)-3,7,11-triazaspiro[5.6]dodecane
2-methyl-5-[3-(pyridin-4-yl)azetidine-1-carbonyl]pyrazine
N-[(5-{[3-(methylsulfanyl)phenyl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl)methyl]cyclobutanecarboxamide
6-methyl-3-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-ylmethyl}-4H-chromen-4-one
1-[(3-methoxyphenyl)methyl]-N-[(3-methylpyridin-4-yl)methyl]-6-oxopiperidine-3-carboxamide
(2S,3R)-2-[(2,7-dimethylquinolin-4-yl)formamido]-3-hydroxybutanamide
N-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]-1-methyl-2-(morpholin-4-yl)-1H-1,3-benzodiazole-5-carboxamide
N-[(1-benzylpyrrolidin-3-yl)methyl]-6-(morpholin-4-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
N-[(3-propyl-1,2-oxazol-5-yl)methyl]-6-(5,6,7,8-tetrahydro-1,6-naphthyridin-6-yl)pyridine-3-carboxamide
2-({[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}(propan-2-yl)amino)ethan-1-ol
1-(1-ethyl-3-methyl-1H-pyrazole-5-carbonyl)-4-[(2-methylphenyl)sulfanyl]piperidine
4-{[3-(5-methylfuran-2-yl)phenyl]methyl}morpholine-2-carboxamide
2-{4-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]piperidin-1-yl}-7-methanesulfonyl-4-methylquinazoline
3-(4-hydroxyphenyl)-N-{[1-(2-methoxyethyl)pyrrolidin-3-yl]methyl}-1H-pyrazole-5-carboxamide
1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
3-(carbamoylamino)-N-{5H,6H,7H,8H,9H,10H,11H-cycloocta[b]indol-2-ylmethyl}propanamide
N-[(3S,5S)-5-(diethylcarbamoyl)-1-(1H-imidazol-2-ylmethyl)pyrrolidin-3-yl]pyridine-3-carboxamide
7-methoxy-1-methyl-N-(1-propyl-1H-1,3-benzodiazol-5-yl)-1,2,3,4-tetrahydroisoquinoline-2-carboxamide
5-(2-methoxyacetamido)-1-methyl-2-(pyridin-4-yl)-N-{spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-5-ylmethyl}-1H-1,3-benzodiazole-7-carboxamide
5-(hydroxymethyl)-2-methyl-4-{[2-(4-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]methyl}pyridin-3-ol
4-(2,1,3-benzoxadiazol-5-ylmethyl)-1-[(3,5-dimethylphenyl)methyl]piperazin-2-one
3-{1-[6-(trifluoromethyl)pyridin-3-yl]-1H-1,3-benzodiazol-2-yl}propanoic acid
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
1-(carbamoylmethyl)-N-{[5-(thiophen-2-yl)-1H-pyrazol-4-yl]methyl}piperidine-3-carboxamide
5-[3-(methoxymethyl)piperidine-1-carbonyl]-N-methyl-N-(3-methylbutyl)pyridin-2-amine
1,3-dimethyl-4-{6-methyl-2-[1-(propan-2-yl)-1H-pyrazol-4-yl]quinoline-4-carbonyl}piperazin-2-one
2-(pyridin-4-ylmethyl)-8-{thieno[3,2-d]pyrimidin-4-yl}-2,8-diazaspiro[5.5]undecan-3-one
2-chloro-N-[(3R,4S)-4-cyclopropyl-1-methylpyrrolidin-3-yl]-4-fluorobenzamide
4-(4-{4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}piperidin-1-yl)-5-propylpyrimidine
4-methyl-3-oxo-N-{[3-(thiophen-2-yl)-1H-pyrazol-4-yl]methyl}-3,4-dihydroquinoxaline-2-carboxamide
N-[3-(5-amino-1,3,4-thiadiazol-2-yl)propyl]-2-(2,3-dihydro-1H-inden-1-yl)acetamide
3-(3,5-dimethyl-1H-pyrazol-4-yl)-2-methoxyquinoline
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-N,3-dimethylthiophene-2-sulfonamide
3-[1-(cyclopent-1-ene-1-carbonyl)piperidin-3-yl]-N-methyl-N-[2-(pyridin-2-yl)ethyl]propanamide
N-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]-3-(3-fluorophenyl)-N-methyl-1H-pyrazole-4-carboxamide
5-[5-(piperidine-1-carbonyl)furan-2-yl]-1,2,3,4-tetrahydroisoquinoline
4-[2-(3-{[2-(4-fluorophenyl)azetidin-1-yl]methyl}phenoxy)ethyl]morpholine
4-(pyrimidin-2-yl)-2-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}phenol
N-{4-[2-(3-cyanophenyl)-1H-imidazol-1-yl]-2-methylphenyl}butanamide
3-(5-{2-[3-(oxolan-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}-1,2,4-oxadiazol-3-yl)pyridine
3-ethyl-8-(5-methyl-2,3-dihydro-1H-indole-2-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(3R,5S)-5-{4-[4-(2-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}pyrrolidin-3-ol
1-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]-3,3-diphenylpiperidine